Compile Data Set for Download or QSAR
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Found 220 with Last Name = 'figler' and Initial = 'h'
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317873((2R,3R,4S,5R)-2-(6-(2-hydroxy-1,1,3,3-tetramethyli...)
Affinity DataKi:  0.790nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317893(CHEMBL1095001 | N6-[4-(4-(3,5-Di-tert-butyl-4-hydr...)
Affinity DataKi:  2.22nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317887(CHEMBL1094995 | N6-[4-[2-[3,5-di-tert-butylbenzami...)
Affinity DataKi:  2.25nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317888(CHEMBL1094996 | N6-[4-[2-[3,4,5-Trimethoxybenzamid...)
Affinity DataKi:  4.26nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317892(CHEMBL1095000 | N6-[4-[2-[3,4,5-Trimethoxybenzamid...)
Affinity DataKi:  5.04nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317890(CHEMBL1094998 | N6-[4-[2-[3,5-Di-tert-butyl-4-hydr...)
Affinity DataKi:  5.63nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50292320(CHEMBL400746 | N-(4-(9-((2R,3R,4S,5R)-3,4-dihydrox...)
Affinity DataKi:  7nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50292320(CHEMBL400746 | N-(4-(9-((2R,3R,4S,5R)-3,4-dihydrox...)
Affinity DataKi:  7nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  7.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317885(CHEMBL1098715 | N6-(3,5-Di-tert-butyl-4-hydroxyphe...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317891(CHEMBL1094999 | N6-[4-[2-[3,5-Di-tert-butylbenzami...)
Affinity DataKi:  9.02nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM81971(1,3-Diethyl-8-phenyl-3,7-dihydro-purine-2,6-dione ...)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50219389(3,5-di-tert-butyl-N-(6-(9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  14nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50292321(CHEMBL249677 | N6-[6-[1,1,3,3-tetramethylisoindoli...)
Affinity DataKi:  15nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM82558(CAS_163889 | CHEMBL355370 | I-ABOPX | NSC_163889)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317889(CHEMBL1094997 | N6-[4-[2-[1,1,3,3-Tetramethylisoin...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317888(CHEMBL1094996 | N6-[4-[2-[3,4,5-Trimethoxybenzamid...)
Affinity DataKi:  26.2nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317878(CHEMBL1098520 | N6-(4-(2-Aminoethyl)-2,6-di-tert-b...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82558(CAS_163889 | CHEMBL355370 | I-ABOPX | NSC_163889)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50219387(3,5-di-tert-butyl-N-(2-{4-[9-((2R,3R,4S,5R)-3,4-di...)
Affinity DataKi:  32nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82558(CAS_163889 | CHEMBL355370 | I-ABOPX | NSC_163889)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50219389(3,5-di-tert-butyl-N-(6-(9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  40nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317893(CHEMBL1095001 | N6-[4-(4-(3,5-Di-tert-butyl-4-hydr...)
Affinity DataKi:  42.1nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317886(CHEMBL1094994 | N6-[4-[2-[3,5-Di-tert-butyl-4-hydr...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50292322((2R,3R,4S,5R)-2-(6-((1-hydroxy-2,2,5,5-tetramethyl...)
Affinity DataKi:  50nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317876((2R,3R,4S,5R)-2-(6-(1-hydroxy-2,2,6,6-tetramethylp...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50292322((2R,3R,4S,5R)-2-(6-((1-hydroxy-2,2,5,5-tetramethyl...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50292322((2R,3R,4S,5R)-2-(6-((1-hydroxy-2,2,5,5-tetramethyl...)
Affinity DataKi:  50nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50292319(CHEMBL250316 | N6-(2,2,6,6-tetramethylpiperidin-1-...)
Affinity DataKi:  50nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
Affinity DataKi:  51.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317889(CHEMBL1094997 | N6-[4-[2-[1,1,3,3-Tetramethylisoin...)
Affinity DataKi:  53.1nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50317880(CHEMBL1099126 | N6-(1,1,3,3-Tetramethylisoindolin-...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM82558(CAS_163889 | CHEMBL355370 | I-ABOPX | NSC_163889)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317892(CHEMBL1095000 | N6-[4-[2-[3,4,5-Trimethoxybenzamid...)
Affinity DataKi:  76.8nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50219387(3,5-di-tert-butyl-N-(2-{4-[9-((2R,3R,4S,5R)-3,4-di...)
Affinity DataKi:  84nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50292321(CHEMBL249677 | N6-[6-[1,1,3,3-tetramethylisoindoli...)
Affinity DataKi:  89nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82558(CAS_163889 | CHEMBL355370 | I-ABOPX | NSC_163889)
Affinity DataKi:  95nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317873((2R,3R,4S,5R)-2-(6-(2-hydroxy-1,1,3,3-tetramethyli...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50292323(CHEMBL400567 | N6-(1,1,3,3-tetramethylisoindolin-2...)
Affinity DataKi:  100nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317890(CHEMBL1094998 | N6-[4-[2-[3,5-Di-tert-butyl-4-hydr...)
Affinity DataKi:  105nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317891(CHEMBL1094999 | N6-[4-[2-[3,5-Di-tert-butylbenzami...)
Affinity DataKi:  128nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317878(CHEMBL1098520 | N6-(4-(2-Aminoethyl)-2,6-di-tert-b...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  156nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50292320(CHEMBL400746 | N-(4-(9-((2R,3R,4S,5R)-3,4-dihydrox...)
Affinity DataKi:  230nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50317886(CHEMBL1094994 | N6-[4-[2-[3,5-Di-tert-butyl-4-hydr...)
Affinity DataKi:  243nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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