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BDBM100365 US10189794, Compound I-209::US10618902, Compound I-209::US10774052, Compound I-209::US9695132, I-209

SMILES: COc1ccc(cc1)N1Cc2cnc(NC3COCC3NC(=O)C=C)nc2N(C)C1=O

InChI Key: InChIKey=NJDHFNVZECIIBG-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 100365
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Fibroblast growth factor receptor 4 (Human)	BDBM100365 (US9695132, I-209 \| US10189794, Compound I-209 \| US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	7.5	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100365 (US9695132, I-209 \| US10189794, Compound I-209 \| US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100365 (US9695132, I-209 \| US10189794, Compound I-209 \| US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	5.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100365 (US9695132, I-209 \| US10189794, Compound I-209 \| US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair