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BDBM250301 US10501411, Example 211::US11697636, Example 211::US9452980, 211

SMILES: COC(=O)c1ccc(COc2ccc(cc2)C(=O)Nc2ccc(cc2)C2CNCCO2)cc1

InChI Key: InChIKey=BWCYBKOHQWMMEA-UHFFFAOYSA-N

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 250301
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Trace amine-associated receptor 1 (Rat)	BDBM250301 (US9452980, 211 \| US10501411, Example 211 \| US11697...) Show SMILES Show InChI	GoogleScholar	UniChem		0.900	-12.8	n/a	n/a	n/a	n/a	n/a	7.4	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Trace amine-associated receptor 1 (Rat)	BDBM250301 (US9452980, 211 \| US10501411, Example 211 \| US11697...) Show SMILES Show InChI	GoogleScholar	UniChem		0.900	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Trace amine-associated receptor 1 (Rat)	BDBM250301 (US9452980, 211 \| US10501411, Example 211 \| US11697...) Show SMILES Show InChI	GoogleScholar	UniChem		0.900	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Trace amine-associated receptor 1 (Mouse)	BDBM250301 (US9452980, 211 \| US10501411, Example 211 \| US11697...) Show SMILES Show InChI	GoogleScholar	UniChem		4	-11.9	n/a	n/a	n/a	n/a	n/a	7.4	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Trace amine-associated receptor 1 (Mouse)	BDBM250301 (US9452980, 211 \| US10501411, Example 211 \| US11697...) Show SMILES Show InChI	GoogleScholar	UniChem		4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Trace amine-associated receptor 1 (Mouse)	BDBM250301 (US9452980, 211 \| US10501411, Example 211 \| US11697...) Show SMILES Show InChI	GoogleScholar	UniChem		4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair