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Patent: (prefix with "US" like US6078908)
PatentDataCompoundsHGNC
(for human-derived proteins)
Patent TitleOrganizationDepositionDownloads
US20200361871A1 233 229 HGNC:21625 COMPOUNDS TBA 01/13/222D 3D TSV
US11124497 463 179 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. 01/13/222D 3D TSV
US11072585 122 117 HGNC:6666 Fluorinated lysyl oxidase-like 2 inhibitors and uses thereof PHARMAKEA, INC. 01/09/222D 3D TSV
US11071729 29 29 HGNC:4594 1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyridinyl-2′-ones Addex Pharmaceuticals S.A.; Janssen Pharmaceuticals, Inc. 01/07/222D 3D TSV
US11071788 26 21 HGNC:6388 Antibody drug conjugates of kinesin spindel protein (KSP) inhibitors with antiB7H3-antibodies BAYER PHARMA AKTIENGESELLSCHAFT 01/07/222D 3D TSV
US11071721 107 101 Bicyclic amide compounds and methods of use thereof Genentech, Inc. 01/07/222D 3D TSV
US11072617 225 223 Bicyclic sulfones and sulfoxides and methods of use thereof Genentech, Inc. 01/07/222D 3D TSV
US11072611 367 215 HGNC:3357 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders GALAPAGOS NV 01/07/222D 3D TSV
US11072607 46 41 Inhibitors of RIP1 kinase and methods of use thereof Genentech, Inc. 01/07/222D 3D TSV
US11072619 39 13 HGNC:6190 HGNC:6192 HGNC:6193 Pyrazole[1,5-a] pyrimidine derivatives as kinase JAK inhibitors Celon Pharma S.A. 01/07/222D 3D TSV
US11072626 31 31 HGNC:6563 Small molecule inhibitors of Galectin-3 Bristol-Myers Squibb Company 01/07/222D 3D TSV
US11071730 205 201 HGNC:6863 Substituted 6-azabenzimidazole compounds Gilead Sciences, Inc. 01/07/222D 3D TSV
US11072582 277 275 HGNC:4501 Substituted pyrrolidines as G-protein coupled receptor 43 agonists Epics Therapeutics 01/07/222D 3D TSV
US11046714 161 146 HGNC:263 2,2-difluorodioxolo A2A receptor antagonists Merck Sharp & Dohme Corp. 12/28/212D 3D TSV
US11046713 40 19 HGNC:644 Androgen receptor modulating compounds ORION CORPORATION 12/28/212D 3D TSV
US11046725 52 26 HGNC:6561 HGNC:6563 Galactoside inhibitor of galectins GALECTO BIOTECH AB 12/28/212D 3D TSV
US11046712 181 175 HGNC:7056 Glycosidase inhibitors Asceneuron SA 12/28/212D 3D TSV
US11046702 199 198 HGNC:4597 Imidazopyrimidine and imidazotriazine derivative, and pharmaceutical composition comprising the same SK BIOPHARMACEUTICALS CO., LTD. 12/28/212D 3D TSV
US11046710 48 48 HGNC:438 Sulfonamide compounds Daiichi Sankyo Company, Limited; Sanford Burnham Prebys Medical Discovery Institute 12/28/212D 3D TSV
US11046662 48 45 HGNC:12716 HGNC:497 HGNC:18083 HGNC:17961 2-aryl-4-hydroxy-1,3-thiazole derivatives useful as TRPM8-inhibitors in treatment of neuralgia, pain, COPD and asthma DOMPÉ FARMACEUTICI S.P.A. 12/27/212D 3D TSV
US11046691 749 729 2-oxoquinazoline derivatives as methionine adenosyltransferase 2A inhibitors IDEAYA BIOSCIENCES, INC. 12/27/212D 3D TSV
US11046646 10 5 HGNC:3167 HGNC:3165 Alkylphenyl compounds Bristol-Myers Squibb Company 12/27/212D 3D TSV
US11046658 260 127 HGNC:8978 HGNC:8977 Aminopyrazine derivatives as PI3K-γ inhibitors Incyte Corporation 12/27/212D 3D TSV
US11045455 135 26 HGNC:6190 HGNC:2596 HGNC:6192 HGNC:6193 HGNC:6251 HGNC:2637 HGNC:2625 HGNC:12440 Azetidine derivative, preparation method therefor, and use thereof SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. 12/27/212D 3D TSV
US11046649 149 148 HGNC:6059 Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase Board of Regents, The University of Texas System 12/27/212D 3D TSV
US11046671 26 12 HGNC:15631 HGNC:15632 Dihydropyrimidinyl benzazepine carboxamide compounds Hoffmann-La Roche Inc. 12/27/212D 3D TSV
US11046682 39 39 Fused heterocyclic derivatives, their preparation methods thereof and medical uses thereof Beijing Innocare Pharma Tech Co., Ltd 12/27/212D 3D TSV
US11046696 520 198 HGNC:9967 Fused pyrimidine compound or salt thereof Taiho Pharmaceutical Co., Ltd. 12/27/212D 3D TSV
US11046680 486 436 HGNC:339 Heteroaryl-substituted triazoles as APJ receptor agonists AMGEN INC. 12/27/212D 3D TSV
US11046652 39 36 Hydroxamic acids comprising pyrazole moiety and uses thereof HAWAII BIOTECH, INC. 12/27/212D 3D TSV
US11046672 414 70 HGNC:8803 HGNC:3763 HGNC:6307 HGNC:8804 HGNC:3690 HGNC:3688 Indolinones compounds and their use in the treatment of fibrotic diseases RespiVert Limited 12/27/212D 3D TSV
US11046688 205 202 HGNC:12401 Inhibitor compounds Cancer Research Technology Limited 12/27/212D 3D TSV
US11046651 75 35 HGNC:3023 HGNC:5295 HGNC:5182 Piperazine substituted azapine derivatives and uses thereof ALAIRION, INC. 12/27/212D 3D TSV
US11046670 63 27 HGNC:8157 Piperazinyl norbenzomorphan compounds and methods for using the same BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 12/27/212D 3D TSV
US11045448 41 41 HGNC:7010 Piperidines as covalent menin inhibitors THE REGENTS OF THE UNIVERSITY OF MICHIGAN 12/27/212D 3D TSV
US11045457 445 208 HGNC:11330 HGNC:11333 Piperidinyl-3-(aryloxy)propanamides and propanoates Takeda Pharmaceutical Company Limited 12/27/212D 3D TSV
US11046689 289 159 HGNC:6251 HGNC:3467 Selective estrogen receptor down-regulators AstraZeneca AB 12/27/212D 3D TSV
US11046675 8 8 Substituted isoquionline derivatives as immunomudulators Bristol-Myers Squibb Company 12/27/212D 3D TSV
US11046681 33 33 HGNC:12630 Substituted piperidines for the treatment of cancer LES LABORATOIRES SERVIER; VERNALIS (R&D) LTD 12/27/212D 3D TSV
US11046698 1366 1145 TYK2 inhibitors and uses thereof Nimbus Lakshmi, Inc. 12/27/212D 3D TSV
US11046686 30 30 HGNC:17967 Thiadiazole IRAK4 compounds Gilead Sciences, Inc. 12/27/212D 3D TSV
US11066365 273 271 1-cyano-pyrrolidine compounds as USP30 inhibitors Mission Therapeutics Limited 12/23/212D 3D TSV
US11066414 981 964 HGNC:3236 Cot modulators and methods of use thereof Gilead Sciences, Inc. 12/23/212D 3D TSV
US11066413 60 57 HGNC:263 Aminopyrimidine five-membered heterocyclic compound, and intermediate, preparation method, pharmaceutical composition and application thereof GUANGZHOU MAXINOVEL PHARMACEUTICALS CO., LTD. 12/20/212D 3D TSV
US11066409 217 211 HGNC:8537 Bicyclic nitrogen-containing heterocyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. 12/20/212D 3D TSV
US11066404 6 6 HGNC:1771 Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors Incyte Corporation 12/20/212D 3D TSV
US11066406 60 15 Small molecule inhibitors of the JAK family of kinases Janssen Pharmaceutica NV 12/20/212D 3D TSV
US11066396 1453 478 HGNC:4852 HGNC:14064 HGNC:14068 HGNC:13315 3-aryl- heteroaryl substituted 5-trifluoromethyl oxadiazoles as histonedeacetylase 6 (HDAC6) inhibitors MERCK SHARP & DOHME CORP. 12/19/212D 3D TSV
US11065253 471 329 HGNC:9413 Arylquinazolines MERCK PATENT GMBH 12/19/212D 3D TSV
US11065231 55 55 HGNC:17967 Compounds and methods for the targeted degradation of interleukin-1 receptor- associated kinase 4 polypeptides ARVINAS OPERATIONS, INC. 12/19/212D 3D TSV
US11065249 32 26 HGNC:16940 Diacylglycerol acyl transferase 2 inhibitor Pfizer Inc. 12/19/212D 3D TSV
US11066360 104 102 HGNC:6371 Human plasma kallikrein inhibitors BioCryst Pharmaceuticals, Inc. 12/19/212D 3D TSV
US11066363 22 13 HGNC:11305 HGNC:11306 Substituted 6,11-dihydro-5H-benzo[B]carbazoles as inhibitors of ALK and SRPK DANA-FARBER CANCER INSTITUTE, INC. 12/19/212D 3D TSV
US11040966 1982 987 HGNC:4849 HGNC:4848 Benzimidazole-proline derivatives IDORSIA PHARMACEUTICALS LTD 12/14/212D 3D TSV
US11040034 272 135 HGNC:2592 HGNC:2591 Metalloenzyme inhibitor compounds PHASEBIO PHARMACEUTICALS, INC. 12/14/212D 3D TSV
US11041859 70 10 HGNC:17927 HGNC:30402 HGNC:23116 Methods of identifying SENP1 inhibitors CITY OF HOPE 12/14/212D 3D TSV
US11040968 17 17 HGNC:6857 Pyridine derivative as ASK1 inhibitor and preparation method and use thereof TBA 12/14/212D 3D TSV
US11040984 22 11 HGNC:3236 Quinazoline compound for EGFR inhibition MEDSHINE DISCOVERY INC. 12/14/212D 3D TSV
US11040980 33 32 HGNC:1133 Substituted pyrazolo[3,4-d]pyrimidines as kinase inhibitors Principia Biopharma Inc. 12/14/212D 3D TSV
US11040979 20 4 HGNC:6342 Substituted pyrrolo[1,2-b]pyridazines for treating disorders related to KIT and PDGFR Blueprint Medicines Corporation 12/14/212D 3D TSV
US11040967 15 11 HGNC:12440 TYK2 inhibitors, uses, and methods for production thereof Nimbus Lakshmi, Inc. 12/14/212D 3D TSV
US11040970 54 42 HGNC:10935 VMAT2 inhibitor compounds and compositions thereof Neurocrine Biosciences, Inc. 12/14/212D 3D TSV
US11034715 248 146 HGNC:8021 Ectonucleotidase inhibitors and methods of use thereof Calithera Biosciences, Inc. 12/06/212D 3D TSV
US11034717 33 11 Farnesoid X receptor modulators Intercept Pharmaceuticals, Inc. 12/06/212D 3D TSV
US11034991 6 5 HGNC:29079 Methods to determine KDM1A target engagement and chemoprobes useful therefor Oryzon Genomics S.A. 12/06/212D 3D TSV
US11034671 100 99 HGNC:6857 Apoptosis signal-regulating kinase inhibitors and uses thereof SICHUAN HAISCO PHARMACEUTICAL CO., LTD. 12/05/212D 3D TSV
US11033547 127 100 HGNC:9644 Carboxamide-pyrimidine derivatives as SHP2 antagonists Merck Patent GmbH 12/05/212D 3D TSV
US11033539 1210 551 HGNC:1954 HGNC:1953 HGNC:1950 HGNC:1952 HGNC:1951 Compounds of formulas (VII), (VIII), (IX), (XI), (XII), (XIII), and (XIV) as muscarinic receptor 4(M4) antagonists for treating neurological diseases Neurocrine Biosciences, Inc. 12/05/212D 3D TSV
US11034678 17 16 HGNC:16940 Diacylglycerol acyl transferase 2 inhibitors Pfizer Inc. 12/05/212D 3D TSV
US11034699 17 17 HGNC:4596 Ethynyl derivatives Hoffmann-La Roche Inc. 12/05/212D 3D TSV
US11034705 52 52 Fused tricyclic ring derivatives as Src homology-2 phosphate inhibitors Nikang Therapeutics, Inc. 12/05/212D 3D TSV
US11034692 420 390 HGNC:6863 Naphthyridines as inhibitors of HPK1 Genentech, Inc. 12/05/212D 3D TSV
US11034670 70 53 HGNC:270 HGNC:272 Poly-ADP ribose polymerase (PARP) inhibitors Mitobridge, Inc. 12/05/212D 3D TSV
US11034698 115 94 Pyrazolo[ 1,5a]pyrimidine derivatives as IRAK4 modulators Genentech, Inc. 12/05/212D 3D TSV
US11034658 65 65 Pyridinyl pyrazoles as modulators of RORγT Janssen Pharmaceutica NV 12/05/212D 3D TSV
US11034691 995 366 HGNC:3169 HGNC:3167 HGNC:3165 HGNC:14299 HGNC:3170 Sphinogosine-1 -phosphate receptor modulators for treatment of cardiopulmonary disorders THE SCRIPPS RESEARCH INSTITUTE 12/05/212D 3D TSV
US11034661 67 67 HGNC:6059 Substituted N′-hydroxycarbamimidoyl-1,2,5-oxadiazole compounds as indoleamine 2,3-dioxygenase IDO inhibitors Merck Sharp & Dohme Corp. 12/05/212D 3D TSV
US11034694 837 825 HGNC:6863 Substituted isoindolin-1-ones and 2,3-dihydro-1H-pyrrolo[3,4-c]pyridin-1-ones as HPK1 antagonists Nimbus Saturn, Inc. 12/05/212D 3D TSV
US11028054 35 35 HGNC:2867 1, 4, 6-trisubstituted-2-alkyl-1H-benzo[d]imidazole derivatives as dihydroorotate oxygenase inhibitors Merck Patent GmbH 11/29/212D 3D TSV
US11021493 720 166 HGNC:934 HGNC:2529 HGNC:933 1,4-thiazine dioxide and 1,2,4-thiadiazine dioxide derivatives as beta-secretase inhibitors and methods of use Amgen Inc. 11/29/212D 3D TSV
US11026923 606 192 HGNC:8775 HGNC:8774 HGNC:8776 1H-pyrazolo[4,3-b]pyridines as PDE1 inhibitors H. Lundbeck A/S 11/29/212D 3D TSV
US11028101 3 3 HGNC:10894 3-oxa-8-azabicyclo[3.2.1]octane derivatives and their use in the treatment of cancer and hemoglobinopathies CTXT PTY LTD 11/29/212D 3D TSV
US11028093 867 205 HGNC:6190 HGNC:6192 HGNC:6193 HGNC:12440 4,6-substituted-pyrazolo[1,5-a]pyrazines as janus kinase inhibitors ARRAY BIOPHARMA INC.; CELGENE CORPORATION 11/29/212D 3D TSV
US11021475 37 35 Amide-substituted heterocyclic compounds useful as modulators of IL-12, IL-23 and/or IFN alpha responses Bristol-Myers Squibb Company 11/29/212D 3D TSV
US11021511 20 6 Cyclic dinucleotides as sting agonists Janssen Biotech, Inc. 11/29/212D 3D TSV
US11028083 163 145 HGNC:23393 HGNC:18241 Ethanediamine-heterocycle derivatives as inhibitors of protein arginine methyltransferases Board of Regents, The University of Texas System 11/29/212D 3D TSV
US11026937 134 134 HGNC:18368 Heteroaryl inhibitors of PAD4 Padlock Therapeutics, Inc. 11/29/212D 3D TSV
US11028067 15 7 HGNC:12437 HGNC:4623 Heteroarylsulfonyl-substituted pyridines and their use in the treatment of cancer Oblique Therapeutics AB 11/29/212D 3D TSV
US11028058 12 12 HGNC:263 Heterocyclic compounds as adenosine antagonists NUVATION BIO INC. 11/29/212D 3D TSV
US11021478 24 23 HGNC:1232 Indolizine derivatives and their application in medicine KIND PHARMACEUTICAL 11/29/212D 3D TSV
US11028066 97 97 HGNC:29079 Inhibitors of lysine specific demethylase-1 Celgene Quanticel Research, Inc. 11/29/212D 3D TSV
US11021467 405 131 HGNC:8978 HGNC:8980 HGNC:8977 Phosphatidylinositol 3-kinase inhibitors Gilead Sciences, Inc. 11/29/212D 3D TSV
US11026936 57 34 HGNC:8810 Piperidinyl-propanone derivatives Merck Patent GmbH 11/29/212D 3D TSV
US11028041 36 18 HGNC:5253 Second generation GRP94-selective inhibitors University of Kansas 11/29/212D 3D TSV
US11026958 41 36 HGNC:1960 Substituted 6-membered aryl or heteroaryl allosteric modulators of nicotinic acetylcholine receptors Merck Sharp & Dohme Corp. 11/29/212D 3D TSV
US11021481 837 812 HGNC:6863 Substituted isoindolin-1-ones and 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-ones as HPK1 antagonists Nimbus Saturn, Inc. 11/29/212D 3D TSV
US11028085 837 823 HGNC:6863 Substituted isoindolin-1-ones and 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-ones as hpk1 antagonists Nimbus Saturn, Inc. 11/29/212D 3D TSV
US11028092 124 60 HGNC:8795 Substituted pyrazolo[3,4-d]pyrimidines as PDE9 inhibitors Merck Sharp & Dohme Corp. 11/29/212D 3D TSV
US11028080 44 36 Substituted pyrimidines as LRKK2 inhibitors DENALI THERAPEUTICS INC. 11/29/212D 3D TSV
US11028051 14 7 Tetrahydroquinoline-based bromodomain inhibitors St. Jude Children''s Research Hospital 11/29/212D 3D TSV
US11028075 182 90 HGNC:10597 Therapeutic compounds and methods of use thereof Genentech, Inc. 11/29/212D 3D TSV
US11021463 202 145 HGNC:6371 Therapeutic inhibitory compounds ATTUNE PHARMACEUTICALS, INC. 11/29/212D 3D TSV
US11021515 404 207 Therapeutically active compounds and their methods of use Agios Pharmaceuticals, Inc. 11/29/212D 3D TSV
US11028064 146 76 HGNC:6307 Tricyclic heterocyclic derivatives and uses thereof AUCKLAND UNISERVICES LIMITED 11/29/212D 3D TSV
US11028104 83 42 HGNC:12008 HGNC:20692 Xanthine derivatives, their use as a medicament, and pharmaceutical preparations comprising the same MAX-DELBRÜCK-CENTRUM FÜR MOLEKULARE MEDIZIN; FORSCHUNGSVERBUND BERLIN E.V. 11/29/212D 3D TSV
US11028090 505 491 HGNC:13575 [1,2,4]Triazolo[4,3-a]quinoxaline derivative, method for preparing same, and pharmaceutical composition for preventing or treating BET protein-related diseases, containing same as active ingredient Dong Wha Pharm. Co., Ltd.; Korea Research Institute of Chemical Technology 11/29/212D 3D TSV
US11020398 376 299 HGNC:1133 Amino-pyrrolopyrimidinone compounds and methods of use thereof ArQule, Inc. 11/28/212D 3D TSV
US11020381 174 169 HGNC:10597 Biaryloxy derivatives as TTX-S blockers RaQualia Pharma Inc.; XuanZhu Pharma Co., Ltd. 11/28/212D 3D TSV
US11021457 150 150 Class of isoindolone-imide ring-1,3-dione-2-ene compounds, composition and use thereof WIGEN BIOMEDICINE TECHNOLOGY (SHANGHAI) CO., LTD. 11/28/212D 3D TSV
US11020397 70 44 HGNC:12805 HGNC:17989 Compounds and their use for reducing uric acid levels Acquist LLC 11/28/212D 3D TSV
US11020395 154 115 HGNC:339 Cycloalkyl substituted triazole compounds as agonists of the APJ receptor AMGEN INC. 11/28/212D 3D TSV
US11020380 410 396 HGNC:2348 Therapeutic compounds CELGENE QUANTICEL RESEARCH, INC. 11/28/212D 3D TSV
US11021454 44 27 HGNC:12805 Type of aryl benzofuran amidated derivative and medical use thereof CHINA PHARMACEUTICAL UNIVERSITY 11/28/212D 3D TSV
US11014905 114 36 HGNC:3023 HGNC:5286 2,6-disubstituted pyridine derivative SUMITOMO DAINIPPON PHARMA CO., LTD. 11/22/212D 3D TSV
US11014923 152 37 HGNC:3690 HGNC:3691 HGNC:3689 HGNC:3688 Bicyclic heterocycles as FGFR4 inhibitors Incyte Corporation 11/22/212D 3D TSV
US11014911 1035 569 HGNC:1780 HGNC:1771 HGNC:4617 HGNC:1777 HGNC:1722 HGNC:1773 CDK2 inhibitors Pfizer Inc. 11/22/212D 3D TSV
US11014912 68 68 Cyanopyrrolidine derivatives with activity as inhibitors of USP30 MISSION THERAPEUTICS LIMITED 11/22/212D 3D TSV
US11014920 36 35 HGNC:3530 Factor XIIa inhibitors Merck Sharp & Dohme Corp. 11/22/212D 3D TSV
US11014930 78 78 HGNC:9967 Fused pyrimidine compound or salt thereof Taiho Pharmaceutical Co., Ltd. 11/22/212D 3D TSV
US11014909 81 72 HGNC:3020 Heteroaromatic compounds and their use as dopamine D1 ligands Pfizer Inc. 11/22/212D 3D TSV
US11013718 9 9 HGNC:29079 LSD1 inhibitors and medical uses thereof Constellation Pharmaceuticals, Inc. 11/22/212D 3D TSV
US11014929 126 126 HGNC:6863 Pyrazolopyrimidine compounds and uses thereof Incyte Corporation 11/22/212D 3D TSV
US11014913 855 800 Pyridazinones as PARP7 inhibitors Ribon Therapeutics, Inc. 11/22/212D 3D TSV
US11014926 35 30 HGNC:7110 HGNC:7111 Pyrrolo-, pyrazolo-, imidazo-pyrimidine and pyridine compounds that inhibit MNK1 and MNK2 eFFECTOR Therapeutics, Inc. 11/22/212D 3D TSV
US11013745 80 79 Triazolopyrimidine, triazolopyridine compounds, and the composition thereof for treating PRC2-mediated diseases SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES; SUZHOU SUPLEAD LIFE SCIENCES CO., LTD. 11/22/212D 3D TSV
US11014963 205 202 Trifluoromethylpropanamide derivatives as HTRA1 inhibitors Hoffmann-La Roche Inc. 11/22/212D 3D TSV
US11008338 48 25 HGNC:934 HGNC:933 C5-C6-oxacyclic fused iminothiazine dioxide compounds bearing an ether linker as BACE inhibitors, compositions, and their use Merck Sharp & Dohme Corp. 11/15/212D 3D TSV
US11008314 623 155 HGNC:1133 HGNC:6193 HGNC:6171 HGNC:12434 Compounds and methods for modulating interleukin-2-inducible t-cell kinase Corvus Pharmaceuticals, Inc. 11/15/212D 3D TSV
US11008336 22 8 HGNC:10259 HGNC:10258 Compounds useful for inhibiting RORγt Eli Lilly and Company 11/15/212D 3D TSV
US11007200 16 8 HGNC:8157 Cycloalkyl-diamines for the treatment of pain MediSynergics, LLC 11/14/212D 3D TSV
US11008301 42 21 HGNC:3827 HGNC:3826 Piperidinone formyl peptide 2 receptor agonists Bristol-Myers Squibb Company 11/14/212D 3D TSV
US11008312 373 359 Pyridazine derivatives as RORc modulators Genentech, Inc. 11/14/212D 3D TSV
US11008308 435 420 HGNC:29232 Quinazolinones as PARP14 inhibitors Ribon Therapeutics Inc. 11/14/212D 3D TSV
US11008304 85 85 HGNC:6857 Tetrazole containing apoptosis signal-regulating kinase 1 inhibitors and methods of use thereof Enanta Pharmaceuticals, Inc. 11/14/212D 3D TSV
US11000525 30 15 HGNC:7218 HGNC:12015 1-[2-(aminomethyl)benzyl]-2-thioxo-1,2,3,5-tetrahydro-4H-pyrrolo[3,2-d]pyrimidin-4-ones as inhibitors of myeloperoxidase ASTRAZENECA AB 11/08/212D 3D TSV
US11001596 70 8 HGNC:5383 HGNC:5382 7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitors Eli Lilly and Company 11/08/212D 3D TSV
US11001586 178 88 HGNC:7027 HGNC:12446 Alkyl pyrrolopyrimidine analogs and methods of making and using same The University of North Carolina at Chapel Hill 11/08/212D 3D TSV
USRE48547 6 6 HGNC:6027 Aminopyrimidinecarboxamides as CXCR2 modulators Syntrix Biosystems Inc. 11/08/212D 3D TSV
US11001575 923 899 HGNC:6871 Benzolactam compounds as protein kinase inhibitors OTSUKA PHARMACEUTICAL CO., LTD. 11/08/212D 3D TSV
US11000528 26 11 Compound useful for the treatment of degenerative and inflammatory diseases GALAPAGOS NV 11/08/212D 3D TSV
US10995099 93 59 HGNC:85 HGNC:84 Compounds and their uses as ACC inhibitors Nanjing Ruijie Pharmatech Co., Ltd. 11/08/212D 3D TSV
US11000515 25 25 Compounds that interact with the Ras superfamily for the treatment of cancers, inflammatory diseases, rasopathies, and fibrotic disease Shy Therapeutics LLC 11/08/212D 3D TSV
US11001555 22 22 Difluoroketamide derivatives as HTRA1 inhibitors Hoffman-La Roche Inc. 11/08/212D 3D TSV
US11001583 16 16 Dihydropyrrolopyridine inhibitors of ROR-gamma Vitae Pharmaceuticals, LLC 11/08/212D 3D TSV
US11001600 13 13 HGNC:2771 Disubstituted compounds for treatment of medical disorders Achillion Pharmaceuticals, Inc. 11/08/212D 3D TSV
US11001568 170 44 HGNC:29012 HGNC:17071 HGNC:18039 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. 11/08/212D 3D TSV
US11001578 188 92 HGNC:6371 HGNC:6357 N-((HET)arylmethyl)-heteroaryl-carboxamides compounds as plasma kallikrein inhibitors KALVISTA PHARMACEUTICALS LIMITED 11/08/212D 3D TSV
US11001589 51 51 HGNC:3650 Pyrazole derivatives useful as 5-lipoxygenase activating protein (FLAP) inhibitors ASTRAZENECA AB 11/08/212D 3D TSV
US11001595 32 13 HGNC:3763 HGNC:2861 HGNC:6307 HGNC:8804 HGNC:3236 Pyrimidine compounds and pyrimido indole compounds and methods of use Duquesne University of The Holy Spirit 11/08/212D 3D TSV
US11001572 40 10 HGNC:3690 HGNC:3691 HGNC:3689 HGNC:3688 Pyrimidine derivative, method for preparing same and use thereof in medicine TBA 11/08/212D 3D TSV
US11001561 146 136 HGNC:9644 Pyrimidinone derivatives as SHP2 antagonists Merck Patent GmbH 11/08/212D 3D TSV
US11001563 81 81 HGNC:550 SSAO inhibitor TBA 11/08/212D 3D TSV
US10995070 15 15 HGNC:84 Acetyl-CoA carboxylase modulators Monsanto Technology LLC 11/04/212D 3D TSV
US10994015 521 108 HGNC:3430 HGNC:3431 HGNC:3236 EGFR proteolysis targeting chimeric molecules and associated methods of use ARVINAS OPERATIONS, INC.; YALE UNIVERSITY 11/04/212D 3D TSV
US10995072 124 57 HGNC:3538 Inhibitors of protease-activated receptor-2 Heptares Therapeutics Limited 11/04/212D 3D TSV
US10995088 309 162 HGNC:6833 HGNC:6834 HGNC:2671 HGNC:6664 HGNC:6666 Methylamine derivatives as lysysl oxidase inhibitors for the treatment of cancer THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL 11/04/212D 3D TSV
US10995073 253 218 HGNC:8605 HGNC:270 PARG inhibitory compounds Cancer Research Technology Limited 11/04/212D 3D TSV
US10995084 192 116 HGNC:16709 Pyrrolidine derivative KISSEI PHARMACEUTICAL CO., LTD. 11/04/212D 3D TSV
US10995090 21 19 HGNC:7056 Substituted dihydrobenzofuran glycosidase inhibitors Asceneuron SA 11/04/212D 3D TSV
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