BDBM50049785 1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-{4-methyl-3-[methyl-(1H-tetrazol-5-yl)-amino]-phenyl}-urea::CHEMBL168253

SMILES CN(c1nnn[nH]1)c1cc(NC(=O)N[C@@H]2N=C(C3CCCCC3)c3ccccc3N(C)C2=O)ccc1C

InChI Key InChIKey=BIOMOYOMCAMNGH-QHCPKHFHSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50049785   

TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049785(1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049785(1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed