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Patent: (prefix with "US" like US6078908)
PatentDataPatent TitleOrganizationDepositionDownloads
US9670211 45 Aza-oxo-indoles for the treatment and prophylaxis of respiratory syncytial virus infection HOFFMANN-LA ROCHE INC. 07/07/182D 3D TSV
US9670216 57 Cannabinoid-2 agonists ALLERGAN, INC. 07/07/182D 3D TSV
US9670204 211 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders GALAPAGOS NV 07/07/182D 3D TSV
US9670210 116 Cyclopropylamines as LSD1 inhibitors Incyte Corporation 07/07/182D 3D TSV
US9670220 66 Fused heterocyclic derivatives as S1P modulators Abbvie B.V.; AbbiVie Inc. 07/07/182D 3D TSV
US9670203 142 Fused tricyclic urea compounds as Raf kinase and/or Raf kinase dimer inhibitors BeiGene, Ltd. 07/07/182D 3D TSV
US9670212 191 Inhibitors of PI3K-delta and methods of their use and manufacture Exelixis, Inc. 07/07/182D 3D TSV
US9670209 69 Muscarinic agonists ACADIA PHARMACEUTICALS INC.; ALLERGAN, INC. 07/07/182D 3D TSV
US9670213 109 Pteridine ketone derivative and applications thereof as EGFR, BLK, and FLT3 inhibitor East China University of Science and Technology 07/07/182D 3D TSV
US9670208 48 Serine/threonine kinase inhibitors Array BioPharma Inc.; Genentech, Inc. 07/07/182D 3D TSV
US9670214 404 Small molecule myristate inhibitors of Bcr-abl and methods of use DANA-FARBER CANCER INSTITUTE, INC.; THE SCRIPPS RESEARCH INSTITUTE 07/07/182D 3D TSV
US9670136 210 (Hetero)aryl cyclopropylamine compounds as LSD1 inhibitors ORYZON GENOMICS S.A. 05/19/182D 3D TSV
US9670142 171 1,3-diaminocyclopentane carboxamide derivatives Merck Patent GmbH 05/19/182D 3D TSV
US9669034 227 4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group BAYER INTELLECTUAL PROPERTY GMBH 05/19/182D 3D TSV
US9670161 20 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group BAYER PHARMA AKTIENGESELLSCHAFT 05/19/182D 3D TSV
US9670157 271 Benzylamine derivatives Kalvista Pharmaceuticals Limited 05/19/182D 3D TSV
US9669035 66 Combinations comprising PDE 2 inhibitors such as 1-aryl-4-methyl-[1,2,4]triazolo-[4,3-A]]quinoxaline compounds and PDE 10 inhibitors for use in the treatment of neurological of metabolic disorders JANSSEN PHARMACEUTICA NV 05/19/182D 3D TSV
US9669095 13 Cyclosporin analogues for preventing or treating hepatitis C infection ENANTA PHARMACEUTICALS, INC. 05/19/182D 3D TSV
US9670195 3 Glycosidase inhibitors and uses thereof Alectos Therapeutics Inc.; Merck Sharp & Dohme Corp. 05/19/182D 3D TSV
US9669029 114 Heteroaromatic phenylimidazole derivatives as PDE10A enzyme inhibitors H. Lundbeck A/S 05/19/182D 3D TSV
US9669031 313 MNK inhibitors and methods related thereto eFFECTOR THERAPEUTICS, INC. 05/19/182D 3D TSV
US9670201 104 Methyl- and trifluoromethyl-substituted pyrrolopyridine modulators of RORC2 and methods of use thereof Pfizer Inc. 05/19/182D 3D TSV
US9670191 116 Pyridyl-and pyrimidinyl-substituted pyrrole-, thiophene- and furane-derivatives as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. 05/19/182D 3D TSV
US9669028 175 Substituted 5-(pyrazin-2-yl)-1H-pyrazolo [3, 4-B] pyridine and pyrazolo [3, 4-B] pyridine derivatives as protein kinase inhibitors ARRIEN PHARMACEUTICALS LLC 05/19/182D 3D TSV
US9670181 87 Substituted 6,7-dialkoxy-3-isoquinolinol derivatives as inhibitors of phosphodiesterase 10 (PDE 10A) ALLERGAN, INC.; EXONHIT THERAPEUTICS SA 05/19/182D 3D TSV
US9670194 71 Substituted aminopyrimidine compounds and methods of use CALITOR SCIENCES, LLC; SUNSHINE LAKE PHARMA CO., LTD. 05/19/182D 3D TSV
US9670166 273 Substituted bicyclic dihydropyrimidinones and their use as inhibitors of neutrophil elastase activity Boehringer Ingelheim International GmbH 05/19/182D 3D TSV
US9670202 22 Substituted triazolopyridines BAYER PHARMA AKTIENGESELLSCHAFT 05/19/182D 3D TSV
US9670196 13 Thiazole-substituted aminoheteroaryls as Spleen Tyrosine Kinase inhibitors Merck Sharp & Dohme Corp. 05/19/182D 3D TSV
US9670193 138 Trifluoromethyl-oxadiazole derivatives and their use in the treatment of disease Novartis AG 05/19/182D 3D TSV
US9676728 19 2-benzyl-benzimidazole complement factor B inhibitors and uses thereof Novartis AG 04/16/182D 3D TSV
US9675697 203 BET bromodomain inhibitors and therapeutic methods using the same THE REGENTS OF THE UNIVERSITY OF MICHIGAN 04/16/182D 3D TSV
US9676721 112 Compounds and compositions for the inhibition of NAMPT FORMA TM, LLC 04/16/182D 3D TSV
US9676701 287 Cyclopropylamine derivatives useful as LSD1 inhibitors ORYZON GENOMICS, S.A. 04/16/182D 3D TSV
US9676732 74 Ethynyl derivatives HOFFMANN-LA ROCHE INC. 04/16/182D 3D TSV
US9676712 15 Lactam compounds as EP4 receptor-selective agonists for use in the treatment of EP4-mediated diseases and conditions CAYMAN CHEMICAL COMPANY, INC. 04/16/182D 3D TSV
US9676720 29 Substituted biaryl compound UBE INDUSTRIES, LTD. 04/16/182D 3D TSV
US9675616 13 Arylaminoalcohol-substituted 2,3-dihydroimidazo[1,2-C]quinolines BAYER INTELLECTUAL PROPERTY GMBH 04/12/182D 3D TSV
US9688710 328 Inhibitors of sodium glucose cotransporter 1 Lexicon Pharmaceuticals, Inc. 04/12/182D 3D TSV
US9675614 334 PRMT5 inhibitors and uses thereof Epizyme, Inc. 04/12/182D 3D TSV
US9688696 116 Piperidine/piperazine derivatives Janssen Pharmaceutica N.V. 04/12/182D 3D TSV
US9688816 46 Polyetherimide compositions and methods for the manufacture and use thereof SABIC GLOBAL TECHNOLOGIES B.V. 04/12/182D 3D TSV
US9675612 45 Substituted thiazolopyrimidines BAYER PHARMA AKTIENGESELLSCHAFT 04/12/182D 3D TSV
US9688680 950 Compositions useful for treating disorders related to kit BLUEPRINT MEDICINES CORPORATION 03/27/182D 3D TSV
US9688695 384 Imidazothiadiazole and imidazopyrazine derivatives as protease activated receptor 4 (PAR4) inhibitors for treating platelet aggregation BRISTOL-MYERS SQUIBB COMPANY 03/27/182D 3D TSV
US9688678 37 Oxindole compounds carrying a nitrogen-bound spiro substituent and use thereof for treating vasopressin-related diseases AbbVie Deutschland GmbH & Co. KG 03/27/182D 3D TSV
US9688683 31 Substituted condensed pyrimidine compounds Dalhousie University 03/27/182D 3D TSV
US9688684 278 Substituted tetrazolo[1,5-a]pyrazines as ROR-gamma inhibitors Merck Patent GmbH 03/27/182D 3D TSV
US9688676 65 Tyrosine kinase inhibitors PRINCIPIA BIOPHARMA INC. 03/27/182D 3D TSV
US9688672 450 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH NOVARTIS AG 03/19/182D 3D TSV
US9688668 150 Long chain base sphingosine kinase inhibitors University of Virginia Patent Foundation 03/19/182D 3D TSV
US9688664 8 Modulators of fatty acid amide hydrolase Janssen Pharmaceutica NV 03/19/182D 3D TSV
US9688669 125 Oxazolidinones as modulators of mGluR5 Bristol-Myers Squibb Company 03/19/182D 3D TSV
US9688661 139 Substituted pyrroles active as kinases inhibitors NERVIANO MEDICAL SCIENCES S.R.L. 03/19/182D 3D TSV
US9675593 518 Anti-fibrotic pyridinones INTERMUNE, Inc. 03/16/182D 3D TSV
US9675594 46 Arylpyrrolopyridine derived compounds as LRRK2 inhibitors H. Lundbeck A/S 03/16/182D 3D TSV
US9675539 2 Cosmetic and pharmaceutical compositions and methods using 2-decarboxy-2-phosphinico derivatives Duke University 03/16/182D 3D TSV
US9675571 28 Inhibitors of indoleamine 2,3-dioxygenase (IDO) Bristol-Myers Squibb Company 03/16/182D 3D TSV
US9688645 25 Macrocyclic urea and sulfamide derivatives as inhibitors of TAFIa SANOFI 03/16/182D 3D TSV
US9675591 9 Methods for treating seizure disorders and pain SRMLSC 03/16/182D 3D TSV
US9675605 83 Substituted naphthyridine and quinoline compounds as MAO inhibitors Dart NeuroScience (Cayman) Ltd. 03/16/182D 3D TSV
US9688642 96 Substituted pyrazines as GPR40 agonists Janssen Pharmaceutica NV 03/12/182D 3D TSV
US9688643 325 Triazine derivative and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. 03/12/182D 3D TSV
US9688638 35 Opioid agonists and uses thereof Nektar Therapeutics 03/11/182D 3D TSV
US9682995 359 Amino-substituted isothiazoles BAYER PHARMA AKTIENGESELLSCHAFT 03/10/182D 3D TSV
US9682993 22 Anticancer compounds St. Jude Children's Research Hospital 03/10/182D 3D TSV
US9682983 326 BMP inhibitors and methods of use thereof The Brigham and Women's Hospital, Inc.; Dept. of Health and Human Services, National Institutes of Health 03/10/182D 3D TSV
US9688615 706 Benzimidazole inhibitors of the sodium channel DEGIACOMO, INTERIM TRUSTEE, MARK G. 03/10/182D 3D TSV
US9688624 12 DP2 antagonist and uses thereof Brickell Biotech, Inc. 03/10/182D 3D TSV
US9687494 21 Iminothiadiazine dioxide compounds as BACE inhibitors, compositions, and their use Ambit Biosciences 03/10/182D 3D TSV
US9688629 262 Indole carboxamide compounds Bristol-Myers Squibb Company 03/10/182D 3D TSV
US9687479 520 Multisubstituted aromatic compounds as serine protease inhibitors VERSEON CORPORATION 03/10/182D 3D TSV
US9687478 34 Quinuclidine derivatives and medicinal compositions containing the same ALMIRALL, S.A. 03/10/182D 3D TSV
US9687483 5 Treatment of cerebral cavernous malformations and cerebral aneurysms with Rho kinase inhibitors BIOAXONE BIOSCIENCES, INC. 03/10/182D 3D TSV
US9682991 198 Tricyclic compounds for use as kinase inhibitors FUNDACIÓN CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS CARLOS III 03/10/182D 3D TSV
US9682971 220 1,2,5-Substituted benzimidazoles as flap modulators JANSSEN PHARMACEUTICA NV 02/14/182D 3D TSV
US9682980 85 Positive allosteric modulators of mGluR2 Bristol-Myers Squibb Company 02/14/182D 3D TSV
US9682976 324 Protein kinase C inhibitors and uses thereof Rigel Pharmaceuticals, Inc. 02/14/182D 3D TSV
US9682959 6 Ethynyl derivatives HOFFMANN-LA ROCHE INC. 02/13/182D 3D TSV
US9682965 75 Fumagillol heterocyclic compounds and methods of making and using same Zafgen, Inc. 02/13/182D 3D TSV
US9682966 563 Kappa opioid ligands The Scripps Research Institute 02/13/182D 3D TSV
US9682967 50 N-substituted-5-substituted phthalamic acids as sortilin inhibitors H. Lundbeck A/S 02/13/182D 3D TSV
US9682960 137 Non-steroidal antiandrogens and selective androgen receptor modulators with a pyridyl moiety ENDORECHERCHE, INC. 02/13/182D 3D TSV
US9682969 31 Phthalazinone compounds and methods for the treatment of cystic fibrosis Flatley Discovery Lab, LLC 02/13/182D 3D TSV
US9682968 110 Piperidinyl-indole derivatives complement factor B inhibitors and uses thereof Novartis AG 02/13/182D 3D TSV
US9682963 28 Pyridine derivatives as soft rock inhibitors Redx Pharma PLC 02/13/182D 3D TSV
US9682961 26 Quinazoline derivative CARNA BIOSCIENCES, INC.; NATIONAL CANCER CENTER 02/13/182D 3D TSV
US9682953 166 Amide compounds, compositions and applications thereof ADVINUS THERAPEUTICS LIMITED 02/07/182D 3D TSV
US9687476 60 Bisaryl-bonded aryltriazolones and use thereof Bayer Intellectual Property GmbH 02/07/182D 3D TSV
US9682141 2516 Combination of kinase inhibitors and uses thereof Intellikine LLC 02/07/182D 3D TSV
US9682957 192 Diamide compounds having muscarinic receptor antagonist and β2 adrenergic receptor agonist activity Theravance Respiratory Company, LLC 02/07/182D 3D TSV
US9682940 502 Indazole derivatives useful as CB-1 inverse agonists Janssen Pharmaceutica NV 02/07/182D 3D TSV
US9682955 280 Quinazoline derivatives useful as CB-1 inverse agonists Janssen Pharmaceutica NV 02/07/182D 3D TSV
US9682910 35 Series of skin-whitening (lightening) compounds Unigen, Inc. 02/07/182D 3D TSV
US9695195 162 5-HT3 receptor antagonists Takeda Pharmaceutical Company Limited 02/06/182D 3D TSV
US9695205 53 Amide compounds for treatment of complement mediated disorders Achillion Pharmaceuticals, Inc. 02/06/182D 3D TSV
US9695197 11 Glycosidase inhibitors and uses thereof Alectos Therapeutics Inc.; Merck Sharp & Dohme Corp. 02/06/182D 3D TSV
US9695200 175 Heterocyclic ITK inhibitors for treating inflammation and cancer Confluence Life Sciences, Inc. 02/06/182D 3D TSV
US9695151 90 3,4-dihydro-2H-isoquinoline-1-one and 2,3-dihydro-isoindol-1-one compounds Hoffmann-La Roche Inc. 01/26/182D 3D TSV
US9695152 84 3,4-dihydro-2H-isoquinoline-1-one and 2,3-dihydro-isoindol-1-one compounds Hoffmann-La Roche Inc. 01/26/182D 3D TSV
US9695194 126 Benzoxazinone derivatives for treatment of skin diseases SIXERA PHARMA AB 01/26/182D 3D TSV
US9695172 15 Diazepane derivatives and uses thereof Dana-Farber Cancer Institute, Inc. 01/26/182D 3D TSV
US9695175 51 Highly selective c-Met inhibitors as anticancer agents CB THERAPEUTICS INC. 01/26/182D 3D TSV
US9695181 15 Hydroximic acid derivatives and medical applications therof DOUBLE RIDER MEDICINE CO., LTD. 01/26/182D 3D TSV
US9695174 21 Inhibitor of breast cancer resistance protein (BCRP) Millennium Pharmaceuticals, Inc. 01/26/182D 3D TSV
US9695165 82 Inhibitors of the fibroblast growth factor receptor BLUEPRINT MEDICINES CORPORATION 01/26/182D 3D TSV
US9695179 17 Methods and compositions for inhibition of bromodomain-containing proteins ConverGene LLC 01/26/182D 3D TSV
US9695170 217 Naphthyridine derivatives as inhibitors of Hypoxia inducible factor (HIF) hydroxylase FibroGen, Inc. 01/26/182D 3D TSV
US9695160 36 Piperazine derivatives for treating disorders The University of Nottingham; NewSouth Innovations PTY Limited 01/26/182D 3D TSV
US9695183 702 Substituted 7-azabicycles and their use as orexin receptor modulators JANSSEN PHARMACEUTICA NV 01/26/182D 3D TSV
US9695180 119 Substituted imidazo[1,2-a]pyrazines as LSD1 inhibitors Incyte Corporation 01/26/182D 3D TSV
US9695168 158 Substituted imidazo[1,5-α]pyridines and imidazo[1,5-α]pyrazines as LSD1 inhibitors Incyte Corporation 01/26/182D 3D TSV
US9695176 4 Substituted imidazo[1,5-a]pyrazines as CGRP receptor antagonists Bristol-Myers Squibb Company 01/26/182D 3D TSV
US9695167 13 Substituted triazolo[1,5-a]pyridines and triazolo[1,5-a]pyrazines as LSD1 inhibitors Incyte Corporation 01/26/182D 3D TSV
US9695185 5 Synthetic methods for spiro-oxindole compounds Xenon Pharmaceuticals Inc. 01/26/182D 3D TSV
US9695163 76 Thiazole orexin receptor antagonists MERCK SHARP & DOHME CORP 01/26/182D 3D TSV
US9695149 235 1,2,6-substituted benzimidazoles as flap modulators JANSSEN PHARMACEUTICA NV 01/19/182D 3D TSV
US9695118 394 Benzamide derivative Chugai Seiyaku Kabushiki Kaisha 01/19/182D 3D TSV
US9694016 2555 Biaryl amide compounds as kinase inhibitors NOVARTIS AG 01/19/182D 3D TSV
US9695128 13 Ethynyl derivatives Hoffmann-La Roche Inc. 01/19/182D 3D TSV
US9695132 194 Heteroaryl compounds and uses thereof Celgene CAR LLC; Sanofi 01/19/182D 3D TSV
US9694018 12 IBAT inhibitors for the treatment of liver disease Albireo AB 01/19/182D 3D TSV
US9694015 59 Methods for the treatment of locally advanced breast cancer Celgene Corporation 01/19/182D 3D TSV
US9694024 17 Methods of treating retroviral infections and related dosage regimes Chimerix, Inc. 01/19/182D 3D TSV
US9694012 76 Pyrazol derivatives Hoffmann-La Roche Inc. 01/19/182D 3D TSV
US9694011 6 Substituted pyrazolopyrimidines as kinases inhibitors Jiangsu Medolution Ltd 01/19/182D 3D TSV
US9695131 56 Substituted uracils as chymase inhibitors Bayer Pharma Aktiengesellschaft 01/19/182D 3D TSV
US9693997 356 Antiviral compounds HOFFMANN-LA ROCHE INC. 01/14/182D 3D TSV
US9693992 251 IRE-1α inhibitors MannKind Corporation 01/14/182D 3D TSV
US9694002 648 Substituted benzamides and methods of use thereof GENENTECH, INC.; XENON PHARMACEUTICALS INC. 01/14/182D 3D TSV
US9527838 54 2-pyridinecarboxamide derivatives, compositions containing such compounds, and methods of treatment Merck Sharp & Dohme Corp. 12/04/172D 3D TSV
US9540323 274 7-hydroxy-indolinyl antagonists of P2Y1 receptor Bristol-Myers Squibb Company 12/04/172D 3D TSV
US9522914 174 Azole derivative TAISHO PHARMACEUTICAL CO., LTD 12/04/172D 3D TSV
US9527839 25 Benzimidazole tetrahydropyran derivatives Merck Sharp & Dohme Corp. 12/04/172D 3D TSV
US9527857 217 HSPC-sparing treatments for RB-positive abnormal cellular proliferation GI Therapeutics, Inc. 12/04/172D 3D TSV
US9533969 6 Materials and method for inhibiting replication protein A and uses thereof Indiana University Research and Technology Corporation 12/04/172D 3D TSV
US9533992 75 PDE9 inhibitors with imidazo triazinone backbone TBA 12/04/172D 3D TSV
US9532990 119 Polyfluorinated compounds acting as bruton tyrosine kinase inhibitors Zhejiang DTRM Biopharma Co. Ltd. 12/04/172D 3D TSV
US9527851 130 Pyrrole six-membered heteroaryl ring derivative, preparation method thereof, and medicinal uses thereof Jiangsu Hengrui Medicine Co., Ltd.; Shanghai Hengrui Pharmaceutical Co., Ltd. 12/04/172D 3D TSV
US9504692 48 Selective inhibition of MALT1 protease by phenothiazine derivatives HELMHOLTZ ZENTRUM MUNCHEN, DEUTSCHES FORSCHUNGSZENTRUM FUR GESUNDHEIT UND UMWELT (GMBH) 12/04/172D 3D TSV
US9533989 123 Substituted pyrimidine-5-carboxamides as spleen tyrosine kinase inhibitors Ziarco Pharma Ltd. 12/04/172D 3D TSV
US9533985 193 Sulfonamide derivative and medicinal use thereof EA Pharma Co., Ltd. 12/04/172D 3D TSV
US9522881 71 Hydroxyindole carboxylic acid based inhibitors for oncogenic Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) Indiana University Research and Technology Corporation 11/27/172D 3D TSV
US9512115 58 Inhibitors PROBIODRUG AG 11/27/172D 3D TSV
US9505766 158 Kinase inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 11/27/172D 3D TSV
US9522910 16 Protein kinase inhibitors (variants), use thereof in treating oncological diseases and a pharmaceutical composition based thereon OBSHCHESTVO S OGRANICHENNOY OTVETSTVENNOSTYOU “FUSION PHARMA” 11/27/172D 3D TSV
US9505762 338 Purine derivatives as CB2 receptor agonists HOFFMANN-LA ROCHE INC. 11/27/172D 3D TSV
US9512141 84 Pyrazine derivatives as CB2 receptor agonists HOFFMANN-LA ROCHE INC. 11/27/172D 3D TSV
US9512132 76 Pyrazole compounds as CB2 agonists Hoffmann-La Roche Inc. 11/27/172D 3D TSV
US9522886 195 Pyridine derivatives HOFFMANN-LA ROCHE INC. 11/27/172D 3D TSV
US9505749 527 Quinazolinone compounds and derivatives thereof AMGEN INC. 11/27/172D 3D TSV
US9505780 114 Thienopyranones as kinase and epigenetic inhibitors SignalRx Pharmaceuticals, Inc. 11/27/172D 3D TSV
US9512121 47 [1,2,4] triazol [4,3-A] pyridine derivative, preparation method therefor or medical application thereof Jiangsu Hansoh Pharmaceutical Co., Ltd. 11/27/172D 3D TSV
US9499492 130 4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl amines containing a sulfoximine group Bayer Pharma Aktiengesellschaft 11/20/172D 3D TSV
US9499502 733 5-substituted iminothiazines and their mono- and dioxides as BACE inhibitors, compositions, and their use Merck Sharp & Dohme Corp. 11/20/172D 3D TSV
US9512084 40 Amino pyrimidine derivatives Novartis AG 11/20/172D 3D TSV
US9499547 110 Amino-substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH 11/20/172D 3D TSV
US9493490 60 Boron-containing small molecules Anacor Pharmaceuticals, Inc. 11/20/172D 3D TSV
US9493486 113 Diazaspirocycloalkane and azaspirocycloalkane Hoffmann-La Roches Inc. 11/20/172D 3D TSV
US9505745 110 Enhancer of zeste homolog 2 inhibitors GlaxoSmithKline Intellectual Property (No. 2) Limited 11/20/172D 3D TSV
US9526727 30 Inhibitors of beta-secretase Vitae Pharmaceutical, Inc. 11/20/172D 3D TSV
US9499482 247 Pyrrolone or pyrrolidinone melanin concentrating hormone receptor-1 antagonists Bristol-Myers Squibb Company 11/20/172D 3D TSV
US9512114 52 Substituted aminopyrimidine compounds and methods of use CALITOR SCIENCES, LLC; SUNSHINE LAKE PHARMA CO., LTD. 11/20/172D 3D TSV
US9512126 25 Substituted imidazopyridazines Bayer Intellectual Property GmbH 11/20/172D 3D TSV
US9512169 23 3-substituted estra-1,3,5(10),16-tetraene derivatives, methods for the production thereof, pharmaceutical preparations containing same, and use thereof for the production of medicaments BAYER PHARMA AKTIENGESELLSCHAFT 11/13/172D 3D TSV
US9512068 14 Augmenting moieties for anti-inflammatory compounds RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY; LEHIGH UNIVERSITY 11/13/172D 3D TSV
US9493448 168 Cycloalkane derivatives DAIICHI SANKYO COMPANY, LIMITED 11/13/172D 3D TSV
US9511061 6 Incontinence treatment methods IXALTIS 11/13/172D 3D TSV
US9505753 69 Inhibitors of D-amino acid oxidase THE JOHNS HOPKINS UNIVERSITY 11/13/172D 3D TSV
US9512082 7 Inhibitors of glutaminyl cyclase PROBIODRUG AG 11/13/172D 3D TSV
US9493446 1134 Orexin receptor antagonists which are [ortho bi-(hetero-)aryl]-[2-(meta bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone derivatives ACTELION PHARMACEUTICALS LTD. 11/13/172D 3D TSV
US9512065 5 Polymorphs of N-[(R)-1-[(S)-1-(4-aminomethyl-benzylcarbamoyl)-2-phenyl-ethylcarbamoyl]-2-(4-ethoxy-phenyl)-ethyl]-benzamide hydrochloride Kalvista Pharmaceuticals Limited 11/13/172D 3D TSV
US9493485 178 Spirocyclic dihydro-thiazine and dihydro-oxazine BACE inhibitors, and compositions and uses thereof Imago Pharmaceuticals, Inc. 11/13/172D 3D TSV
US9505786 59 Substituted annulated triazines and use thereof BAYER PHARMA AKTIENGESELLSCHAFT; BAYER INTELLECTUAL PROPERTY GMBH 11/13/172D 3D TSV
US9522888 952 Substituted bicyclic compounds Bristol-Myers Squibb Company 11/13/172D 3D TSV
US9512130 4 Substituted imidazopyridazines BAYER PHARMA AKTIENGESELLSCHAFT 11/13/172D 3D TSV
US9493441 222 Acyclic cyanoethylpyrazoles as janus kinase inhibitors Merck Sharp & Dohme Corp. 11/06/172D 3D TSV
US9489013 194 C6-azaspiro iminothiadiazine dioxides as bace inhibitors, compositions, and their use Merck Sharp & Dohme Corp. 11/06/172D 3D TSV
US9493440 239 Compounds inhibiting leucine-rich repeat kinase enzyme activity Merck Sharp & Dohme Corp. 11/06/172D 3D TSV
US9493432 214 Cyclopentylbenzamide derivatives and their use for the treatment of psychotic and cognitive disorders Takeda Pharmaceuticals Company Limited 11/06/172D 3D TSV
US9487511 375 Cyclopropanamine compound and use thereof Takeda Pharmaceutical Company Limited 11/06/172D 3D TSV
US9522883 1 Glycosidase inhibitors and uses thereof Alectos Therapeutics Inc.; Merck Sharp & Dohme Corp. 11/06/172D 3D TSV
US9505736 16 Histone deacetylase inhibitors and compositions and methods of use thereof CHDI Foundation, Inc. 11/06/172D 3D TSV
US9493435 182 IRE-1α inhibitors MannKing Corporation 11/06/172D 3D TSV
US9492453 77 Protein kinase B inhibitors AstraZeneca AB 11/06/172D 3D TSV
US9505773 18 Rapamycin analogues and their pharmaceutical use Isomerase Therapeutics Ltd. 11/06/172D 3D TSV
US9504684 11 Syk inhibitors Gilead Sciences, Inc. 11/06/172D 3D TSV
US9487512 159 (Hetero)aryl cyclopropylamine compounds as LSD1 inhibitors Oryzon Genomics S.A. 10/30/172D 3D TSV
US9487490 63 3-cyclohexenyl and cyclohexyl substituted indole and indazole compounds as RORgammaT inhibitors and uses thereof Merck Sharp & Dohme Corp. 10/30/172D 3D TSV
US9481672 253 Bicyclically substituted uracils and the use thereof Bayer Pharma Aktiengesellschaft 10/30/172D 3D TSV
US9487483 128 Complement pathway modulators and uses thereof Novartis AG 10/30/172D 3D TSV
US9505754 4 Compound useful for the treatment of degenerative and inflammatory diseases GALAPAGOS NV 10/30/172D 3D TSV
US9487462 114 Inhibitors of matrix metalloproteinases PharmaHungary 2000 Kft.; TargetEx Kft. 10/30/172D 3D TSV
US9481648 347 Kinase inhibitors Respivert Limited; Topivert Pharma Limited 10/30/172D 3D TSV
US9505743 3 Matrix metalloproteinase inhibitors and methods for the treatment of pain and other diseases TBA 10/30/172D 3D TSV
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US9403827 32 Substituted purinone compounds NOVARTIS AG 07/24/172D 3D TSV
US9403831 42 Triazolopyrazine derivative and use thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY; HANDOK INC. 07/24/172D 3D TSV
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US9394275 191 Diamide compounds having muscarinic receptor antagonist and BETA2 adrenergic receptor agonist activity Theravance Respiratory Company, LLC 07/18/172D 3D TSV
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US9388165 22 Isoquinoline-5-carboxamide derivative having inhibitory activity for protein kinase HANMI PHARM. CO., LTD. 07/17/172D 3D TSV
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US9388210 17 Neuroactive 17(20)-Z-vinylcyano-substituted steroids, prodrugs thereof, and methods of treatment using same WASHINGTON UNIVERSITY 07/17/172D 3D TSV
US9394282 406 Pyrazole carboxamides as Janus kinase inhibitors Merck Sharp & Dohme Corp. 07/17/172D 3D TSV
US9394290 90 Selective CYP11B1 inhibitors for the treatment of cortisol dependent diseases UNIVERSITAET DES SAARLANDES CAMPUS SAARBRUECKEN 07/17/172D 3D TSV
US9394303 31 Small molecule inhibitors of MCL-1 and uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN 07/17/172D 3D TSV
US9393232 171 Substituted 5-(3,5-dimethylisoxazol-4-yl)indoline-2-ones BeiGene, Ltd. 07/17/172D 3D TSV
US9394263 237 Substituted hetero-azepinones F. HOFFMANN-LA ROCHE AG 07/17/172D 3D TSV
US9394250 56 Substituted pyrrolidines as factor xia inhibitors for the treatment thromboembolic diseases ONO PHARMACEUTICAL CO., LTD. 07/17/172D 3D TSV
US9402842 12 Synthesis and use of dual tyrosyl-DNA phosphodiesterase I (Tdp1)—topoisomerase I (Top1) inhibitors Purdue Research Foundation 07/17/172D 3D TSV
US9394293 17 TRPV1 antagonists including dihydroxy substituent and uses thereof Purdue Pharma L.P. 07/17/172D 3D TSV
US9394254 6 Antibiotic and anti-parasitic agents that modulate class II fructose 1,6-bisphosphate aldolase The University of Denver and Regis University 07/10/172D 3D TSV
US9403822 5 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. 07/10/172D 3D TSV
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US9402878 2 Depsipeptide and uses thereof NovoBiotic Pharmaceuticals, LLC 07/10/172D 3D TSV
US9388139 97 Derivatives of celeboxib, use thereof and preparation thereof German University; Southern Research Institute 07/10/172D 3D TSV
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US9365572 65 PI3K and/or mTOR inhibitor Xuanzhu Pharma Co., Ltd. 07/10/172D 3D TSV
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US9388171 28 Serine/threonine kinase inhibitors GENETECH, INC.; ARRAY BIOPHARMA INC. 07/10/172D 3D TSV
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US9388162 146 Substituted morphinans and the use thereof Purdue Pharma L.P. 07/10/172D 3D TSV
US9388136 35 Tert-butyl N-[2-{4-[6-amino-5-(2,4-difluorobenzoyl)-2-oxopyridin-1(2H)-yl]-3,5-difluorophenyl}ethyl]-L-alaninate or a salt, hydrate or solvate thereof Chroma Therapeutics Ltd 07/10/172D 3D TSV
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US9365562 126 1,3 substituted azetidine PDE10 inhibitors Merck Sharp & Dohme Corp. 07/03/172D 3D TSV
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US9365508 26 Aroyl thiourea derivatives University Court of the University of St Andrews; University Court of the University of Dundee 07/03/172D 3D TSV
US9365534 43 Arylated camphenes, processes for their preparation and uses thereof YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. 07/03/172D 3D TSV
US9365529 68 Benzenesulfonamide compounds, method for synthesizing same, and use thereof in medicine as well as in cosmetics GALDERMA RESEARCH & DEVLOPMENT 07/03/172D 3D TSV
US9359371 77 Bicyclic substituted pyrimidine compounds XUANZHU PHARMA CO., LTD. 07/03/172D 3D TSV
US9365511 26 Biphenyl-ethyl-pyrrolidine derivatives as histamine H3 receptor modulators for the treatment of cognitive disorders ARENA PHARMACEUTICALS, INC. 07/03/172D 3D TSV
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US9365502 18 Neuroactive substituted cyclopenta[b]phenanthrenes as modulators for GABA type-A receptors WASHINGTON UNIVERSITY 07/03/172D 3D TSV
US9365539 11 Prolylcarboxypeptidase inhibitors Merck Sharp & Dohme Corp. 07/03/172D 3D TSV
US9365576 279 Pyrrolopyrrolidinone compounds Novartis AG 07/03/172D 3D TSV
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US9359338 366 Cyclopropanecarboxamido-substitute aromatic compounds as anti-tumor agents CROWN BIOSCIENCE INC. (Taiwan) 06/27/172D 3D TSV
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US9388170 7 Substituted aminoquinazolines useful as kinases inhibitors TBA 06/27/172D 3D TSV
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US9359341 11 Aldehyde derivative of substitute oxazolidinones WANBURY LTD. 06/26/172D 3D TSV
US9353089 180 Compositions and methods for the treatment of malaria Saint Louis University; Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences 06/26/172D 3D TSV
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US9359348 11 Cyclopropyl imidazopyridine PDE10 inhibitors Merck Sharp & Dohme Corp. 06/26/172D 3D TSV
US9365558 99 Dihydropyridinone MGAT2 inhibitors Bristol-Myers Squibb Company 06/26/172D 3D TSV
US9359339 19 Glucagon receptor antagonist compounds, compositions containing such compounds and methods of use Merck Sharp & Dohme Corp. 06/26/172D 3D TSV
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US9353104 130 Substituted pyridizinone derivatives as PDE10 inhibitors Merck Sharp & Dohme Corp. 06/26/172D 3D TSV
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US9393245 88 Tricyclic compounds as modulators of TNF-alpha synthesis and as PDE4 inhibitors vTv Therapeutics LLC 06/26/172D 3D TSV
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US9346829 31 5-HT3 receptor antagonists Takeda Phamaceutical Company Limited 06/19/172D 3D TSV
US9353081 132 Bicyclic dihydroquinoline-2-one derivatives Hoffmann-La Roche Inc. 06/19/172D 3D TSV
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US9359301 14 Ethynyl derivatives Hoffmann-La Roche Inc. 06/19/172D 3D TSV
US9346814 250 FAP inhibitors Universiteit Antwerp; Fox Chase Cancer Center 06/19/172D 3D TSV
US9346821 66 Heterocyclic carboxylic acid ester derivative AJINOMOTO CO., INC. 06/19/172D 3D TSV
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US9351965 152 Indazole derivatives useful as ERK inhibitors Merck Sharp & Dohme Corp. 06/19/172D 3D TSV
US9359293 24 Methods of treatment using modulators of SIRT2 CORNELL UNIVERSITY 06/19/172D 3D TSV
US9346786 123 Pyrrolidine compounds Hoffmann-La Roche Inc. 06/19/172D 3D TSV
US9353066 228 Substituted phenyl-Spleen Tyrosine Kinase (Syk) inhibitors Merck Sharp & Dohme Corp.; Merck Canada Inc. 06/19/172D 3D TSV
US9359330 25 Substituted piperidines as sodium channel blockers Purdue Pharma L.P. 06/19/172D 3D TSV
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US9345742 42 Aminostatin derivatives for the treatment of arthrosis MERCK PATENT GMBH 06/12/172D 3D TSV
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US9353067 3 Heterocyclic compounds and uses thereof in the treatment of sexual disorders ATIR Holding S.A. 06/12/172D 3D TSV
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US9353083 4 Oxazetidine derivatives, process for preparing them and use in human medicine and in cosmetics GALDERMA RESEARCH & DEVELOPMENT 06/12/172D 3D TSV
US9358227 12 Pharmaceutical uses of 6-amino quinazoline or 3-cyano quinoline derivatives Jiangsu Hengrui Medicine Co., Ltd.; Shanghai Hengrui Pharmaceutical Co., Ltd. 06/12/172D 3D TSV
US9346839 11 Phosphonate derivatives and methods of use thereof in the treatment of Alzheimer's disease University of Kansas 06/12/172D 3D TSV
US9351973 15 Pyrazolopyridyl compounds as aldosterone synthase inhibitors Merck Sharp & Dohme Corp. 06/12/172D 3D TSV
US9346794 85 Substituted 4-pyridones and their use as inhibitors of neutrophil elastase activity Boehringer Ingelheim International GmbH 06/12/172D 3D TSV
US9346795 186 Substituted sulfonamides useful as antiapoptotic Bcl inhibitors Bristol-Myers Squibb Company 06/12/172D 3D TSV
US9353113 13 Tetrahydrocarboline derivative ONO PHARMACEUTICAL CO., LTD. 06/12/172D 3D TSV
US9346827 11 5-amino-oxazepine and 5-amino-thiazepane compounds as beta secretase antagonists and methods of use Amgen Inc. 06/05/172D 3D TSV
US9346782 60 Alkyl linked quinolinyl modulators of RORγt Janssen Pharmaceutica NV 06/05/172D 3D TSV
US9346818 42 Benzodioxole derivative and preparation method and use thereof Zhejiang Hisun Pharmaceutical Co., Ltd. 06/05/172D 3D TSV
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US9346803 44 Indomethacin analogs for the treatment of castrate-resistant prostate cancer Vanderbilt University; The Trustees of the University of Pennsylvania 06/05/172D 3D TSV
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US9339501 54 17a-hydroxylase/C17,20-lyase inhibitors NOVARTIS AG 05/31/172D 3D TSV
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US9340500 154 Aromatic heterocyclic derivative having TRPV4-inhibiting activity SHIONOGI & CO., LTD. 05/31/172D 3D TSV
US9340537 173 Benzamide derivatives for inhibiting the activity of ABL1, ABL2 and BCR-ABL1 NOVATIS AG 05/31/172D 3D TSV
US9334269 337 Carboxamides as inhibitors of voltage-gated sodium channels AMGEN INC. 05/31/172D 3D TSV
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US9334286 108 Pharmacologically active compounds Cancer Research Technology Limited 05/31/172D 3D TSV
US9340530 84 Preparation and use of bicyclic himbacine derivatives as PAR-1 receptor antagonists Merck Sharp & Dohme Corp. 05/31/172D 3D TSV
US9340507 111 Substituted 4-pyridones and their use as inhibitors of neutrophil elastase activity Boehringer Ingelheim International GmbH 05/31/172D 3D TSV
US9353062 2 Substituted quinolines as bruton's tyrosine kinases inhibitors HangzhouDeRenYuCheng Biotechnology Ltd 05/31/172D 3D TSV
US9334290 152 Substituted tetrahydrocarbazole and carbazole carboxamide compounds Bristol-Myers Squibb Company 05/31/172D 3D TSV
US9340510 245 Tetrahydroisoquinoline derivatives, pharmaceutical compositions and uses thereof Boehringer Ingelheim International GmbH 05/31/172D 3D TSV
US9346822 4 Thienopyrimidine compounds and use thereof Takeda Pharmaceutical Company Limited 05/31/172D 3D TSV
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US9334279 129 Hepatitis C virus inhibitors Bristol-Myers Squibb Company 05/22/172D 3D TSV
US9345740 24 IAP antagonists Bristol-Myers Squibb Company 05/22/172D 3D TSV
US9340521 130 Method for dual inhibition of SGLT1 and SGLT2 using diphenylmethane derivatives GREEN CROSS CORPORATION 05/22/172D 3D TSV
US9340542 20 Propellane-based compounds and the use thereof Purdue Pharma L.P. 05/22/172D 3D TSV
US9340504 6 Pyridine and piperidine derivatives as novel sodium channel blockers Purdue Pharma L.P. 05/22/172D 3D TSV
US9346810 249 Pyrrolopyrimidine compounds and uses thereof HUTCHISON MEDIPHARMA LIMITED 05/22/172D 3D TSV
US9334288 34 Selective β-glucuronidase inhibitors as a treatment for side effects of camptothecin antineoplastic agents The University of North Carolina at Chapel Hill 05/22/172D 3D TSV
US9345789 13 Specific inhibitors and active site probes for legumain The Board of Trustees of the Leland Stanford Junior University 05/22/172D 3D TSV
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US9334268 25 4-amino-imidazoquinoline compounds HOFFMAN-LA ROCHE INC. 05/15/172D 3D TSV
US9340534 4 Compounds and methods for treating ocular diseases ALLERGAN, INC. 05/15/172D 3D TSV
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US9321791 46 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions Boehringer Ingelheim International GmbH 05/08/172D 3D TSV
US9326978 16 A3 adenosine receptor allosteric modulators The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden 05/08/172D 3D TSV
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US9328123 5 Rotenone derivatives and a use thereof Korea Atomic Energy Research Institute 05/08/172D 3D TSV
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US9328112 193 Tetracyclic CDK9 kinase inhibitors AbbVie Inc. 05/03/172D 3D TSV
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US9320741 14 Compositions and methods for treating neoplasia, inflammatory disease and other disorders DANA-FARBER CANCER INSTITUTE, INC. 05/01/172D 3D TSV
US9321743 25 Compositions and methods of inhibiting N-acylethanolamine-hydrolyzing acid amidase The Regents of the University of California; Universita Degli Studi Di Parma; Universita Degli Studi Di Urbino “Carlo Bo” 05/01/172D 3D TSV
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US8987473 72 Ring-fused compound Sato Pharmaceutical Co., Ltd. 09/03/152D 3D TSV
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US8987335 35 Substituted (E)-N′-(1-phenylethylidene)benzohydrazide analogs as histone demethylase inhibitors University of Utah Research Foundation 09/03/152D 3D TSV
US8987445 181 Sulfonamide compounds having TRPM8 antagonistic activity Mitsubishi Tanabe Pharma Corporation 09/03/152D 3D TSV
US8987314 725 Amide, urea or sulfone amide linked benzothiazole inhibitors of endothelial lipase Bristol-Myers Squibb Company 08/25/152D 3D TSV
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US8980932 40 Cancer targeting using carbonic anhydrase isoform IX inhibitors Stichting Maastricht Radiation Oncology “Maastro-Clinic”; Université Montpellier 2 Sciences et Techniques 08/19/152D 3D TSV
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US8987248 26 Substituted piperidines as Par-1 antagonists Bayer Intellectual Property GmbH 08/19/152D 3D TSV
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US8975250 13 5 oxo-5,8-dihydropyrido[2,3-d]pyrimidine derivatives as CaMKII kinase inhibitors for treating cardiovascular diseases SANOFI 08/03/152D 3D TSV
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US8962651 8 Compounds for the treatment of hepatitis C Bristol-Myers Squibb Company 07/22/152D 3D TSV
US8962674 93 Curcumin derivative Tokyo Institute of Technology; Kyoto University 07/22/152D 3D TSV
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US8962630 205 Pyrrolopyrimidine compounds and their uses Novartis AG 07/22/152D 3D TSV
US8962664 3 Selective glycosidase inhibitors and uses thereof Simon Fraser University 07/22/152D 3D TSV
US8962859 12 Spiro-amino-imidazo-fused heterocyclic compounds as beta-secretase modulators and methods of use Amgen Inc. 07/22/152D 3D TSV
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US8962608 1192 Cycloalkylnitrile pyrazole carboxamides as janus kinase inhibitors Merck Sharp & Dohme Corp. 07/15/152D 3D TSV
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US8962612 20 Tetrahydroisoquinoline derivative Astellas Pharma Inc. 07/15/152D 3D TSV
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US8952150 30 Prostaglandin transporter inhibitors and uses thereof Albert Einstein College of Medicine of Yeshiva University 06/29/152D 3D TSV
US8952128 168 Somatostatin-dopamine chimeric analogs Ipsen Pharma S.A.S. 06/29/152D 3D TSV
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US8969568 125 Substituted naphthyridines and their use as medicaments Boehringer Ingelheim Pharma GmbH & Co. KG 06/22/152D 3D TSV
US8969333 6 Therapeutic compositions and methods The Penn State Research Foundation 06/22/152D 3D TSV
US8969394 24 Thiophenecarboxamide derivatives as EP4 receptor ligands Merck Frosst Canada Ltd. 06/22/152D 3D TSV
US8969335 189 Benzonitrile derivatives as kinase inhibitors MERCK PATENT GmbH 06/16/152D 3D TSV
US8940739 190 Compound of a reverse-turn mimetic and a production method and use therefor JW Pharmaceutical Corporation 06/16/152D 3D TSV
US8940893 17 Heteroaromatic compounds as BTK inhibitors Boehringer Ingelheim International GmbH 06/16/152D 3D TSV
US8940748 21 Iminothiadiazine dioxide compounds as BACE inhibitors, compositions, and their use Merck Sharp & Dohme Corp. 06/16/152D 3D TSV
US8940720 77 Macrocycles as factor XIa inhibitors Bristol-Myers Squibb Company 06/16/152D 3D TSV
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US8940744 33 Pyrazolopyrimidine compounds as kinase inhibitors Principia Biopharma Inc. 06/16/152D 3D TSV
US8969341 345 Pyrazolopyrrolidine compounds Novartis AG 06/16/152D 3D TSV
US8969352 164 Substituted 2-azabicycles and their use as orexin receptor modulators Janssen Pharmaceutica NV 06/16/152D 3D TSV
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US8937095 12 Anticancer compounds Boehringer Ingelheim International GmbH 06/08/152D 3D TSV
US8937193 50 Apogossypolone derivatives as anticancer agents Sanford-Burnham Medical Research Institute 06/08/152D 3D TSV
US8937092 22 Aryl or N-heteroaryl substituted methanesulfonamide derivatives as vanilloid receptor ligands Gruenenthal GmbH 06/08/152D 3D TSV
US8940736 142 Imidazotriazinecarbonitriles useful as kinase inhibitors Bristol-Myers Squibb Company 06/08/152D 3D TSV
US8940719 16 Lithocholic acid analogues that inhibit sialyltransferase Academia Sinica 06/08/152D 3D TSV
US8937084 27 Nitrogen containing morphinan derivatives and the use thereof Purdue Pharma L.P. 06/08/152D 3D TSV
US8937068 220 Pyridopyrazine derivatives and their use Zentaris GmbH 06/08/152D 3D TSV
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US8933098 4 Dimethyl-benzoic acid compounds Eli Lilly and Company 06/01/152D 3D TSV
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US8927730 16 Intramolecular hydrogen-bonded nitric oxide synthase inhibitors Northwestern University 06/01/152D 3D TSV
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US8933099 139 Monocyclic pyridine derivative Eisai R&D Management Co., Ltd. 06/01/152D 3D TSV
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US8933040 7 Selective glycosidase inhibitors and uses thereof TBA 06/01/152D 3D TSV
US8933056 55 Soft protease inhibitors and pro-soft forms thereof Trustees of Tufts College 06/01/152D 3D TSV
US8921559 61 4-substituted-cyclohexylamino-4-piperidinyl-acetamide antagonists of CCR2 Janssen Pharmaceutica NV 05/26/152D 3D TSV
US8927520 6 Antibacterial compounds Institut Pasteur; Institut Curie 05/26/152D 3D TSV
US8921397 263 Benzofurane-piperidine compounds Hoffmann-La Roche Inc. 05/26/152D 3D TSV
US8921412 16 C-aryl ansa SGLT2 inhibitors Green Cross Corporation 05/26/152D 3D TSV
US8927534 24 Compounds for the inhibition of integrins and use thereof Shire Orphan Therapies GmbH 05/26/152D 3D TSV
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US8921424 13 Histone deacetylase inhibitors, process for preparation and uses thereof Zhejiang Hisun Pharmaceutical Co. Ltd.; Central South University 05/26/152D 3D TSV
US8921421 2 Inhibitors of dimethylarginine dimethylaminohydrolase Christian-Albrechts-Universitaet Zu Kiel 05/26/152D 3D TSV
US8921389 217 Naphthyridine derivatives as inhibitors of hypoxia inducible factor (HIF) hydroxylase Fibrogen, Inc. 05/26/152D 3D TSV
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US8927536 14 Tetrahydrothiazepine derivative Daiichi Sankyo Company, Limited 05/26/152D 3D TSV
US8653304 10 2,3-dihydro-1H-indene-2-yl urea derivative and pharmaceutical application of same Toray Industries, Inc. 05/18/152D 3D TSV
US8916594 27 5-membered ring heteroaromatic derivatives having NPY Y5 receptor antagonistic activity Shionogi & Co., Ltd. 05/18/152D 3D TSV
US8921404 9 Azole derivatives in the form of lipase and phospholipase inhibitors Sanofi 05/18/152D 3D TSV
US8921370 20 Bicyclo[3.2.1]octyl amide derivatives and uses of same H. Lundbeck A/S 05/18/152D 3D TSV
US8921373 25 Compounds having TRPV1 antagonistic activity and uses thereof Shionogi & Co., Ltd. 05/18/152D 3D TSV
US8653257 5 Dibenzothiazepine derivatives and uses thereof—424 Astrazeneca AB 05/18/152D 3D TSV
US8921364 56 Modulators of calcium release-activated calcium channel Rhizen Pharmaceuticals SA 05/18/152D 3D TSV
US8916600 20 Phenyl and benzodioxinyl substituted indazoles derivatives Astrazeneca AB; Bayer Pharma Aktiengesellschaft 05/18/152D 3D TSV
US8921368 103 Pyrrolopyridazine JAK3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases Bristol-Myers Squibb Company 05/18/152D 3D TSV
US8921319 60 Serine protease inhibitors The Medicines Company (Leipzig) GmbH 05/18/152D 3D TSV
US8653100 267 Tetrahydroisoquinolines, pharmaceutical compositions containing them, and their use in therapy AbbVie Inc.; AbbVie Deutschland GmbH & Co. KG 05/18/152D 3D TSV
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US8912208 4 (4-{4-[5-(benzooxazol-2-ylamino)-pyridin-2-yl]-phenyl}-cyclohexyl)-acetic acid useful for treating or preventing conditions or disorders associated with DGAT1 activity Novartis AG 05/11/152D 3D TSV
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US8912181 115 Bicyclic compound or salt thereof Taiho Pharmaceutical Co., Ltd. 05/11/152D 3D TSV
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US8916553 45 Sulfonamide compounds useful as CYP17 inhibitors Bristol-Myers Squibb Company 05/11/152D 3D TSV
US8912213 12 Synthesis and use of dual tyrosyl-DNA phosphodiesterase I (TDP1)- topoisomerase I (TOP1) inhibitors Purdue Research Foundation 05/11/152D 3D TSV
US8906943 19 Synthetic compounds and methods to decrease nicotine self-administration TBA 05/11/152D 3D TSV
US8895581 96 1H-imidazo[4,5-c]quinolines Boehringer Ingelheim International GmbH 05/04/152D 3D TSV
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US8901315 337 Thienopyrazole derivative having PDE7 inhibitory activity Daiichi Sankyo Company, Limited 05/04/152D 3D TSV
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US8889684 10 Azaindolylphenyl sulfonamides as serine/threonine kinase inhibitors Boehringer Ingelheim International GmbH 04/27/152D 3D TSV
US8889671 80 Compounds and methods for treating bacterial infections AstraZeneca AB 04/27/152D 3D TSV
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US8614195 22 Glycoside derivatives and uses thereof Novartis AG 04/27/152D 3D TSV
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US8889696 65 Substituted pyrido[2,3-d]pyrimidin-7(8H)-ones and therapeutic uses thereof Temple University—Of The Commonwealth System Of Higher Education 04/27/152D 3D TSV
US8889724 7 Tetrazole compounds for reducing uric acid Wellstat Therapeutics Corporation 04/27/152D 3D TSV
US8877733 2 1′-substituted pyrimidine N-nucleoside analogs for antiviral treatment Gilead Sciences, Inc. 04/20/152D 3D TSV
US8884017 21 2-heteroarylcarboxylic acid amides Bayer Intellectual Property GmbH 04/20/152D 3D TSV
US8883759 20 Anti-tumor effect potentiator Taiho Pharmaceutical Co., Ltd. 04/20/152D 3D TSV
US8883784 15 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases AbbVie Inc. 04/20/152D 3D TSV
US8883771 150 Bivalent inhibitors of IAP proteins and therapeutic methods using the same The Regents of the University of Michigan 04/20/152D 3D TSV
US8614213 83 Cyclohexyl amide derivatives and their use as CRF-1 receptor antagonists Novartis AG 04/20/152D 3D TSV
US8883797 12 Metalloenzyme inhibitor compounds Viamet Pharmaceuticals, Inc. 04/20/152D 3D TSV
US8889668 31 Oxadiazole diaryl compounds Merck Serono SA 04/20/152D 3D TSV
US8877741 485 Pyrrolidine derivatives, pharmaceutical compositions and uses thereof Boehringer Ingelheim International GmbH 04/20/152D 3D TSV
US8614220 15 Substituted pyrazolo-quinazoline derivatives, process for their preparation and their use as kinase inhibitors Nerviano Medical Sciences S.r.l. 04/20/152D 3D TSV
US8883846 5 Synthesis of bicyclic compounds and method for their use as therapeutic agents UVic Industry Partnerships Inc. 04/20/152D 3D TSV
US8877798 71 1-aryl-3-azabicyclo[3.1.0]hexanes: preparation and use to treat neuropsychiatric disorders Neurovance, Inc. 04/13/152D 3D TSV
US8877944 96 3-oxo-2,3-dihydro-1H-isoindole-4-carboxamides as PARP inhibitors Nerviano Medical Sciences S.R.L. 04/13/152D 3D TSV
US8877778 285 Benzofurane compounds Hoffmann-La Roche Inc. 04/13/152D 3D TSV
US8877967 42 Compositions and methods for inhibition of cathepsins OXiGENE, Inc.; Baylor University 04/13/152D 3D TSV
US8871738 76 Fused bicyclic oxazolidinone CETP inhibitor Merck Sharp & Dohme Corp. 04/13/152D 3D TSV
US8877795 33 Identification of stabilizers of multimeric proteins The Board of Trustees of the Leland Stanford Junior University 04/13/152D 3D TSV
US8877791 8 Inhibitors of pyruvate kinase and methods of treating disease Beth Israel Deaconess Medical Center, Inc. 04/13/152D 3D TSV
US8871728 49 Non-peptide macrocyclic histone deacetylese (HDAC) inhibitors and methods of making and using thereof Georgia Tech Research Corporation 04/13/152D 3D TSV
US8877757 7 Pyrazine derivatives and use as PI3K inhibitors Merck Serono SA 04/13/152D 3D TSV
US8877775 37 Substituted 2-aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C Boehringer Ingelheim International GmbH 04/13/152D 3D TSV
US8877786 7 Substituted carbamoylmethylamino acetic acid derivatives as novel NEP inhibitors Novartis AG 04/13/152D 3D TSV
US8871778 44 Substituted pyrimidine compounds and their use as SYK inhibitors Genosco; Oscotec, Inc. 04/13/152D 3D TSV
US8865911 180 Compounds and their use as BACE inhibitors Astrazeneca AB 04/06/152D 3D TSV
US8865655 4 Depsipeptides and their therapeutic use Karus Therapeutics Limited 04/06/152D 3D TSV
US8871934 680 Fluorene compound and pharmaceutical use thereof Japan Tobacco Inc. 04/06/152D 3D TSV
US8865706 30 Heteroaryl-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds Pfizer Inc. 04/06/152D 3D TSV
US8871790 475 Heterocyclic modulators of lipid synthesis 3-V Biosciences, Inc. 04/06/152D 3D TSV
US8865662 5 Macrolides and their use Basilea Pharmaceutica AG 04/06/152D 3D TSV
US8865698 105 Method of treatment using substituted pyrazolo[1,5-a]pyrimidine compounds Array BioPharma Inc. 04/06/152D 3D TSV
US8865714 35 Piperazine compound capable of inhibiting prostaglandin D synthase Taiho Pharmaceutical Co., Ltd. 04/06/152D 3D TSV
US8865701 11 Spiropyrrolidine beta-secretase inhibitors for the treatment of alzheimer'S disease Merck Sharp & Dohme Corp. 04/06/152D 3D TSV
US8871783 26 Substituted 2-aza-bicyclo[2.2.1]heptane-3-carboxylic acid (cyano-methyl)-amides inhibitors of cathepsin C Boehringer Ingelheim International GmBh 04/06/152D 3D TSV
US8865726 144 Substituted pyrazolo[1,5-a]pyrimidine compounds as mTOR inhibitors Array BioPharma Inc. 04/06/152D 3D TSV
US8865686 8 Tetracycline compounds as tyrosyl-DNA phosphodiesterase I inhibitors The United States of America, as Represented by the Secretary, Dept. of Health and Human Services 04/06/152D 3D TSV
US8859534 106 2-carboxamide-7-piperazinyl-benzofuran derivatives Acturum Life Science AB 03/16/152D 3D TSV
US8853224 62 Acyclic amine inhibitors of nucleoside phosphorylases and hydrolases Industrial Research Limited; Albert Einstein College of Medicine of Yeshiva University 03/16/152D 3D TSV
US8859596 128 Compounds as cannabinoid receptor ligands AbbVie Inc. 03/16/152D 3D TSV
US8859586 50 Cyclohexyl isoquinolinone compounds Novartis AG 03/16/152D 3D TSV
US8853215 17 Derivatives of N-acyl-N′-phenylpiperazine useful (inter alia) for the prophylaxis or treatment of diabetes Takeda Pharmaceutical Company Limited 03/16/152D 3D TSV
US8853203 366 Diazepinone derivatives Novartis AG 03/16/152D 3D TSV
US8853227 9 Methotrexate adjuvants to reduce toxicity and methods for using the same Tosk, Incorporated 03/16/152D 3D TSV
US8865750 10 Small molecule inhibitors of RGS proteins The Regents of The University of Michigan; The University of Bath 03/16/152D 3D TSV
US8853212 17 Substituted aminotetrahydrothiopyrans and derivatives thereof as dipeptidyl peptidase-IV inhibitors for the treatment of diabetes Merck Sharp & Dohme Corp 03/16/152D 3D TSV
US8853193 170 Thienopyrimidines containing a substituted alkyl group for pharmaceutical compositions Boehringer Ingelheim International GmbH 03/16/152D 3D TSV
US8853206 11 Triazolium salts as PAR1 inhibitors, production thereof, and use as medicaments Sanofi 03/16/152D 3D TSV
US8853226 26 Tricyclic compounds as modulators of TNF-α synthesis and as PDE4 inhibitors High Point Pharmaceuticals, LLC 03/16/152D 3D TSV
US8853258 197 C-linked hydroxamic acid derivatives useful as antibacterial agents Pfizer Inc. 03/09/152D 3D TSV
US8853228 67 Heterocyclic analogs of propargyl-linked inhibitors of dihydrofolate reductase University of Connecticut 03/09/152D 3D TSV
US8853207 12 Heterocyclic pyrazole compounds, method for preparing the same and use thereof Development Center for Biotechnology 03/09/152D 3D TSV
US8846601 142 Melanocortin receptor-specific peptides Palatin Technologies, Inc. 03/09/152D 3D TSV
US8853242 18 Nitrogenous-ring acylguanidine derivative Astellas Pharma Inc. 03/09/152D 3D TSV
US8846658 184 Oxazine derivatives and their use in the treatment of neurological disorders Novartis AG 03/09/152D 3D TSV
US8846698 511 Pyrrolo[2,3-d]pyrimidine tropomysin-related kinase inhibitors Pfizer Limited 03/09/152D 3D TSV
US8846000 35 Radiolabeled PDE10 inhibitors Merck Sharp & Dohme Corp. 03/09/152D 3D TSV
US8846657 356 Substituted imidazopyridines as HDM2 inhibitors Merck Sharp & Dohme Corp. 03/09/152D 3D TSV
US8846656 146 Tetrahydropyrido-pyridine and tetrahydropyrido-pyrimidine compounds and use thereof as C5a receptor modulators Novartis AG 03/09/152D