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Patent: (prefix with "US" like US6078908)
PatentDataPatent TitleOrganizationDepositionDownloads
US9549932 488 2-(morpholin-4-yl)-1,7-naphthyridines Bayer Pharma Aktiengesellschaft 11/29/182D 3D TSV
US9718828 489 BTK Inhibitors MERCK SHARP & DOHME CORP.; MERCK SHARP & DOHME B.V. 11/29/182D 3D TSV
US9550771 93 Keto-imidazopyridine derivatives as RORc modulators Genentech, Inc. 11/29/182D 3D TSV
US9718822 68 Macrocyclic compounds as Trk kinase inhibitors Array BioPharma, Inc. 11/29/182D 3D TSV
US9718854 20 Selective glycosidase inhibitors and uses thereof Alectos Therapeutics Inc.; Merck Sharp & Dohme Corp. 11/29/182D 3D TSV
US9718820 90 Substituted aza-bicyclic imidazole derivatives useful TRPM8 receptor modulators JANSSEN PHARMACEUTICA NV 11/29/182D 3D TSV
US9550775 130 Substituted triazolopyridines and methods of use thereof GENENTECH, INC.; XENON PHARMACEUTICALS INC. 11/29/182D 3D TSV
US9718814 375 Cyclopropanamine compound and use thereof Takeda Pharmaceutical Company Limited 11/28/182D 3D TSV
US9718819 182 Non-nucleoside reverse transcriptase inhibitors Merck Sharp & Dohme Corp. 11/28/182D 3D TSV
US9718812 213 Substituted thiazole or oxazole P2X7 receptor antagonists Axxam S.P.A. 11/28/182D 3D TSV
US9718809 87 Bisarylsulfonamides useful in the treatment of inflammation and cancer Kancera AB 11/27/182D 3D TSV
US9718800 115 Chromenone derivatives ASTRAZENECA AB 11/27/182D 3D TSV
US9718808 144 Inhibitors of the renal outer medullary potassium channel Merck Sharp & Dohme Corp. 11/27/182D 3D TSV
US9718793 138 Isoxazole compounds as inhibitors of heat shock proteins Vernalis (R&D) Ltd.; Cancer Research Technology Limited; The Institute of Cancer Research 11/27/182D 3D TSV
US9718792 101 Isoxazoline hydroxamic acid derivatives as LpxC inhibitors Novartis AG 11/27/182D 3D TSV
US9718790 2250 Triazine derivative and pharmaceutical composition having an analgesic activity comprising the same SHIONOGI & CO., LTD. 11/27/182D 3D TSV
US9718803 375 Unsaturated nitrogen heterocyclic compounds useful as PDE10 inhibitors Amgen Inc. 11/27/182D 3D TSV
US9718771 48 Aniline derivative, pharmaceutical composition containing same, and use thereof KISSEI PHARMACEUTICAL CO., LTD. 11/16/182D 3D TSV
US9718787 9 Poly (ADP-ribose) polymerase inhibitor CHENGDU DIAO PHARMACEUTICAL GROUP CO., LTD. 11/16/182D 3D TSV
US9718780 6 Substituted pyridines as sodium channel blockers TBA 11/16/182D 3D TSV
US9714242 13 Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists Bayer Intellectual Property GmbH 11/15/182D 3D TSV
US9714234 70 Carbazole carboxamide compounds Bristol-Myers Squibb Company 11/15/182D 3D TSV
US9713651 56 Compositions, methods, and systems for the synthesis and use of imaging agents Lantheus Medical Imaging, Inc. 11/15/182D 3D TSV
US9714236 207 Compounds and methods for inhibiting JAK ASTRAZENECA AB 11/15/182D 3D TSV
US9713612 30 Compounds for treatment of cancer CUREGENIX, INC. 11/15/182D 3D TSV
US9714252 7 Cyclic sulfonamides as sodium channel blockers Purdue Pharma L.P. 11/15/182D 3D TSV
US9714241 375 Cyclopropanamine compound and use thereof Takeda Pharmaceutical Company Limited 11/15/182D 3D TSV
US9714266 46 Estra-1,3,5(10),16-tetraene-3-carboxamides for inhibition of 17.beta.-hydroxysteroid dehydrogenase (AKR1C3) BAYER PHARMA AKTIENGESELLSCHAFT 11/15/182D 3D TSV
US9714224 8 Heterocyclic compounds and methods of their use NOVARTIS AG 11/15/182D 3D TSV
US9714230 511 Histone demethylase inhibitors Celgene Quantical Research, Inc. 11/15/182D 3D TSV
US9713606 584 Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C Boehringer Ingelheim International GmbH 11/15/182D 3D TSV
US9714247 452 Multiple kinase pathway inhibitors Tolero Pharmaceuticals, Inc.; Mannkind Corporation 11/15/182D 3D TSV
US9717745 5 Pharmaceutical compositions and their use for treatment of cancer and autoimmune diseases ZHEJIANG DTRM BIOPHARMA CO. LTD. 11/15/182D 3D TSV
US9718760 257 Plasminogen activator inhibitor-1 inhibitors and methods of use thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY 11/15/182D 3D TSV
US9714249 134 Pyrazolo-pyrrolidin-4-one derivatives and their use in the treatment of disease Novartis AG 11/15/182D 3D TSV
US9714235 40 Quinazoline derivatives, compositions thereof, and use as pharmaceuticals Shanghai Fochon Pharmaceutical Co., Ltd. 11/15/182D 3D TSV
US9717714 14 Spirocyclic CETP inhibitors Merck Sharp & Dohme Corp. 11/15/182D 3D TSV
US9714221 654 Substituted 6,7-dihydro-5H-benzo[7]annulene compounds, processes for their preparation and therapeutic uses thereof SANOFI 11/15/182D 3D TSV
US9714232 72 Substituted piperazine compounds and methods of use thereof SUNSHINE LAKE PHARMA CO., LTD. 11/15/182D 3D TSV
US9714244 46 Substituted pyrido[4,3-d]pyrimidines as Wee-1 inhibitors ALMAC DISCOVERY LIMITED 11/15/182D 3D TSV
US9556130 73 4-oxo-3,4-dihydro-1,2,3-benzotriazine modulators of GPR139 Takeda Pharmaceutical Company Limited 11/08/182D 3D TSV
US9550741 612 Benzoisothiazole compounds and methods of treating schizophrenia Shanghai Institute of Pharmaceutical Industry 11/08/182D 3D TSV
US9556150 59 Inhibitors of bruton's tyrosine kinase Hoffmann-La Roche Inc.; Chugai Pharmaceutical Co. 11/08/182D 3D TSV
US9708370 88 Azapeptides as CD36 binding compounds VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP 11/07/182D 3D TSV
US9546162 91 Compounds and methods for skin repair ALLERGAN, INC. 11/07/182D 3D TSV
US9533987 230 Heterocyclic derivates Kalvista Pharmaceuticals Limited 11/07/182D 3D TSV
US9546164 648 Substituted benzamides and methods of use thereof GENENTECH, INC.; XENON PHARMACEUTICALS INC. 11/07/182D 3D TSV
US9708337 36 Aryl amide-based kinase inhibitors Bristol-Myers Squibb Company 11/05/182D 3D TSV
US9708336 2511 Metallo-beta-lactamase inhibitors Merck Sharp & Dohme Corp. 11/05/182D 3D TSV
US9708359 143 Pyrrolopyrimidine nucleosides and analogs thereof Chimerix, Inc.; The Regents of the University of Michigan 11/05/182D 3D TSV
US9708340 96 Urea derivatives and their use as fatty-acid binding protein (FABP) inhibitors Hoffmann-La Roche Inc. 11/05/182D 3D TSV
US9708333 86 Fused bicyclic 1,2,4-triazine compounds as TAM inhibitors Incyte Corporation 11/01/182D 3D TSV
US9708309 24 Arylcyclopropylamine based demethylase inhibitors of LSD1 and their medical use ORYZON GENOMICS, S.A. 10/31/182D 3D TSV
US9708311 143 Benzimidazole derivatives as EP4 antagonists BAYER PHARMA AKTIENGESELLSCHAFT 10/31/182D 3D TSV
US9708318 856 Bicyclic heterocycles as FGFR4 inhibitors Incyte Corporation 10/31/182D 3D TSV
US9708302 46 Flouro-naphthyl derivatives HOFFMANN-LA-ROCHE INC. 10/31/182D 3D TSV
US9708313 142 Substituted pyrido[3,4-b]pyrazines as GPR6 modulators Takeda Pharmaceutical Company Limited 10/31/182D 3D TSV
US9708325 62 Sulfonimidoylpurinone compounds and derivatives for the treatment and prophylaxis of virus infection Hoffmann-La Roche Inc. 10/31/182D 3D TSV
US9708279 100 2-acylaminothiazoles for the treatment of cancer UNIVERSITÁ DEGLI STUDI DI MILANO—BICOCCA; UNIVERSITÈ DE GENÈVE; UNIVERSITÈ CLAUDE BERNARD LYON 1 10/30/182D 3D TSV
US10053471 17 Azabenzimidazole derivatives Boehringer Ingelheim International GmbH 10/30/182D 3D TSV
US9708266 40 Cyclohexyl pyridine derivative KISSEI PHARMACEUTICAL CO., LTD. 10/30/182D 3D TSV
US9708253 135 Cyclohexyl sulfone RORγ modulators Bristol-Myers Squibb Company 10/30/182D 3D TSV
US9701672 77 Dihydropyridinone MGAT2 inhibitors for use in the treatment of metabolic disorders Bristol-Myers Squibb Company 10/30/182D 3D TSV
US9708275 12 Heterocyclic compounds and methods for their use NOVARTIS AG 10/30/182D 3D TSV
US9707233 368 Heterocyclylamines as PI3K inhibitors Incyte Holdings Corporation; Incyte Corporation 10/30/182D 3D TSV
US9708272 22 Inhibitors of α-amino-β-carboxymuconic acid semialdehyde decarboxylase TES Pharma S.r.l. 10/30/182D 3D TSV
US9700563 3 Kappa opioid receptor compounds MediSynergies, LLC 10/30/182D 3D TSV
US10053462 195 P2X7 modulators Janssen Pharmaceutica NV 10/30/182D 3D TSV
US9701669 34 Preparation and use of 7a-amide substituted- 6,6-difluoro bicyclic himbacine derivatives as PAR-1 receptor antagonists Merck Sharp & Dohme Corp. 10/30/182D 3D TSV
US9708269 7 Process for making isoquinoline compounds FibroGen, Inc. 10/30/182D 3D TSV
US9701670 374 Pyrazolyl-ureas as kinase inhibitors RESPIVERT LIMITED; TOPIVERT PHARMA LIMITED 10/30/182D 3D TSV
US10053465 286 Pyrrolopyrimidine derivatives as TAM inhibitors Incyte Corporation 10/30/182D 3D TSV
US9708268 42 ROR modulators and their uses INNOV17 LLC 10/30/182D 3D TSV
US9707205 16 S1P receptors modulators and their use thereof AKAAL PHARMA PTY LTD. 10/30/182D 3D TSV
US9701693 4 Selective glycosidase inhibitors and uses thereof Alectos Therapeutics Inc.; Merck Sharp & Dohme Corp. 10/30/182D 3D TSV
US9701685 18 Spiropyrrolidines as MDM2 inhibitors Hudson Biopharma Inc. 10/30/182D 3D TSV
US9708295 51 Substituted 2-aminopyridine protein kinase inhibitor CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD.; Centaurus Biopharma Co., Ltd.; LIANYUNGANG RUNZHONG PHARMACEUTICAL CO., LTD. 10/30/182D 3D TSV
US10053463 422 Substituted [1,2,4]triazolo[4,3-a]pyrazines as P2X7 modulators Janssen Pharmaceutica NV 10/30/182D 3D TSV
US9708270 91 Substituted spiropiperidinyl compounds useful as GPR120 agonists Merck Sharp & Dohme Corp. 10/30/182D 3D TSV
US9701663 37 Sulfonamide retinoic acid receptor-related orphan receptor modulators and uses thereof INNOV17 LLC 10/30/182D 3D TSV
US9708274 328 Sulfoximine substituted quinazolines for pharmaceutical compositions EVOTEC INTERNATIONAL GMBH 10/30/182D 3D TSV
US10053461 41 Tetracyclic 4-oxo-pyridine-3-carboxylic acid derivatives for the treatment and prophylaxis of hepatitis B virus infection Hoffmann-La Roche Inc. 10/30/182D 3D TSV
US9701638 16 Therapeutic hydroxyquinolones Rutgers, The State University of New Jersey 10/30/182D 3D TSV
US9701691 25 Thienopyrimidine compounds Hoffman-La Roche Inc. 10/30/182D 3D TSV
US9550763 437 Heterocyclic ring and carbocyclic derivative SHIONOGI & CO., LTD. 10/19/182D 3D TSV
US9546173 190 Substituted pyrrolo[3,4-d]pyrimidines as kinase inhibitors Novartis AG 10/19/182D 3D TSV
US10053433 20 Androgen receptor antagonists The Regents of the University of California 10/18/182D 3D TSV
US10053454 88 Carbazole compounds useful as bromodomain inhibitors Bristol-Myers Squibb Company 10/18/182D 3D TSV
US10053456 375 Cyclopropanamine compound and use thereof Takeda Pharmaceutical Company Limited 10/18/182D 3D TSV
US10053455 22 Diazaspiroalkaneone-substituted oxazole derivatives as spleen tyrosine kinase inhibitors AB SCIENCE 10/18/182D 3D TSV
US10053434 24 Histone deacetylase inhibitors and compositions and methods of use thereof CHDI FOUNDATION, INC. 10/18/182D 3D TSV
US10053458 216 Pyrimidine-2,4-diamine derivative and anticancer pharmaceutical composition comprising same as effective ingredient KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY 10/18/182D 3D TSV
US10053431 514 Tetrahydro-benzodiazepinones Hoffmann-La Roche Inc. 10/18/182D 3D TSV
US9556139 260 6-substituted phenoxychroman carboxylic acid derivatives Array BioPharma Inc. 10/17/182D 3D TSV
US9556135 339 Amino-dihydrothiazine and amino-dioxido dihydrothiazine compounds as beta-secretase antagonists and methods of use Amgen, Inc. 10/17/182D 3D TSV
US10047118 7 C17-aryl substituted betulinic acid analogs ViiV HEALTHCARE UK (NO.5) LIMITED 10/17/182D 3D TSV
US10047086 158 Imidazopyridines and imidazopyrazines as LSD1 inhibitors Incyte Corporation 10/17/182D 3D TSV
US9556143 18 Metalloenzyme inhibitor compounds Viamet Pharmaceuticals, Inc. 10/17/182D 3D TSV
US9556168 60 N-alkylated indole and indazole compounds as RORgammaT inhibitors and uses thereof Merck Sharp & Dohme Corp. 10/17/182D 3D TSV
US9556148 86 N-cyanomethylamides as inhibitors of janus kinase Cadila Healthcare Limited 10/17/182D 3D TSV
US10052306 333 Selective octahydro-cyclopenta[C] pyrrole negative modulators of NR2B CADENT THERAPEUTICS, INC. 10/17/182D 3D TSV
US9555024 35 Substituted (E)-N′-(1-phenylethylidene)benzohydrazide analogs as histone demethylase inhibitors University of Utah Research Foundation 10/17/182D 3D TSV
US9555022 102 Substituted triazolopyridines Bayer Intellectual Property GmbH 10/17/182D 3D TSV
US10047080 42 (R)-2-methyl-piperazine derivatives as CXCR3 receptor modulators IDORSIA PHARMACEUTICALS LTD. 10/10/182D 3D TSV
US10045974 14 2-amino-6-(difluoromethyl)-5,5-difluoro-6-phenyl-3,4,5,6-tetrahydropyridines as BACE1 inhibitors H. Lundbeck A/S 10/10/182D 3D TSV
US9556175 46 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and thier use as pharmaceutical compositions Boehringer Ingelheim International GmbH 10/10/182D 3D TSV
US10047073 12 Histone deacetylase inhibitors and compositions and methods of use thereof CHDI FOUNDATION, INC 10/10/182D 3D TSV
US10047084 43 Imidazolone derivatives, pharmaceutical compositions and uses thereof BEIJING FORELANDPHARMA CO. LTD. 10/10/182D 3D TSV
US10047093 120 Substituted imidazo[1,2-B]pyridazines as protein kinase inhibitors TOLERO PHARMACEUTICALS, INC. 10/10/182D 3D TSV
US9556191 8 Aminoquinazoline derivatives and their salts and methods of use thereof SUNSHINE LAKE PHARMA CO., LTD. 10/05/182D 3D TSV
US9556160 76 Guanidine compound Astellas Pharma Inc. 10/03/182D 3D TSV
US9562012 23 PPAR-sparing compounds for the treatment of metabolic diseases Metabolic Solutions Development Company, LLC 10/03/182D 3D TSV
US9561238 6 Pharmaceutical compositions comprising estetrol derivatives for use in cancer therapy Donesta Bioscience B.V. 10/03/182D 3D TSV
US10047098 188 C5-C6-oxacyclic fused iminopyrimidinone compounds as bace inhibitors, compositions, and their use Merck Sharp & Dohme Corp. 10/02/182D 3D TSV
US10047103 384 Imidazothiadiazole and imidazopyrazine derivatives as protease activated receptor 4 (PAR4) inhibitors for treating platelet aggregation Bristol-Myers Squibb Company; Universite de Montreal 10/02/182D 3D TSV
US10047097 105 Method of treatment using substituted pyrazolo[1,5-a] pyrimidine compounds Array BioPharma Inc. 10/02/182D 3D TSV
US10047092 276 Substituted [1,2,4]triazolo[4,3-a]pyrazines as P2X7 modulators Janssen Pharmaceutica NV 10/02/182D 3D TSV
US10047096 454 Substituted pyridobenzodiazepinone-derivatives and use thereof Bayer Pharma Aktiengesellschaft 10/02/182D 3D TSV
US9556181 21 Substituted pyrazolopyrimidinylamino-indazoles BAYER PHARMA AKTIENGESELLSCHAFT 09/30/182D 3D TSV
US9540377 1285 2,6,7,8 substituted purines as HDM2 inhibitors Merck Sharp & Dohme Corp. 09/26/182D 3D TSV
US9556157 6 Enhancer of zeste homolog 2 inhibitors GlaxoSmithKline Intellectual Property (No.2) Limited 09/26/182D 3D TSV
US9556170 3 Substituted-1H-benzo[d]imidazole series compounds as lysine-specific demethylase 1 (LSD1) inhibitors University of Utah Research Foundation 09/26/182D 3D TSV
US9546152 448 2-pyridyloxy-3-substituted-4-nitrile orexin receptor antagonists MERCK SHARP & DOHME CORP. 09/18/182D 3D TSV
US9546153 514 Bicyclic heterocycle substituted pyridyl compounds useful as kinase modulators Bristol-Myers Squibb Company 09/18/182D 3D TSV
US9533992 75 PDE9 inhibitors with imidazo triazinone backbone TBA 09/18/182D 3D TSV
US9550778 52 Substituted 6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analogs as negative allosteric modulators of mGluR5 Vanderbilt University 09/18/182D 3D TSV
US9556111 23 Tertiary amines for use in the treatment of cardiac disorders UNIVERSITETET I OSLO 09/18/182D 3D TSV
US9556145 22 2-pyridyloxy-4-ester orexin receptor antagonists MERCK SHARP & DOHME CORP. 09/07/182D 3D TSV
US9540359 15 Dihydrooxazine or oxazepine derivatives having BACE1 inhibitory activity Shionogi & Co., Ltd. 09/07/182D 3D TSV
US9556147 7 Inhibitors of bruton's tyrosine kinase HOFFMANN-LA INC. 09/07/182D 3D TSV
US9550781 26 Kinase modulating compounds, compositions containing the same and use thereof Centaurus Biopharma Co., Ltd.; Chia Tai Tianqing Pharmaceutical Group Co., Ltd. 09/07/182D 3D TSV
US9556132 41 Tetrazole derivatives and their use as potassium channel modulators Saniona A/S 09/07/182D 3D TSV
US9540396 38 6-arylamino pyridone carboxamide as MEK inhibitors Centaurus Biopharma Co., Ltd.; Chia Tai Tianqing Pharmaceutical Group Co., Ltd. 08/28/182D 3D TSV
US9550755 5 Complement pathway modulators and uses thereof NOVARTIS AG 08/28/182D 3D TSV
US9546168 29 ERK inhibitors Merck Sharp & Dohme Corp. 08/28/182D 3D TSV
US9550774 2 Dihydropyrido pyrimidine compounds as autotaxin inhibitors Eli Lilly and Company 08/25/182D 3D TSV
US9527857 211 HSPC-sparing treatments for RB-positive abnormal cellular proliferation GI Therapeutics, Inc. 08/25/182D 3D TSV
US9540379 222 (1,2,4)triazolo[4,3-A]quinoxaline derivatives as inhibitors of phosphodiesterases Boehringer Ingelheim International GmbH 08/24/182D 3D TSV
US9539260 567 Dihydro-benzo-oxazine and dihydro-pyrido-oxazine derivatives NOVARTIS AG 08/24/182D 3D TSV
US9540357 74 15-aryl prostaglandins as EP4 agonists, and methods of use thereof Allergan, Inc. 08/16/182D 3D TSV
US9540323 274 7-hydroxy-indolinyl antagonists of P2Y1 receptor Bristol-Myers Squibb Company 08/16/182D 3D TSV
US9540388 197 P2X7 modulators Janssen Pharmaceutica NV 08/16/182D 3D TSV
US9527851 130 Pyrrole six-membered heteroaryl ring derivative, preparation method thereof, and medicinal uses thereof Jiangsu Hengrui Medicine Co., Ltd.; Shanghai Hengrui Pharmaceutical Co., Ltd. 08/16/182D 3D TSV
US9540352 14 Substituted 1,7-naphthyridines as dopamine D1 ligands Pfizer Inc. 08/16/182D 3D TSV
US9670229 31 5-HT3 receptor antagonists Takeda Pharmaceutical Company Limited 08/07/182D 3D TSV
US9522914 174 Azole derivative TAISHO PHARMACEUTICAL CO., LTD 08/07/182D 3D TSV
US9540364 19 Benzimidazole tetrahydrofuran derivatives Merck Sharp & Dohme Corp. 08/07/182D 3D TSV
US9676777 3 Compounds useful for producing an optically active diazabicyclooctane compound MEIJI SEIKA PHARMA CO., LTD. 08/07/182D 3D TSV
US9533999 64 Fused thiazin-3-ones as KCA3.1 inhibitors Boehringer Ingelheim International GmbH 08/07/182D 3D TSV
US9670231 368 Fused tricyclic amide compounds as multiple kinase inhibitors BeiGene, Ltd. 08/07/182D 3D TSV
US9670230 12 Heteroaryl compounds and methods of use thereof Sunovion Pharmaceuticals Inc. 08/07/182D 3D TSV
US9676783 105 Method of treatment using substituted pyrazolo[1,5-A] pyrimidine compounds Array BioPharma, Inc. 08/07/182D 3D TSV
US9670255 3 Modified biotin, mutant streptavidin, and use thereof SAVID THERAPEUTICS INC. 08/07/182D 3D TSV
US9676786 4 Pharmacologically active compounds THE UNIVERSITY OF LIVERPOOL 08/07/182D 3D TSV
US9676792 4 Pyrimido-diazepinone compounds and methods of treating disorders Dana-Farber Cancer Institute, Inc. 08/07/182D 3D TSV
US9540384 58 Pyrrolidino heterocycles Hoffmann-La Roche, Inc. 08/07/182D 3D TSV
US9533995 14 Substituted N-heteroaryl spirolactam bipyrrolidines, preparation and therapeutic use thereof Sanofi 08/07/182D 3D TSV
US9676782 342 Substituted pyrazolo[1,5-a]pyrazines as negative allosteric modulators of metabotropic glutamate receptor 3 Vanderbilt University 08/07/182D 3D TSV
US9540373 27 Substituted spirocycles Boehringer Ingelheim International GmbH 08/07/182D 3D TSV
US9676818 32 Toll-like receptor 2-agonistic lipopeptides, and method of making the same University of Kansas 08/07/182D 3D TSV
US9670211 45 Aza-oxo-indoles for the treatment and prophylaxis of respiratory syncytial virus infection HOFFMANN-LA ROCHE INC. 07/07/182D 3D TSV
US9670216 58 Cannabinoid-2 agonists ALLERGAN, INC. 07/07/182D 3D TSV
US9670204 211 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders GALAPAGOS NV 07/07/182D 3D TSV
US9670210 116 Cyclopropylamines as LSD1 inhibitors Incyte Corporation 07/07/182D 3D TSV
US9670220 66 Fused heterocyclic derivatives as S1P modulators Abbvie B.V.; AbbiVie Inc. 07/07/182D 3D TSV
US9670203 142 Fused tricyclic urea compounds as Raf kinase and/or Raf kinase dimer inhibitors BeiGene, Ltd. 07/07/182D 3D TSV
US9670212 191 Inhibitors of PI3K-delta and methods of their use and manufacture Exelixis, Inc. 07/07/182D 3D TSV
US9670209 69 Muscarinic agonists ACADIA PHARMACEUTICALS INC.; ALLERGAN, INC. 07/07/182D 3D TSV
US9670213 175 Pteridine ketone derivative and applications thereof as EGFR, BLK, and FLT3 inhibitor East China University of Science and Technology 07/07/182D 3D TSV
US9670208 48 Serine/threonine kinase inhibitors Array BioPharma Inc.; Genentech, Inc. 07/07/182D 3D TSV
US9670214 404 Small molecule myristate inhibitors of Bcr-abl and methods of use DANA-FARBER CANCER INSTITUTE, INC.; THE SCRIPPS RESEARCH INSTITUTE 07/07/182D 3D TSV
US9670136 210 (Hetero)aryl cyclopropylamine compounds as LSD1 inhibitors ORYZON GENOMICS S.A. 05/19/182D 3D TSV
US9670142 171 1,3-diaminocyclopentane carboxamide derivatives Merck Patent GmbH 05/19/182D 3D TSV
US9669034 227 4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group BAYER INTELLECTUAL PROPERTY GMBH 05/19/182D 3D TSV
US9670161 20 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group BAYER PHARMA AKTIENGESELLSCHAFT 05/19/182D 3D TSV
US9670157 271 Benzylamine derivatives Kalvista Pharmaceuticals Limited 05/19/182D 3D TSV
US9669035 66 Combinations comprising PDE 2 inhibitors such as 1-aryl-4-methyl-[1,2,4]triazolo-[4,3-A]]quinoxaline compounds and PDE 10 inhibitors for use in the treatment of neurological of metabolic disorders JANSSEN PHARMACEUTICA NV 05/19/182D 3D TSV
US9669095 13 Cyclosporin analogues for preventing or treating hepatitis C infection ENANTA PHARMACEUTICALS, INC. 05/19/182D 3D TSV
US9670195 3 Glycosidase inhibitors and uses thereof Alectos Therapeutics Inc.; Merck Sharp & Dohme Corp. 05/19/182D 3D TSV
US9669029 114 Heteroaromatic phenylimidazole derivatives as PDE10A enzyme inhibitors H. Lundbeck A/S 05/19/182D 3D TSV
US9669031 313 MNK inhibitors and methods related thereto eFFECTOR THERAPEUTICS, INC. 05/19/182D 3D TSV
US9670201 104 Methyl- and trifluoromethyl-substituted pyrrolopyridine modulators of RORC2 and methods of use thereof Pfizer Inc. 05/19/182D 3D TSV
US9670191 116 Pyridyl-and pyrimidinyl-substituted pyrrole-, thiophene- and furane-derivatives as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. 05/19/182D 3D TSV
US9669028 175 Substituted 5-(pyrazin-2-yl)-1H-pyrazolo [3, 4-B] pyridine and pyrazolo [3, 4-B] pyridine derivatives as protein kinase inhibitors ARRIEN PHARMACEUTICALS LLC 05/19/182D 3D TSV
US9670181 87 Substituted 6,7-dialkoxy-3-isoquinolinol derivatives as inhibitors of phosphodiesterase 10 (PDE 10A) ALLERGAN, INC.; EXONHIT THERAPEUTICS SA 05/19/182D 3D TSV
US9670194 71 Substituted aminopyrimidine compounds and methods of use CALITOR SCIENCES, LLC; SUNSHINE LAKE PHARMA CO., LTD. 05/19/182D 3D TSV
US9670166 297 Substituted bicyclic dihydropyrimidinones and their use as inhibitors of neutrophil elastase activity Boehringer Ingelheim International GmbH 05/19/182D 3D TSV
US9670202 22 Substituted triazolopyridines BAYER PHARMA AKTIENGESELLSCHAFT 05/19/182D 3D TSV
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US9402878 2 Depsipeptide and uses thereof NovoBiotic Pharmaceuticals, LLC 07/10/172D 3D TSV
US9388139 97 Derivatives of celeboxib, use thereof and preparation thereof German University; Southern Research Institute 07/10/172D 3D TSV
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US9388136 35 Tert-butyl N-[2-{4-[6-amino-5-(2,4-difluorobenzoyl)-2-oxopyridin-1(2H)-yl]-3,5-difluorophenyl}ethyl]-L-alaninate or a salt, hydrate or solvate thereof Chroma Therapeutics Ltd 07/10/172D 3D TSV
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US9365562 126 1,3 substituted azetidine PDE10 inhibitors Merck Sharp & Dohme Corp. 07/03/172D 3D TSV
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US9359371 77 Bicyclic substituted pyrimidine compounds XUANZHU PHARMA CO., LTD. 07/03/172D 3D TSV
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US9365502 18 Neuroactive substituted cyclopenta[b]phenanthrenes as modulators for GABA type-A receptors WASHINGTON UNIVERSITY 07/03/172D 3D TSV
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US9353089 180 Compositions and methods for the treatment of malaria Saint Louis University; Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences 06/26/172D 3D TSV
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US8980905 10 Benzodioxole or benzodioxepine heterocyclic compounds as phosphodiesterase inhibitors Leo Pharma A/S 08/10/152D 3D TSV
US8975415 367 Chromane compounds CoMentis, Inc. 08/10/152D 3D TSV
US8980916 3 Factor IXa inhibitors Merck Sharp & Dohme Corp.; Mochida Pharmaceutical Co., Ltd. 08/10/152D 3D TSV
US8980904 18 Heterocyclic substituted pyrimidine compound Xuanzhu Pharma Co., Ltd. 08/10/152D 3D TSV
US8975409 18 Phenyl derivative ONO Pharmaceutical Co., Ltd. 08/10/152D 3D TSV
US8975417 716 Pyrazolopyrrolidine derivatives and their use in the treatment of disease Novartis AG 08/10/152D 3D TSV
US8980906 50 Pyridonemorphinan analogs and biological activity on opioid receptors Purdue Pharma L.P. 08/10/152D 3D TSV
US8980929 14 Substituted seven-membered heterocyclic compounds as dipeptidyl peptidase-iv inhibitors for the treatment of diabetes Merck Sharp & Dohme Corp. 08/10/152D 3D TSV
US8975250 13 5 oxo-5,8-dihydropyrido[2,3-d]pyrimidine derivatives as CaMKII kinase inhibitors for treating cardiovascular diseases SANOFI 08/03/152D 3D TSV
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US8975249 94 Heterocyclic compounds and uses thereof Celgene Avilomics Research, Inc. 08/03/152D 3D TSV
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US8962860 19 Inhibitors of glutaminyl cyclase Probiodrug AG 08/03/152D 3D TSV
US8975247 27 Methods and compositions of treating a flaviviridae family viral infection The Board of Trustees of the Leland Stanford Junion University 08/03/152D 3D TSV
US8975252 2 Morpholine derivative Shanghai Pharmaceuticals Holding Co., Ltd.; Mitsubishi Tanabe Pharma Corporation 08/03/152D 3D TSV
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US8975265 371 Substituted imidazo[1,2-a]pyrimidines and —pyridines Bayer Intellectual Property GmbH 08/03/152D 3D TSV
US8975282 8 Substituted pyrazolone compounds and methods of use Sunshine Lake Pharma Co., Ltd.; Calitor Sciences, LLC 08/03/152D 3D TSV
US8975267 51 Tricyclic pyrrolo derivatives, process for their preparation and their use as kinase inhibitors Nerviano Medical Sciences S.r.l. 08/03/152D 3D TSV
US8962637 76 Bicyclic compounds and their uses as dual c-SRC/JAK inhibitors Debiopharm S.A.; Aurigene Discovery Technologies Ltd. 07/22/152D 3D TSV
US8962651 8 Compounds for the treatment of hepatitis C Bristol-Myers Squibb Company 07/22/152D 3D TSV
US8962674 93 Curcumin derivative Tokyo Institute of Technology; Kyoto University 07/22/152D 3D TSV
US8962837 24 Nitrogen heterocycle derivatives, preparation thereof and application thereof in human therapeutics Pierre Fabre Medicament 07/22/152D 3D TSV
US8962646 38 Peripherally acting opioid compounds Alkermes, Inc. 07/22/152D 3D TSV
US8962659 4 Phenoxyethyl piperidine compounds Eli Lilly and Company 07/22/152D 3D TSV
US8962641 490 Pyrimidine-substituted pyrrolidine derivatives, pharmaceutical compositions and uses thereof Boehringer Ingelheim International GmbH 07/22/152D 3D TSV
US8962630 205 Pyrrolopyrimidine compounds and their uses Novartis AG 07/22/152D 3D TSV
US8962664 3 Selective glycosidase inhibitors and uses thereof Simon Fraser University 07/22/152D 3D TSV
US8962859 12 Spiro-amino-imidazo-fused heterocyclic compounds as beta-secretase modulators and methods of use Amgen Inc. 07/22/152D 3D TSV
US8962648 231 Tricyclic compounds and PBK inhibitors containing the same OncoTherapy Science, Inc. 07/22/152D 3D TSV
US8957084 9 7,8-cyclicmorphinan analogs Purdue Pharma L.P. 07/15/152D 3D TSV
US8957219 12 Acetic acid amide derivative having inhibitory activity on endothelial lipase Shionogi & Co., Ltd. 07/15/152D 3D TSV
US8957103 18 Conjugated 3-(indolyl)- and 3-(azaindolyl)-4-arylmaleimide compounds and their use in tumor treatment Johannes Gutenberg—Universitat Mainz 07/15/152D 3D TSV
US8962608 1192 Cycloalkylnitrile pyrazole carboxamides as janus kinase inhibitors Merck Sharp & Dohme Corp. 07/15/152D 3D TSV
US8962616 41 Heterocyclic substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds Pfizer Inc. 07/15/152D 3D TSV
US8957093 262 N-biphenylmethylindole modulators of PPARG The Scripps Research Institute 07/15/152D 3D TSV
US8962609 129 Pyrimidine compounds as inhibitors of protein kinases IKK epsilon and/or TBK-1, processes for their preparation, and pharmaceutical compositions containing them Domainex Limited 07/15/152D 3D TSV
US8962611 356 Substituted imidazopyridines as HDM2 inhibitors Merck Sharp & Dohme Corp. 07/15/152D 3D TSV
US8962619 36 Substituted imidazopyridinyl-aminopyridine compounds ArQule, Inc. 07/15/152D 3D TSV
US8962612 20 Tetrahydroisoquinoline derivative Astellas Pharma Inc. 07/15/152D 3D TSV
US8957075 28 O-GlcNAc transferase inhibitors and uses thereof President and Fellows of Harvard College 07/10/152D 3D TSV
US8957077 14 Pyrazolopyrimidine PDE 10 inhibitors Merck Sharp & Dohme Corp. 07/10/152D 3D TSV
US8957074 298 Pyrrolopyrimidine compounds as inhibitors of CDK4/6 Novartis AG 07/10/152D 3D TSV
US8957083 31 Spiro-amino-imidazolone and spiro-amino-dihydro-pyrimidinone compounds as beta-secretase modulators and methods of use Amgen Inc. 07/10/152D 3D TSV
US8957068 870 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH Novartis AG 07/09/152D 3D TSV
US8957064 185 Fused pyrimidines Bayer Intellectual Property GmbH 07/09/152D 3D TSV
US8957059 66 Modulators of serotonin receptors Janssen Pharmaceutica NV 07/09/152D 3D TSV
US8957073 378 Unsaturated nitrogen heterocyclic compounds useful as PDE10 inhibitors Amgen Inc. 07/09/152D 3D TSV
US8957057 4 Use of azaphilone compounds for the modulation of the activity of a nuclear hormone receptor Food Industry Research and Development Institute 07/09/152D 3D TSV
US8952177 191 1,2,6-substituted benzimidazoles as FLAP modulators Janssen Pharmaceutica NV 06/29/152D 3D TSV
US8952157 407 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases AbbVie Inc.; The Walter and Eliza Hall Institute of Medical Research 06/29/152D 3D TSV
US8952036 5 Benzoic acid derivative MDM2 inhibitor for the treatment of cancer Amgen Inc. 06/29/152D 3D TSV
US8952037 98 Heteroaryloxycarbocyclyl compounds as PDE10 inhibitors Amgen Inc. 06/29/152D 3D TSV
US8956589 22 Imaging diagnostic agent and extracorporeal diagnostic agent for incurable neurological diseases Shiga University of Medical Science 06/29/152D 3D TSV
US8952027 12 Inhibitors of syk and JAK protein kinases Portola Pharmaceuticals, Inc. 06/29/152D 3D TSV
US8952025 3 Multifunctional radical quenchers and their uses Arizona Board of Regents, A Body Corporate of the State of Arizona Acting for and on Behalf of Arizona State University 06/29/152D 3D TSV
US8952169 708 N-substituted benzamides and methods of use thereof Xenon Pharmaceuticals Inc.; Genentech, Inc. 06/29/152D 3D TSV
US8952150 30 Prostaglandin transporter inhibitors and uses thereof Albert Einstein College of Medicine of Yeshiva University 06/29/152D 3D TSV
US8952128 168 Somatostatin-dopamine chimeric analogs Ipsen Pharma S.A.S. 06/29/152D 3D TSV
US8969583 55 3-phenyl-5-ureidoisothiazole-4-carboximide and 3-amino-5-phenylisothiazole derivatives as kinase inhibitors Allergan, Inc. 06/22/152D 3D TSV
US8952002 3 Aminoheteroaryl compounds and preparation method and use thereof Shanghai Allist Pharmaceuticals, Inc. 06/22/152D 3D TSV
US8969358 54 Buprenorphine analogs Purdue Pharma L.P. 06/22/152D 3D TSV
US8952008 50 Chemical compounds Pfizer Limited 06/22/152D 3D TSV
US8969348 10 Chymase inhibitors Boehringer Ingelheim International GmbH 06/22/152D 3D TSV
US8969336 95 Diamino heterocyclic carboxamide compound Astellas Pharma Inc.; Kotobuki Pharmaceutical Co., Ltd. 06/22/152D 3D TSV
US8969578 13 Inhibitors of STAT3 University of Central Florida Research Foundation, Inc. 06/22/152D 3D TSV