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BDBM16128 4-(trifluoromethyl)benzene-1-guanidine::CHEMBL43961::phenylguanidine 2

SMILES: NC(=N)Nc1ccc(cc1)C(F)(F)F

InChI Key: InChIKey=IUNFWMWQNWQIFS-UHFFFAOYSA-N

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 16128
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Urokinase-type plasminogen activator (Human)	BDBM16128 (4-(trifluoromethyl)benzene-1-guanidine \| CHEMBL439...) Show SMILES Show InChI	GoogleScholar	UniChem		6.00E+3	-7.41	n/a	n/a	n/a	n/a	n/a	8.1	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Urokinase-type plasminogen activator (Human)	BDBM16128 (4-(trifluoromethyl)benzene-1-guanidine \| CHEMBL439...) Show SMILES Show InChI	GoogleScholar	UniChem		6.49E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Urokinase-type plasminogen activator (Human)	BDBM16128 (4-(trifluoromethyl)benzene-1-guanidine \| CHEMBL439...) Show SMILES Show InChI	GoogleScholar	UniChem		6.49E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine protease 1 (Bovine)	BDBM16128 (4-(trifluoromethyl)benzene-1-guanidine \| CHEMBL439...) Show SMILES Show InChI	GoogleScholar	UniChem		6.31E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine protease 1 (Bovine)	BDBM16128 (4-(trifluoromethyl)benzene-1-guanidine \| CHEMBL439...) Show SMILES Show InChI	GoogleScholar	UniChem		6.31E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Plasminogen (Human)	BDBM16128 (4-(trifluoromethyl)benzene-1-guanidine \| CHEMBL439...) Show SMILES Show InChI	GoogleScholar	UniChem		<1.00E+7	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair