Affinity DataIC50: 398nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+5nMAssay Description:Antagonist activity at rat KOR expressed in CHOK1 cells assessed as inhibition of U50488-induced increase in cAMP accumulation measured after 10 mins...More data for this Ligand-Target Pair
Affinity DataEC50: <7.94E+3nMAssay Description:Agonist activity at rat KOR expressed in CHOK1 cells assessed as increase in cAMP accumulation measured after 10 mins by HTRF assayMore data for this Ligand-Target Pair