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BDBM249306 US10017501, Compound 1020-104::US9458145, 1020-104

SMILES: Cc1noc(C)c1-c1cc(c2nc([nH]c2c1)C1CC1)C(O)(c1ccccn1)c1ccccn1

InChI Key: InChIKey=CMSUJGUHYXQSOK-UHFFFAOYSA-N

Data: 2 KI 2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 249306
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Bromodomain-containing protein 4 [75-147] (Human)	BDBM249306 (US9458145, 1020-104 \| US10017501, Compound 1020-10...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.20	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [368-440] (Human)	BDBM249306 (US9458145, 1020-104 \| US10017501, Compound 1020-10...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	11.7	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [75-147] (Human)	BDBM249306 (US9458145, 1020-104 \| US10017501, Compound 1020-10...) Show SMILES Show InChI	GoogleScholar	UniChem		7.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [368-440] (Human)	BDBM249306 (US9458145, 1020-104 \| US10017501, Compound 1020-10...) Show SMILES Show InChI	GoogleScholar	UniChem		11.7	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair