BDBM50248108 CHEMBL517282::N-(3,5-difluorophenylsulfonyl)-3-(1-methyl-4-(naphthalen-2-yloxy)-1H-indol-3-yl)acrylamide

SMILES Cn1cc(\C=C\C(=O)NS(=O)(=O)c2cc(F)cc(F)c2)c2c(Oc3ccc4ccccc4c3)cccc12

InChI Key InChIKey=ALGHFVPGLKKOKU-ZRDIBKRKSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50248108   

TargetProstaglandin E2 receptor EP3 subtype(Human)
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50248108(CHEMBL517282 | N-(3,5-difluorophenylsulfonyl)-3-(1...)
Affinity DataIC50:  157nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of 10% human serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50248108(CHEMBL517282 | N-(3,5-difluorophenylsulfonyl)-3-(1...)
Affinity DataIC50:  44.9nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of normal bufferMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed