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BDBM186936 US9079895, 24s

SMILES: COc1cccc(OC[C@@H]2CN(CC(=O)N3CCc4ccccc34)CCO2)c1

InChI Key: InChIKey=KJWABLDVLWKPKR-UHFFFAOYSA-N

Data: 4 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 186936
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 1A (Mouse)	BDBM186936 (US9079895, 24s) Show SMILES Show InChI	GoogleScholar	UniChem		371	n/a	n/a	n/a	n/a	n/a	n/a	7.4	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2B (Mouse)	BDBM186936 (US9079895, 24s) Show SMILES Show InChI	GoogleScholar	UniChem		1.65E+3	n/a	n/a	n/a	n/a	n/a	n/a	7.4	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2A (Mouse)	BDBM186936 (US9079895, 24s) Show SMILES Show InChI	GoogleScholar	UniChem		1.95E+3	n/a	n/a	n/a	n/a	n/a	n/a	7.4	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 1B (Mouse)	BDBM186936 (US9079895, 24s) Show SMILES Show InChI	GoogleScholar	UniChem		4.83E+3	n/a	n/a	n/a	n/a	n/a	n/a	7.4	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair