Compile Data Set for Download or QSAR
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Found 42 of affinity data for UniProtKB/TrEMBL: P30987
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM10042((5Z)-7-[(1R,4S,5R,6R)-6-[(1E,3S)-3-hydroxyoct-1-en...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82224(CAS_188200 | ICI 79939 | NSC_188200)
Affinity DataKi:  320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82225(11,9-epoxymethano PGH2)
Affinity DataKi:  360nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82226(9,11-ethano PGH2)
Affinity DataKi:  440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82222(CAS_5311388 | EP045 | NSC_5311388)
Affinity DataKi:  460nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50090136((Z)-7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((E)-(R)-3-hy...)
Affinity DataKi:  770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM81949(9,11-AzoPGH2 | 9,11-azo PGH2 | J389.306E | PGH2, 9...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82220(EP011)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82229(CAS_57576-52-0 | TXA2)
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82223(CAS_71111-01-8 | PTA2)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82228(CAS_74034-56-3 | CTA2)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM10042((5Z)-7-[(1R,4S,5R,6R)-6-[(1E,3S)-3-hydroxyoct-1-en...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50020300((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-oct-1-enyl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM35847((15S)-prostaglandin E2 | (5Z,11alpha,13E,15S)-11,1...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50101828(7-[(1R,2R,3R)-3-Hydroxy-2-((E)-(R)-3-hydroxy-oct-1...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82213(CAS_41598-07-6 | NSC_114678 | PGD2)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82221(10alpha,11alpha-oxido PGA2)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM22319((5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoic acid | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM82227(15-methyl PGF2alpha | CAS_37255 | NSC_37255)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353639(CHEMBL1829806)
Affinity DataIC50:  3.10nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353632(CHEMBL1829812)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353635(CHEMBL1829801)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353643(CHEMBL1829808)
Affinity DataIC50:  9.40nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353645(CHEMBL1829810)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353640(CHEMBL65121)
Affinity DataIC50:  27nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353638(CHEMBL1829805)
Affinity DataIC50:  52nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353636(CHEMBL1829802)
Affinity DataIC50:  91nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353646(CHEMBL1829811)
Affinity DataIC50:  259nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353644(CHEMBL1829809)
Affinity DataIC50:  463nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353641(CHEMBL1829804)
Affinity DataIC50:  1.23E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353634(CHEMBL1828642)
Affinity DataIC50:  1.63E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353642(CHEMBL1829807)
Affinity DataIC50:  1.79E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353633(CHEMBL1829813)
Affinity DataIC50:  2.52E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353637(CHEMBL1829803)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353634(CHEMBL1828642)
Affinity DataKd:  1.00E+4nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353639(CHEMBL1829806)
Affinity DataKd:  26nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353638(CHEMBL1829805)
Affinity DataKd:  11nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353640(CHEMBL65121)
Affinity DataKd:  26nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353637(CHEMBL1829803)
Affinity DataKd:  1.20E+3nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353636(CHEMBL1829802)
Affinity DataKd:  17nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University of Edinburgh

Curated by PDSP Ki Database
LigandPNGBDBM50353635(CHEMBL1829801)
Affinity DataKd:  19nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed