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BDBM50249193 (15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide::CHEMBL514646

SMILES: C[C@]1(CC2c3ccccc3C1c1ccccc21)C(=O)Nc1nccs1

InChI Key:

Data: 4 KI 1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50249193
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glucocorticoid receptor (Human)	BDBM50249193 ((15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	115	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glucocorticoid receptor (Human)	BDBM50249193 ((15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6...) Show SMILES Show InChI	GoogleScholar	UniChem		1.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Progesterone receptor (Human)	BDBM50249193 ((15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6...) Show SMILES Show InChI	GoogleScholar	UniChem		147	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Androgen receptor (Human)	BDBM50249193 ((15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6...) Show SMILES Show InChI	GoogleScholar	UniChem		7.40E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Estrogen receptor (Human)	BDBM50249193 ((15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6...) Show SMILES Show InChI	GoogleScholar	UniChem		1.50E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair