BDBM50058963 Ac-His-DPhe-Arg-DTrp-NH2::Ac-His-DPhe-DArg-DTrp-NH2::CHEMBL433296

SMILES CC(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(N)=O

InChI Key InChIKey=DFCJPPDAOZROBS-AUAHOFGGSA-N

Data  4 IC50  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50058963   

TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]NDP-MSH from Melanocortin 3 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]NDP-MSH from Melanocortin 5 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]NDP-MSH from Melanocortin 4 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataEC50:  2.44E+3nMAssay Description:Functional activity at the mouse melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataEC50:  61.3nMAssay Description:Functional activity at the mouse melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataEC50:  97.2nMAssay Description:Functional activity at the mouse melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataEC50:  154nMAssay Description:Functional activity at the mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058963(Ac-His-DPhe-Arg-DTrp-NH2 | Ac-His-DPhe-DArg-DTrp-N...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]NDP-MSH from Melanocortin 1 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed