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BDBM50133002 (1H-Indol-2-yl)-piperazin-1-yl-methanone::(1H-indol-2-yl)(piperazin-1-yl)methanone::CHEMBL129660

SMILES: O=C(N1CCNCC1)c1cc2ccccc2[nH]1

InChI Key: InChIKey=FIVCRRVYLAXYFC-UHFFFAOYSA-N

Data: 4 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50133002
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histamine H4 receptor (Human)	BDBM50133002 ((1H-Indol-2-yl)-piperazin-1-yl-methanone \| (1H-ind...) Show SMILES Show InChI	GoogleScholar	UniChem		4.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM50133002 ((1H-Indol-2-yl)-piperazin-1-yl-methanone \| (1H-ind...) Show SMILES Show InChI	GoogleScholar	UniChem		38	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM50133002 ((1H-Indol-2-yl)-piperazin-1-yl-methanone \| (1H-ind...) Show SMILES Show InChI	GoogleScholar	UniChem		38	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM50133002 ((1H-Indol-2-yl)-piperazin-1-yl-methanone \| (1H-ind...) Show SMILES Show InChI	GoogleScholar	UniChem		9.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair