BDBM210983 US9247759, 4-17
SMILES COc1ccc(cc1)C(=O)Nc1cnn(Cc2c(C)noc2C)c1
InChI Key InChIKey=IILSWFQBVNCJBK-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 210983
Affinity DataIC50: 700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair