BDBM50001309 (cyclo-[L-propyl-D-phenylalanyl-L-isoleucyl-D-dehydropiperazyl-L-dehydropiperazyl-D(N-methyl)phenylalanyl])(L-365,209)::CHEMBL127686::L-365209
SMILES CC[C@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H]2CCCN2C(=O)[C@@H](Cc2ccccc2)N(C)C(=O)[C@@H]2CCC=NN2C(=O)[C@H]2CCC=NN2C1=O
InChI Key InChIKey=IFHSSGUGRIXWQU-NSTWBPGMSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50001309
Affinity DataKi: 7.30nMAssay Description:Binding affinity towards rat uterine receptor was determined using [3H]oxytocin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Compound was evaluated for OT receptor affinity by displacement of [3H]OT from binding sites in uterine tissue taken from nonlabor pregnant womenMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of [3H]arginine vasopressin binding to rat kidney medulla Vasopressin V2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Inhibition of [3H]arginine vasopressin binding to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 820nMAssay Description:Binding affinity towards rat kidney V2 receptor was determined using [3H]arginine vasopressin as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of [3H]arginine vasopressin binding to AVP-V2 site in rat kidney medulla.More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Concentration required to displace 50% of [3H]oxytocin from rat uterine receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Concentration required to displace 50% of [3H]arginine vasopressin from rat liver arginine vasopressin 1A (AVP-V1a) site.More data for this Ligand-Target Pair