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Patent: (prefix with "US" like US6078908)
PatentDataCompoundsHGNC
(for human-derived proteins)		Patent TitleOrganizationDepositionDownloads
US11225479 30 15 HGNC:4852 HGNC:4853 Bicyclic inhibitors of histone deacetylase Alkermes, Inc. 05/22/222D 3D TSV
US11224601 979 813 Compounds that inhibits MCL-1 protein AMGEN INC. 05/22/222D 3D TSV
US11225492 64 18 HGNC:4852 HGNC:1771 HGNC:14064 Heterocycles useful as anti-cancer agents Hangzhou Innogate Pharma Co., Ltd. 05/22/222D 3D TSV
US11225469 284 275 HGNC:8923 Inhibitors of phosphoglycerate dehydrogenase (PHGDH) and uses thereof Whitehead Institute for Biomedical Research; Dana-Farber Cancer Institute, Inc.; The United States of America, as represented by the Secretary, Department of Health and Human Services 05/22/222D 3D TSV
US11225475 20 10 HGNC:4852 HGNC:4853 Substituted pyridines as inhibitors of histone deacetylase Alkermes, Inc. 05/22/222D 3D TSV
US11225486 252 122 HGNC:8978 HGNC:8977 Tertiary alcohols as PI3K-γ inhibitors Incyte Corporation 05/22/222D 3D TSV
US11220505 16 16 HGNC:5302 5-hydroxytryptamine receptor 7 modulators and their use as therapeutic agents Temple University-Of the Commonwealth System of Higher Education 05/14/222D 3D TSV
US11220494 294 137 HGNC:1773 Cyclin dependent kinase inhibitors Pfizer Inc. 05/14/222D 3D TSV
US11220486 362 333 HGNC:122 Inhibitors of low molecular weight protein tyrosine phosphatase and uses thereof LA JOLLA INSTITUTE OF ALLERGY & IMMUNOLOGY; SANFORD BURNHAM PREBYS MEDICAL DISCOVERY INSTITUTE 05/14/222D 3D TSV
US11219618 24 23 HGNC:8974 Pyridylpyridone compounds Sprint Bioscience AB 05/14/222D 3D TSV
US11220510 30 30 HGNC:263 Pyrrole tricyclic compounds as A2A / A2B inhibitors Incyte Corporation 05/14/222D 3D TSV
US11220524 72 71 HGNC:29652 Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) Prelude Therapeutics Incorporated 05/14/222D 3D TSV
US11220509 528 218 Substituted imidazo[1,2-c]pyrimidines as PRC2 inhibitors MIRATI THERAPEUTICS, INC. 05/14/222D 3D TSV
US11220518 98 93 HGNC:9395 Substituted n-pyrimidin-4-yl-3-amino-pyrrolo[3,4-c]pyrazoles as protein kinase C inhibitors PFIZER INC. 05/14/222D 3D TSV
US11220508 218 217 TYK2 inhibitors and uses thereof Nimbus Lakshmi, Inc. 05/14/222D 3D TSV
US11214576 4 4 HGNC:7056 2,3-dihydrofuro[2,3-b]pyridine compounds Eli Lilly and Company 05/08/222D 3D TSV
US11214573 84 42 Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors Incyte Holdings Corporation; Incyte Corporation 05/08/222D 3D TSV
US11214548 26 17 HGNC:2160 HGNC:2159 Cannabinoid receptor modulators Arena Pharmaceuticals, Inc. 05/08/222D 3D TSV
US11214540 151 88 Compositions for treating neurodegenerative diseases Cognition Therapeutics, Inc. 05/08/222D 3D TSV
US11214565 355 341 Compound, compositions, and methods DENALI THERAPEUTICS INC. 05/08/222D 3D TSV
US11213515 25 25 Compounds that interact with the Ras superfamily for the treatment of cancers, inflammatory diseases, rasopathies, and fibrotic disease SHY Therapeutics LLC 05/08/222D 3D TSV
US11214542 212 103 HGNC:9886 HGNC:17071 HGNC:18039 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. 05/08/222D 3D TSV
US11214554 66 52 HGNC:6059 Indoleamine 2,3-dioxygenase inhibitor, method for preparation and use thereof NANJING HUAWE MEDICINE TECHNOLOGY GROUP CO., LTD. 05/08/222D 3D TSV
US11213525 22 21 HGNC:7056 Linear glycosidase inhibitors Asceneuron SA 05/08/222D 3D TSV
US11214557 42 42 HGNC:17038 MAGL inhibitors H. LUNDBECK A/S 05/08/222D 3D TSV
US11213520 16 16 HGNC:1779 Phenylpyrazolylacetamide compounds and derivatives as CDK8/CDK19 inhibitors Boehringer Ingelheim International GmbH 05/08/222D 3D TSV
US11214574 49 49 HGNC:29652 Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) Prelude Therapeutics, Incorporated 05/08/222D 3D TSV
US11214563 53 52 HGNC:4586 Substituted pyrazolo-pyrazines and their use as GluN2B receptor modulators JANSSEN PHARMACEUTICA NV 05/08/222D 3D TSV
US11214566 18 7 Substituted pyridine derivatives useful as C-FMS kinase inhibitors Janssen Pharmaceutica NV 05/08/222D 3D TSV
US11208411 72 32 HGNC:11283 Compositions and methods for treating parasitic diseases The Regents of the University of California; Washington University 05/03/222D 3D TSV
US11208404 192 109 Compounds useful as inhibitors of ALCAT 1 PERENNA PHARMACEUTICALS, INC. 05/03/222D 3D TSV
US11208414 151 80 HGNC:8021 Ectonucleotidase inhibitors and methods of use thereof CALITHERA BIOSCIENCES, INC. 05/03/222D 3D TSV
US11208418 5 5 HGNC:7967 Nitrogenous tricyclic compounds and uses thereof in medicine SUNSHINE LAKE PHARMA CO., LTD. 05/03/222D 3D TSV
US11208696 31 31 HGNC:12401 Prognostic biomarkers for TTK inhibitor chemotherapy NETHERLANDS TRANSLATIONAL RESEARCH CENTER B.V. 05/03/222D 3D TSV
US11208423 20 20 HGNC:8974 Pyridinamine-pyridone and pyrimidinamine- pyridone compounds Sprint Bioscience AB 05/03/222D 3D TSV
US11208403 267 121 HGNC:7027 Pyridone derivatives having tetrahydropyranylmethyl groups Daiichi Sankyo Company, Limited 05/03/222D 3D TSV
US11208416 42 41 HGNC:29652 Selective inhibitors of protein arginine methytransterase 5 (PRMT5) Prelude Therapeutics Incorporated 05/03/222D 3D TSV
US11208422 188 53 HGNC:6283 HGNC:6278 Substituted bridged diazepane derivatives and use thereof as TASK-1 and TASK-3 inhibitors Bayer Pharma Aktiengesellschaft; Bayer Aktiengesellschaft 05/03/222D 3D TSV
US11208415 416 376 HGNC:6943 HGNC:992 HGNC:990 Substituted indole Mcl-1 inhibitors Vanderbilt University 05/03/222D 3D TSV
US11207302 21 20 HGNC:6059 1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase Incyte Corporation; Incyte Holdings Corporation 05/02/222D 3D TSV
US11208377 119 119 HGNC:1607 3,4-disubstituted 3-cyclobutene-1,2-diones and use thereof ALLERGAN, INC. 05/02/222D 3D TSV
US11208388 98 96 HGNC:1133 Certain chemical entities, compositions, and methods NEUPHARMA, INC 05/02/222D 3D TSV
US11207431 131 27 HGNC:4852 HGNC:14065 HGNC:14064 HGNC:19086 HGNC:14063 HGNC:14068 HGNC:14067 HGNC:13315 HGNC:4854 HGNC:4853 HGNC:18128 HDAC6 inhibitors and imaging agents The General Hospital Corporation 05/02/222D 3D TSV
US11208381 336 55 HGNC:8803 HGNC:3763 HGNC:6307 HGNC:8804 HGNC:3690 HGNC:3688 Indole derivatives and their use as protein kinase inhibitors RESPIVERT LIMITED 05/02/222D 3D TSV
US11207312 828 204 Metallo-beta-lactamase inhibitors and methods of use thereof Merck Sharp & Dohme Corp. 05/02/222D 3D TSV
US11208399 224 117 HGNC:5992 HGNC:11892 NLRP3 inflammasome inhibitors Novartis AG 05/02/222D 3D TSV
US11207298 596 595 Substituted 1H-imidazo[4,5-b]pyridin-2(3H)-ones and their use as GLUN2B receptor modulators JANSSEN PHARMACEUTICA NV 05/02/222D 3D TSV
US11208400 567 526 Substituted 6-(1H-pyrazol-1-yl)pyrimidin-4-amine derivatives and uses thereof Bayer Aktiengesellschaft; Bayer Pharma Aktiengesellschaft 05/02/222D 3D TSV
US11208384 2 1 HGNC:12437 HGNC:4623 Sulfinylpyridines and their use in the treatment of cancer Oblique Therapeutics AB 05/02/222D 3D TSV
US11207325 709 243 HGNC:3188 Triazolopyrimidine compounds and uses thereof Novartis AG 05/02/222D 3D TSV
US11203594 66 28 HGNC:1773 Anti-proliferative agents for treating PAH Pfizer Inc. 04/29/222D 3D TSV
US11203595 52 13 Aza-indazole compounds for use in tendon and/or ligament injuries NOVARTIS AG 04/29/222D 3D TSV
US11203574 302 247 HGNC:6371 Human plasma kallikrein inhibitors BioCryst Pharmaceuticals, Inc. 04/29/222D 3D TSV
US11203586 38 37 Iridinesulfonamide compound and use method thereof Chia Tai Tianqing Pharmaceutical Group Co., Ltd.; Lianyungang Runzhong Pharmaceutical Co., Ltd.; Centaurus Biopharma Co., Ltd. 04/29/222D 3D TSV
US11203600 326 281 Kinase inhibitors and uses thereof DENALI THERAPEUTICS INC. 04/29/222D 3D TSV
US11202743 22 14 HGNC:3553 HGNC:2160 HGNC:2159 Personal care compositions comprising fatty acid amide derivatives Conopco, Inc. 04/29/222D 3D TSV
US11203591 304 302 HGNC:6863 Substituted 6-azabenzimidazole compounds Gilead Sciences, Inc. 04/29/222D 3D TSV
US11203571 100 100 HGNC:10582 Sulfonamides as modulators of sodium channels VERTEX PHARMACEUTICALS INCORPORATED 04/29/222D 3D TSV
US11203601 38 19 HGNC:4617 HGNC:4616 Tricyclic compounds as glycogen synthase kinase 3 (GSK3) inhibitors and uses thereof The Broad Institute, Inc.; Biogen MA Inc. 04/29/222D 3D TSV
US11198699 72 56 HGNC:29652 Compounds targeting PRMT5 Aligos Therapeutics, Inc. 04/25/222D 3D TSV
US11198695 577 573 HGNC:7045 Fused ring derivative having MGAT-2 inhibitory activity SHIONOGI & CO., LTD. 04/25/222D 3D TSV
US11197867 468 113 HGNC:6190 HGNC:6192 HGNC:6193 HGNC:12440 Aminopyrimidinyl compounds Pfizer Inc. 04/24/222D 3D TSV
US11197877 16 16 HGNC:10718 Galactopyranosyl-cyclohexyl derivauves as E-selectin antagonists GLYCOMIMETICS. INC. 04/24/222D 3D TSV
US11198681 192 115 HGNC:18368 Heteroaryl inhibitors of PAD4 Padlock Therapeutics, Inc. 04/24/222D 3D TSV
US11198691 188 92 HGNC:6371 HGNC:6357 N-((het)arylmethyl)-heteroaryl-carboxamides compounds as kallikrein inhibitors KalVista Pharmaceuticals Limited 04/24/222D 3D TSV
US11198680 42 13 HGNC:10251 HGNC:10252 Rho kinase inhibitor BA-1049 (R) and active metabolites thereof BioAxone BioSciences, Inc. 04/24/222D 3D TSV
US11192871 30 30 HGNC:5302 5-hydroxytryptamine receptor 7 activity modulators and their method of use Temple University-Of The Commonwealth System of Higher Education 04/17/222D 3D TSV
US11191762 118 111 HGNC:339 Alkyl substituted triazole compounds as agonists of the APJ Receptor AMGEN INC. 04/17/222D 3D TSV
USRE48841 739 377 HGNC:4849 HGNC:4848 Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor modulators Janssen Pharmaceutica NV 04/17/222D 3D TSV
US11191732 9 8 Glutaminase inhibitor discovery and nanoparticle-enhanced delivery for cancer therapy THE JOHNS HOPKINS UNIVERSITY 04/17/222D 3D TSV
US11191765 49 44 HGNC:17270 Heterocyclic compounds for the inhibition of PASK BioEnergenix LLC 04/17/222D 3D TSV
US11192861 302 246 HGNC:6371 Human plasma kallikrein inhibitors BioCryst Pharmaceuticals, Inc. 04/17/222D 3D TSV
US11192850 136 36 HGNC:9642 HGNC:9644 HGNC:9658 N-aryl oxamic acids Purdue Research Foundation 04/17/222D 3D TSV
US11192893 6 6 Pyrazoloquinazolinone antitumor agents The Rockefeller University 04/17/222D 3D TSV
US11192859 43 43 Quinoline compounds as modulators of RAGE activity and uses thereof TBA 04/17/222D 3D TSV
US11192880 4 4 Quinolone compounds as inhibitors of the BCL6 BTB domain protein-protein interaction and/or as BCL6 degraders ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) 04/17/222D 3D TSV
US11192900 103 68 Substituted 1,6-dihydropyridinones and 1,2-dihydroisoquinolinones as bet inhibitors Nuvation Bio Inc. 04/17/222D 3D TSV
US11179399 92 88 HGNC:8974 6-heterocyclyl-4-morpholin-4-ylpyridine-2-one compounds useful for the treatment of cancer and diabetes SPRINT BIOSCIENCE AB 04/10/222D 3D TSV
US11186588 76 73 HGNC:7794 6H-thieno[2,3-e][1,2,4]triazolo[3,4-c][1,2,4]triazepine derivative AYUMI PHARMACEUTICAL CORPORATION 04/10/222D 3D TSV
US11180460 40 40 HGNC:1133 Amino pyrimidine derivatives Novartis AG 04/10/222D 3D TSV
US11180482 48 46 HGNC:6863 Anilinopyrimidines as haematopoietic progenitor kinase 1 (HPK1) inhibitors ARIAD Pharmaceuticals, Inc. 04/10/222D 3D TSV
US11180502 14 14 HGNC:10597 Azaspiro[4.5]decane derivatives and use thereof Purdue Pharma L.P. 04/10/222D 3D TSV
US11179370 8 8 Cannabinoid receptor antagonists/inverse agonists useful for treating disease conditions, including metabolic disorders and cancers Jenrin Discovery, LLC 04/10/222D 3D TSV
US11186587 51 32 HGNC:85 HGNC:84 Compound as ACC inhibitor and use thereof NANJING SANHOME PHARMACEUTICAL CO., LTD. 04/10/222D 3D TSV
US11180455 172 161 HGNC:8156 Compounds for the treatment of pain TBA 04/10/222D 3D TSV
US11186580 8 4 HGNC:8978 HGNC:8977 Crystalline forms of a phosphoinositide 3-kinase (PI3K) inhibitor Incyte Corporation 04/10/222D 3D TSV
US11186589 106 95 HGNC:6853 Cyanoindoline derivatives as NIK inhibitors Janssen Pharmaceutica NV 04/10/222D 3D TSV
US11179397 147 145 HGNC:9644 Imidazopyrimidine derivatives Gilead Sciences, Inc. 04/10/222D 3D TSV
US11179389 39 38 Purine inhibitors of human phosphatidylinositol 3-kinase delta Merck Sharp & Dohme Corp. 04/10/222D 3D TSV
US11180484 295 59 HGNC:3530 HGNC:6371 HGNC:9475 HGNC:3529 HGNC:3535 HGNC:6357 Pyrazole derivatives as plasma kallikrein inhibitors KalVista Pharmaceuticals Limited 04/10/222D 3D TSV
US11186576 141 130 Pyrazolo[1,5-A][1,3,5]triazine and pyrazolo[1,5-A]pyrimidine derivatives as CDK inhibitors Aurigene Discovery Technologies Limited 04/10/222D 3D TSV
US11186590 23 23 HGNC:11331 Somatostatin modulators and uses thereof CRINETICS PHARMACEUTICALS, INC. 04/10/222D 3D TSV
US11186582 564 562 Substituted [1,2,4]triazolo[1,5-a]pyrimidin-7-yl compounds as PDE2 inhibitors Dart Neuroscience, (Cayman) LTD. 04/10/222D 3D TSV
US11180494 197 183 HGNC:6161 Substituted amino acids as integrin inhibitors Pliant Therapeutics, Inc. 04/10/222D 3D TSV
US11180471 516 254 HGNC:6371 HGNC:3529 Substituted oxopyridine derivatives Bayer Pharma Aktiengesellschaft 04/10/222D 3D TSV
US11186578 6 6 HGNC:1133 Substituted pyrrolo[3,2-d]pyrimidines and pyrazolo[4,3-d]pyrimidines as tyrosine kinase inhibitors Shenzhen TargetRx, Inc. 04/10/222D 3D TSV
US11186579 36 35 HGNC:6059 Therapeutic heterocyclic compounds Gilead Sciences, Inc. 04/10/222D 3D TSV
US11186577 549 212 HGNC:8529 HGNC:897 HGNC:895 HGNC:896 Vasopressin receptor antagonists and products and methods related thereto BLACKTHORN THERAPEUTICS, INC. 04/10/222D 3D TSV
US11180503 90 13 HGNC:8783 HGNC:8775 HGNC:8774 HGNC:8776 HGNC:8778 [1,2,4]Triazolo[4,3-A]pyrazin-6(5H)-one derivatives ELI LILLY AND COMPANY 04/10/222D 3D TSV
US11185537 69 27 3-(5-amino-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof Novartis AG 04/09/222D 3D TSV
US11185100 71 50 HGNC:15661 Methods for modulating taste receptors MARS, INCORPORATED 04/09/222D 3D TSV
US11186566 99 64 Modulator of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator Vertex Pharmaceuticals Incorporated 04/09/222D 3D TSV
US11186554 166 164 Non-fused tricyclic compounds VIVACE THERAPEUTICS, INC. 04/09/222D 3D TSV
US11186544 90 45 HGNC:3827 HGNC:3826 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists Bristol-Myers Squibb Company 04/09/222D 3D TSV
US11173161 73 73 HGNC:19995 4-oxo-3,4-dihydro-1,2,3-benzotriazine modulators of GPR139 Takeda Pharmaceutical Company Limited 04/03/222D 3D TSV
US11173144 8 8 HGNC:290 Adrenergic receptor modulating compounds and methods of using the same The Board of Trustees of the Leland Stanford Junior University 04/03/222D 3D TSV
US11174254 34 17 HGNC:1133 HGNC:3236 Aniline-substituted 1,2-dihydropyrrol[3,4-C]pyridin/pyrimidin-3-one derivative and use thereof YANGTZE RIVER PHARMACEUTICAL GROUP CO., LTD.; SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD. 04/03/222D 3D TSV
US11174268 1277 333 HGNC:10593 HGNC:10585 HGNC:10596 Benzenesulfonamide compouds and their use as therapeutic agents Xenon Pharmaceuticals Inc. 04/03/222D 3D TSV
US11174245 334 124 Benzimidazole compounds and derivatives as EGFR inhibitors Boehringer Ingelheim International GmbH 04/03/222D 3D TSV
US11173162 856 187 HGNC:3690 HGNC:3691 HGNC:3689 HGNC:3688 Bicyclic heterocycles as FGFR4 inhibitors Incyte Corporation 04/03/222D 3D TSV
US11173137 85 59 HGNC:281 HGNC:4598 HGNC:4597 HGNC:4596 HGNC:4594 HGNC:5286 HGNC:4593 HGNC:1954 HGNC:1953 HGNC:1950 HGNC:1952 HGNC:4600 Compositions and methods to modulate chloride ion channel activity The Board of Trustees of the Leland Stanford Junior University 04/03/222D 3D TSV
US11174262 18 18 Compounds, compositions and methods Denali Therapeutics Inc. 04/03/222D 3D TSV
US11174252 487 133 HGNC:1780 HGNC:1771 HGNC:1778 HGNC:1777 HGNC:1722 HGNC:1774 HGNC:1773 HGNC:8977 Heterocyclic compounds as kinase inhibitors NUVATION BIO INC. 04/03/222D 3D TSV
US11174248 32 29 Indazolyl-spiro[2.3]hexane-carbonitrile derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof Merck Sharp & Dohme Corp. 04/03/222D 3D TSV
US11174244 634 303 HGNC:4617 HGNC:3091 Isoquinolin-3-yl carboxamides and preparation and use thereof BioSplice Therapeutics, Inc. 04/03/222D 3D TSV
US11174219 7 7 Neprilysin inhibitors Theravance Biopharma R&D IP, LLC 04/03/222D 3D TSV
US11174250 205 126 HGNC:12757 Substituted carboxamides as inhibitors of WDR5 protein-protein binding Propellon Therapeutics Inc. 04/03/222D 3D TSV
US11174232 95 89 Substituted heterocyclyl derivatives as CDK inhibitors Aurigene Discovery Technologies Limited 04/03/222D 3D TSV
US11174264 21 19 TYK2 inhibitors and uses thereof Nimbus Lakshmi, Inc. 04/03/222D 3D TSV
US10988505 14 5 HGNC:16517 Matriptase inhibitors and uses thereof SOCIÉTÉ DE COMMERCIALISATION DES PRODUITS DE LA RECHERCHE APPLIQUÉE SOCPRA SCIENCES SANTÉ ET HUMAINES S.E.C. 03/30/222D 3D TSV
US11136328 48 11 HGNC:4586 HGNC:6251 HGNC:2625 3,3-difluoropiperidine carbamate heterocyclic compounds as NR2B NMDA receptor antagonists Rugen Holdings (Cayman) Limited 03/27/222D 3D TSV
US11136312 309 71 HGNC:11330 HGNC:11331 HGNC:11334 HGNC:11332 HGNC:11333 3,4,5-trisubstituted-1,2,4-triazoles and 3,4,5-trisubstituted-3-thio-1,2,4-triazoles and uses thereof Board of Trustees of the Southern Illinois University 03/27/222D 3D TSV
US11166958 20 20 HGNC:10478 4-pyrazin-2-ylmethyl-morpholine derivatives and the use thereof as medicament Boehringer Ingelheim International GmbH 03/27/222D 3D TSV
US11168095 209 173 HGNC:6857 ASK1 inhibiting agents BIOGEN MA INC. 03/27/222D 3D TSV
US11136340 91 13 HGNC:6190 HGNC:6192 HGNC:6193 HGNC:11393 HGNC:11390 HGNC:9413 HGNC:12401 Amino-triazolopyridine compounds and their use in treating cancer AstraZeneca AB 03/27/222D 3D TSV
US11168102 253 135 Bicyclic heteroaryl compounds and uses thereof Revolution Medicines, Inc. 03/27/222D 3D TSV
US11136315 35 35 HGNC:6027 CXCR2 antagonist MEDSHINE DISCOVERY INC. 03/27/222D 3D TSV
US11168075 35 34 HGNC:12805 Compounds and their use for reducing uric acid levels Acquist LLC 03/27/222D 3D TSV
US11168080 71 67 Dynamin-1-like protein inhibitors Mitobridge, Inc. 03/27/222D 3D TSV
US11136333 19 10 HGNC:76 Functionalized pyrano[2,3-D]pyrimidin-7-one derivatives and methods for their preparation and use The Texas A&M University System 03/27/222D 3D TSV
US11168089 34 34 HGNC:263 Fused pyrimidine derivatives as A2A / A2B inhibitors Incyte Corporation 03/27/222D 3D TSV
US11136320 25 25 HGNC:3691 Fused ring derivative used as FGFR4 inhibitor JACOBIO PHARMACEUTICALS CO., LTD. 03/27/222D 3D TSV
US11136311 221 214 HGNC:6853 Heteroaromatic derivatives as NIK inhibitors Janssen Pharmaceutica NV 03/27/222D 3D TSV
US11168069 12 6 HGNC:12437 HGNC:4623 Heterocyclylsulfonyl-substituted pyridines and their use in the treatment of cancer Oblique Therapeutics AB 03/27/222D 3D TSV
US11135210 8 8 HGNC:17635 Indane-amines as PD-L1 antagonists ChemoCentryx, Inc. 03/27/222D 3D TSV
US11168083 82 66 HGNC:6371 HGNC:9475 HGNC:3528 HGNC:3309 HGNC:3535 Inhibitors of Plasma Kallikrein and uses thereof Takeda Pharmaceutical Company Limited 03/27/222D 3D TSV
US11135207 42 42 HGNC:13709 Inhibitors of dihydroceramide desaturase for treating disease Centaurus Therapeutics 03/27/222D 3D TSV
US11166942 56 55 Inhibitors of integrated stress response pathway PRAXIS BIOTECH LLC 03/27/222D 3D TSV
US11136329 453 118 HGNC:6190 HGNC:6192 HGNC:6193 HGNC:12440 JAK inhibitors VIMALAN BIOSCIENCES, INC. 03/27/222D 3D TSV
US11136327 77 77 HGNC:3529 Macrocycles as factor XIA inhibitors Bristol-Myers Squibb Company 03/27/222D 3D TSV
US11136337 42 42 HGNC:8127 Pyrazole- and indazole-substituted oxadiazolopyridine derivatives for use as ghrelin O-acyl transferase (GOAT) inhibitors Boehringer Ingelheim International GmbH 03/27/222D 3D TSV
US11168088 178 56 HGNC:1771 HGNC:1722 HGNC:1773 Pyridylamino substituted heterotricyclic compounds, and preparation method and pharmaceutical use thereof TBA 03/27/222D 3D TSV
US11168082 96 95 HGNC:29079 Pyrrolo[2,3-C]pyridines and related analogs as LSD-1 inhibitors THE REGENTS OF THE UNIVERSITY OF MICHIGAN 03/27/222D 3D TSV
US11136325 20 7 HGNC:6857 HGNC:6858 Pyrrolopyrimidine and pyrrolopyridine derivatives GALAPAGOS NV 03/27/222D 3D TSV
US11136326 289 96 HGNC:6190 HGNC:7027 HGNC:12446 HGNC:8977 Pyrrolopyrimidine derivatives as TAM inhibitors Incyte Corporation 03/27/222D 3D TSV
US11136296 252 239 HGNC:9600 Substituted N-arylethyl-2-arylquinoline-4-carboxamides and use thereof Bayer Aktiengesellschaft; Bayer Pharma Aktiengesellschaft 03/27/222D 3D TSV
US11136324 38 38 HGNC:6857 Substituted imidazoles as apoptosis signal regulating kinase 1 inhibitors Jiangsu Hansoh Pharmaceutical Group Co., Ltd.; Shanghai Hansoh Biomedical Co., Ltd. 03/27/222D 3D TSV
US11168090 232 115 HGNC:9967 Substituted pyrazolo[1,5-a]pyrazines as RET kinase inhibitors Array BioPharma Inc. 03/27/222D 3D TSV
US11168070 125 125 HGNC:2348 Therapeutic compounds and uses thereof GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC. 03/27/222D 3D TSV
US11168093 183 135 HGNC:10020 Thienopyridine inhibitors of RIPK2 Celgene Corporation 03/27/222D 3D TSV
US11136336 22 22 HGNC:497 Thienopyrimidones Boehringer Ingelheim International GmbH 03/27/222D 3D TSV
US11161839 234 186 2-quinolone derived inhibitors of BCL6 The Institute of Cancer Research: Royal Cancer Hospital; Cancer Research Technology Limited 03/20/222D 3D TSV
US11161835 15 15 HGNC:12805 Compounds and their use for reducing uric acid levels Acquist LLC 03/20/222D 3D TSV
US11161844 99 37 HGNC:18618 Cyclic substituted imidazo[4,5-c]quinoline derivatives PFIZER INC. 03/20/222D 3D TSV
US11161850 128 113 HGNC:263 Fused pyrazine derivatives as A2A / A2B inhibitors Incyte Corporation 03/20/222D 3D TSV
US11161838 26 13 HGNC:8978 HGNC:8977 Heterocyclic derivatives as PI3K inhibitors Incyte Corporation 03/20/222D 3D TSV
US11161815 65 33 HGNC:12437 HGNC:4623 Hydrocarbylsulfonyl-substituted pyridines and their use in the treatment of cancer Oblique Therapeutics AB 03/20/222D 3D TSV
US11161854 111 77 Indazolyl-spiro[2.2]pentane-carbonitrile derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof Merck Sharp & Dohme Corp. 03/20/222D 3D TSV
US11161849 6 6 HGNC:497 Inhibiting the transient receptor potential al ion channel Eli Lilly and Company 03/20/222D 3D TSV
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