BDBM50415407 CHEMBL612138

SMILES COc1cccc(c1)-c1noc(C)c1C(=O)N(C)c1ccc(Cl)cc1

InChI Key InChIKey=CCCPDKSLSUVEBG-UHFFFAOYSA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50415407   

TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50415407(CHEMBL612138)
Show SMILES COc1cccc(c1)-c1noc(C)c1C(=O)N(C)c1ccc(Cl)cc1
Show InChI InChI=1S/C19H17ClN2O3/c1-12-17(19(23)22(2)15-9-7-14(20)8-10-15)18(21-25-12)13-5-4-6-16(11-13)24-3/h4-11H,1-3H3
Affinity DataEC50:  1nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair