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BDBM50258497 (4-Quinolin-2-ylpiperazin-1-yl)acetic Acid::CHEMBL468498

SMILES: OC(=O)CN1CCN(CC1)c1ccc2ccccc2n1

InChI Key: InChIKey=HCRXUFYSLPXCDW-UHFFFAOYSA-N

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50258497
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 3A (Rat)	BDBM50258497 ((4-Quinolin-2-ylpiperazin-1-yl)acetic Acid \| CHEMB...) Show SMILES Show InChI	GoogleScholar	UniChem		11.2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
D(2) dopamine receptor (Rat)	BDBM50258497 ((4-Quinolin-2-ylpiperazin-1-yl)acetic Acid \| CHEMB...) Show SMILES Show InChI	GoogleScholar	UniChem		919	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 4 (Guinea pig)	BDBM50258497 ((4-Quinolin-2-ylpiperazin-1-yl)acetic Acid \| CHEMB...) Show SMILES Show InChI	GoogleScholar	UniChem		5.75E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 1A (Rat)	BDBM50258497 ((4-Quinolin-2-ylpiperazin-1-yl)acetic Acid \| CHEMB...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2A (Rat)	BDBM50258497 ((4-Quinolin-2-ylpiperazin-1-yl)acetic Acid \| CHEMB...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
D(1A) dopamine receptor (Rat)	BDBM50258497 ((4-Quinolin-2-ylpiperazin-1-yl)acetic Acid \| CHEMB...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair