BDBM211259 US9247759, 10-7
SMILES COC(=O)c1cccc(CN2CC(=O)N(C2=O)c2cnn(Cc3c(C)noc3C)c2)c1
InChI Key InChIKey=BRVFGECVAWZHNJ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 211259
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair