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BDBM50132976 2-[4-(4-Fluoro-phenyl)-1H-pyrazol-3-yl]-6-methyl-pyridine::CHEMBL125846

SMILES: Cc1cccc(n1)-c1n[nH]cc1-c1ccc(F)cc1

InChI Key: InChIKey=VJPFFCRCUZQGJL-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50132976
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
TGF-beta receptor type-1 (Human)	BDBM50132976 (2-[4-(4-Fluoro-phenyl)-1H-pyrazol-3-yl]-6-methyl-p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	41	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132976 (2-[4-(4-Fluoro-phenyl)-1H-pyrazol-3-yl]-6-methyl-p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	139	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132976 (2-[4-(4-Fluoro-phenyl)-1H-pyrazol-3-yl]-6-methyl-p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132976 (2-[4-(4-Fluoro-phenyl)-1H-pyrazol-3-yl]-6-methyl-p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair