BDBM164135 US9062078, 265::US9475819, 265::US9637496, 265::US9695183, 265

SMILES: Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1cnccn1

InChI Key: InChIKey=CVFCIDFMYLGEOP-UHFFFAOYSA-N

Data: 12 KI

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 12 hits for monomerid = 164135   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Orexin/Hypocretin receptor type 1 (Rat)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		20	-9.76	n/a	n/a	n/a	n/a	n/a	n/a	4
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Rat)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Rat)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		20	-11.0	n/a	n/a	n/a	n/a	n/a	n/a	40
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Rat)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		20	-9.76	n/a	n/a	n/a	n/a	n/a	n/a	4
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		23	-9.68	n/a	n/a	n/a	n/a	n/a	n/a	4
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		23	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		23	-9.68	n/a	n/a	n/a	n/a	n/a	n/a	4
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin/Hypocretin receptor type 1 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		23	-9.68	n/a	n/a	n/a	n/a	n/a	n/a	4
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin receptor type 2 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		188	-9.63	n/a	n/a	n/a	n/a	n/a	n/a	40
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin receptor type 2 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		188	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin receptor type 2 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		188	-9.63	n/a	n/a	n/a	n/a	n/a	n/a	40
TBA									Citation and Details
					More data for this Ligand-Target Pair
Orexin receptor type 2 (Human)	BDBM164135 (US9475819, 265 | US9062078, 265 | US9695183, 265 |...) Show SMILES Show InChI	GoogleScholar	UniChem		188	-9.63	n/a	n/a	n/a	n/a	n/a	n/a	40
TBA									Citation and Details
					More data for this Ligand-Target Pair