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Found 156 with Last Name = 'kamisuki' and Initial = 's'
TargetDNA polymerase beta(Rattus norvegicus)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50448689(CHEMBL3127730)
Affinity DataKi:  5.50E+3nMAssay Description:Competitive inhibition of recombinant rat DNA polymerase beta using poly(dA)/oligo(dT)18 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50448689(CHEMBL3127730)
Affinity DataKi:  1.16E+4nMAssay Description:Noncompetitive inhibition of recombinant rat DNA polymerase beta using dTTP as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223758(CHEMBL58925)
Affinity DataIC50:  1nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223748(CHEMBL406322)
Affinity DataIC50:  4nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223740(CHEMBL431679)
Affinity DataIC50:  5nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223762(CHEMBL417588)
Affinity DataIC50:  6nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223756(CHEMBL333710)
Affinity DataIC50:  14nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223759(CHEMBL118469)
Affinity DataIC50:  37nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223754(CHEMBL332885)
Affinity DataIC50:  38nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223738(CHEMBL118450)
Affinity DataIC50:  47nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223737(CHEMBL115852)
Affinity DataIC50:  57nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha subunit B(Bos taurus (bovine))
Kyoto Prefectural University

LigandPNGBDBM33388(dehydroaltenusin derivative, 16)
Affinity DataIC50:  60nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223757(CHEMBL291976)
Affinity DataIC50:  71nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha subunit B(Bos taurus (bovine))
Kyoto Prefectural University

LigandPNGBDBM33387(dehydroaltenusin derivative, 15)
Affinity DataIC50:  90nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223753(CHEMBL119059)
Affinity DataIC50:  140nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223749(CHEMBL332977)
Affinity DataIC50:  150nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha subunit B(Bos taurus (bovine))
Kyoto Prefectural University

LigandPNGBDBM33386(dehydroaltenusin derivative, 14)
Affinity DataIC50:  180nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223750(CHEMBL119731)
Affinity DataIC50:  190nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223739(CHEMBL117056)
Affinity DataIC50:  210nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha subunit B(Bos taurus (bovine))
Kyoto Prefectural University

LigandPNGBDBM33389(dehydroaltenusin derivative, 20)
Affinity DataIC50:  240nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM20182((1S,2R,5S,10S,11S,14R,15R)-14-[(2R)-6-hydroxy-6-me...)
Affinity DataIC50:  300nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha subunit B(Bos taurus (bovine))
Kyoto Prefectural University

LigandPNGBDBM33384(dehydroaltenusin)
Affinity DataIC50:  680nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351538(CHEMBL1824673)
Affinity DataIC50:  700nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223741(CHEMBL333173)
Affinity DataIC50:  720nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha subunit B(Bos taurus (bovine))
Kyoto Prefectural University

LigandPNGBDBM33385(desmethyldehydroaltenusin, 2)
Affinity DataIC50:  890nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351539(CHEMBL1824674)
Affinity DataIC50:  900nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351538(CHEMBL1824673)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223751(CHEMBL119353)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351541(CHEMBL1824676)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351540(CHEMBL1824675)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223760(CHEMBL332071)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223763(CHEMBL261984)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223764(CHEMBL119757)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223755(CHEMBL118108)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223765(CHEMBL420538)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351534(CHEMBL1824669)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351535(CHEMBL1824670)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351529(CHEMBL1824664)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351536(CHEMBL1824671)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351521(CHEMBL1824658)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351537(CHEMBL1824672)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351542(CHEMBL1824661)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351533(CHEMBL1824668)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351531(CHEMBL1824666)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351530(CHEMBL1824665)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351526(CHEMBL1616869)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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