BDBM50168088 CHEMBL3797325

SMILES CC(CC(O)=O)NC(=O)c1ccc(cc1)C(C)n1nc(cc1-c1ccc2OCCc2c1)-c1cc(Cl)cc(Cl)c1

InChI Key InChIKey=BRBJPXYNJFCDKY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50168088   

TargetGlucagon receptor(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50168088(CHEMBL3797325)
Affinity DataIC50:  1.81E+4nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHO-K1 cells after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50168088(CHEMBL3797325)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at wild type human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation incu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed