BDBM20510 (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide::AMG 9810::AMG9810::CHEMBL195789::trans-Cinnamide

SMILES: CC(C)(C)c1ccc(\C=C\C(=O)Nc2ccc3OCCOc3c2)cc1

InChI Key: InChIKey=GZTFUVZVLYUPRG-UHFFFAOYSA-N

Data: 8 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 20510   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	79	n/a	n/a	n/a	n/a	7.4	22
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Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	350	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	294	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	93	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20510 (AMG9810 | (2E)-3-(4-tert-butylphenyl)-N-(2,3-dihyd...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	86	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair