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BDBM50143680 8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decan-7-one::CHEMBL299454

SMILES: Clc1ccccc1N1CCN(CCN2CCC3(CCCC3)CC2=O)CC1

InChI Key: InChIKey=BYHQOSOPNSLUAD-UHFFFAOYSA-N

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50143680
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Alpha-1D adrenergic receptor (Rat)	BDBM50143680 (8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8...) Show SMILES Show InChI	GoogleScholar	UniChem		0.540	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 1A (Human)	BDBM50143680 (8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8...) Show SMILES Show InChI	GoogleScholar	UniChem		1.06	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-1B adrenergic receptor (Human)	BDBM50143680 (8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8...) Show SMILES Show InChI	GoogleScholar	UniChem		35.9	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-1A adrenergic receptor (Human)	BDBM50143680 (8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8...) Show SMILES Show InChI	GoogleScholar	UniChem		70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-1A adrenergic receptor (Human)	BDBM50143680 (8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8...) Show SMILES Show InChI	GoogleScholar	UniChem		71	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-1A adrenergic receptor (Rat)	BDBM50143680 (8-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-8...) Show SMILES Show InChI	GoogleScholar	UniChem		87.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair