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BDBM26179 2,4-dianilino pyrimidine, 36::3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}benzamide::GTC000110A

SMILES: NC(=O)c1cccc(Nc2nccc(Nc3cccc4[nH]ncc34)n2)c1

InChI Key: InChIKey=NQHLFCVNEBJHOT-UHFFFAOYSA-N

Data: 2 KI 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 26179
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Proto-oncogene tyrosine-protein kinase LCK (Mouse)	BDBM26179 (3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	100	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase SYK [355-635] (Human)	BDBM26179 (3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	533	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase (Human)	BDBM26179 (3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	509	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase (Human)	BDBM26179 (3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.44E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase (Human)	BDBM26179 (3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}b...) Show SMILES Show InChI	GoogleScholar	UniChem		48	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase (Human)	BDBM26179 (3-{[4-(1H-indazol-4-ylamino)pyrimidin-2-yl]amino}b...) Show SMILES Show InChI	GoogleScholar	UniChem		1.60E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair