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BDBM25113 5-(4-aminophenyl)thieno[2,3-d]pyrimidin-4-amine::thienopyrimidine analogue, 1

SMILES: Nc1ccc(cc1)-c1csc2ncnc(N)c12

InChI Key: InChIKey=HKNAOIMDZKNBSU-UHFFFAOYSA-N

Data: 4 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 25113
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Serine/threonine-protein kinase PLK4 (Human)	BDBM25113 (5-(4-aminophenyl)thieno[2,3-d]pyrimidin-4-amine \| ...) Show SMILES Show InChI	GoogleScholar	UniChem		9.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Human)	BDBM25113 (5-(4-aminophenyl)thieno[2,3-d]pyrimidin-4-amine \| ...) Show SMILES Show InChI	GoogleScholar	UniChem		>2.00E+4	>-6.34	n/a	n/a	n/a	n/a	n/a	7.5	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK2 (Human)	BDBM25113 (5-(4-aminophenyl)thieno[2,3-d]pyrimidin-4-amine \| ...) Show SMILES Show InChI	GoogleScholar	UniChem		>2.00E+4	>-6.34	n/a	n/a	n/a	n/a	n/a	7.5	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK3 (Human)	BDBM25113 (5-(4-aminophenyl)thieno[2,3-d]pyrimidin-4-amine \| ...) Show SMILES Show InChI	GoogleScholar	UniChem		>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair