BDBM263481 (s)?n-(1-(4-methoxyphenyl)ethyl)-2-(4-oxo-6-(trifluoromethyl)benzo[d][1,2,3]triazin-3 (4h)-yl)acetamide::US10561662, Example 44::US11173161, EX 44::US9556130, test 44
SMILES COc1ccc(cc1)[C@H](C)NC(=O)Cn1nnc2ccc(cc2c1=O)C(F)(F)F
InChI Key InChIKey=FUWMUUAHZQTWMB-NSHDSACASA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 263481
Affinity DataKi: 2.53E+3nM ΔG°: -7.09kcal/molepH: 7.4 T: 2°CAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
Affinity DataKi: 2.53E+3nMAssay Description:Membranes were removed from −80° C., thawed and diluted in cold radioligand assay buffer (20 mM HEPES pH 7.4/5 mM MgCl2/1 mM CaCl2/Roche protea...More data for this Ligand-Target Pair
Affinity DataKi: 2.53E+6nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair