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BDBM50008992 2-Pyridin-3-ylmethyl-1,2-dihydro-indazol-3-one::CHEMBL3144579

SMILES: O=c1n(Cc2cccnc2)[nH]c2ccccc12

InChI Key: InChIKey=SKZAIZCDZYPCRF-UHFFFAOYSA-N

Data: 3 IC50 1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50008992
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Prostaglandin G/H synthase 1/2 (Rat)	BDBM50008992 (2-Pyridin-3-ylmethyl-1,2-dihydro-indazol-3-one \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Polyunsaturated fatty acid 5-lipoxygenase (Human)	BDBM50008992 (2-Pyridin-3-ylmethyl-1,2-dihydro-indazol-3-one \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	1.33E+4	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Polyunsaturated fatty acid 5-lipoxygenase (Rat)	BDBM50008992 (2-Pyridin-3-ylmethyl-1,2-dihydro-indazol-3-one \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Polyunsaturated fatty acid 5-lipoxygenase (Human)	BDBM50008992 (2-Pyridin-3-ylmethyl-1,2-dihydro-indazol-3-one \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair