BDBM211037 US9247759, 4-72
SMILES Cc1noc(C)c1Cn1cc(NC(=O)c2ccc3ocnc3c2)cn1
InChI Key InChIKey=AXBKOAZUUQDADD-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 211037
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair