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BDBM50249106 15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide::CHEMBL475159

SMILES: CC1(CC2c3ccccc3C1c1ccccc21)C(=O)Nc1nccs1

InChI Key:

Data: 1 KI 3 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50249106
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glucocorticoid receptor (Human)	BDBM50249106 (15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	268	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glucocorticoid receptor (Human)	BDBM50249106 (15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	30.7	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glucocorticoid receptor (Human)	BDBM50249106 (15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glucocorticoid receptor (Human)	BDBM50249106 (15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{...) Show SMILES Show InChI	GoogleScholar	UniChem		2.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair