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BDBM315705 US10172859, Example 129::US10172859, Example 137::US10172859, Example 225::US10172859, Example 239::US10172859, Example 244::US10172859, Example 262::US11065253, Example 262::US9732094, Example 262::[2,4-Difluoro-5-(7- morpholin-4-yl- quinazolin-4-yl)- phenyl]-(6- methoxy- pyridazin-3-yl)- methanol (Ena 2)see racemate

SMILES: COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1

InChI Key: InChIKey=MOWXJLUYGFNTAL-UHFFFAOYSA-N

Data: 10 KI  15 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 25 hits for monomerid = 315705   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 18.5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 19n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 18.5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 18.5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
n/an/a<3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
1.25E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
1.25E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
2.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
2.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
2.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
2.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
>2.50E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
>2.50E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
>2.50E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM315705
PNG
(US10172859, Example 244 | US10172859, Example 137 ...)
GoogleScholar
UniChem
>2.50E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair