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BDBM50283311 2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(2-pyridylcarbonylamino)-3H-quinazolin-4-one::CHEMBL74144

SMILES: CCc1nc2ccc(NC(=O)c3ccccn3)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)OCCC(C)C

InChI Key: InChIKey=ARHOSTGQGGKVFS-UHFFFAOYSA-N

Data: 6 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50283311   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Type-1 angiotensin II receptor


(Rabbit)
BDBM50283311
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
GoogleScholar
UniChem
n/an/a 2.30n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Type-1 angiotensin II receptor


(Human)
BDBM50283311
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
GoogleScholar
UniChem
n/an/a 85n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Type-2 angiotensin II receptor


(Rat)
BDBM50283311
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
GoogleScholar
UniChem
n/an/a 0.630n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Type-2 angiotensin II receptor


(Human)
BDBM50283311
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
GoogleScholar
UniChem
n/an/a 37n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Type-2 angiotensin II receptor


(Rat)
BDBM50283311
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
GoogleScholar
UniChem
n/an/a 1.80n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Type-1 angiotensin II receptor A/B


(Rat)
BDBM50283311
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
GoogleScholar
UniChem
n/an/a 1.30n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair