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Found 2 Enz. Inhib. hit(s) with Target = 'Sterol regulatory element-binding protein 2' and Ligand = 'BDBM78179'
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed