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BDBM50184483 1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo-[1,2-b]pyrazol-3-yl]-1H-benzoimidazole::CHEMBL204966

SMILES: Cc1cccc(n1)-c1nn2CCCc2c1-c1ccc2ncn(C)c2c1

InChI Key: InChIKey=SXNCFFITOIFUMU-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50184483
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mitogen-activated protein kinase kinase kinase 20 (Human)	BDBM50184483 (1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.34E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50184483 (1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	22	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50184483 (1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	29	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-2 (Human)	BDBM50184483 (1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	668	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair