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BDBM176223 US10047103, 256::US9688695, 256

SMILES: COc1cc(OCc2csc(NCC3CCCO3)n2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1

InChI Key: InChIKey=CKPKXLBOVYLIRO-UHFFFAOYSA-N

Data: 1 IC50 3 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 176223
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Proteinase-activated receptor 4 (Human)	BDBM176223 (US9688695, 256 \| US10047103, 256) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	7.80	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Human)	BDBM176223 (US9688695, 256 \| US10047103, 256) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	>3.00E+3	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Human)	BDBM176223 (US9688695, 256 \| US10047103, 256) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	7.80	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Prothrombin (Human)	BDBM176223 (US9688695, 256 \| US10047103, 256) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>3.00E+3	n/a	n/a	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair