BDBM50177277 CHEMBL202563::N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-3-p-tolylacrylamide

SMILES CN(C)CCN(C)c1cc(C)c2cc(NC(=O)\C=C\c3ccc(C)cc3)ccc2n1

InChI Key InChIKey=ACSLJTYYCFGVHX-JLHYYAGUSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50177277   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50177277(CHEMBL202563 | N-(2-((2-(dimethylamino)ethyl)(meth...)
Affinity DataIC50:  478nMAssay Description:Displacement of [3H]myo-inositol from human MCH1 receptor expressed in CHO cell by IP3 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50177277(CHEMBL202563 | N-(2-((2-(dimethylamino)ethyl)(meth...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]MCH from human MCH1 receptor expressed in CHO cell by WC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50177277(CHEMBL202563 | N-(2-((2-(dimethylamino)ethyl)(meth...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human MCH1 receptor by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed