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BDBM50292603 2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carboxylate::CHEMBL481153

SMILES: O=C(OCCN1CCCC1)N1c2ccccc2Sc2ccccc12

InChI Key: InChIKey=CJGNMVAAMQAWEF-UHFFFAOYSA-N

Data: 4 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50292603
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histamine H1 receptor (Human)	BDBM50292603 (2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...) Show SMILES Show InChI	GoogleScholar	UniChem		29	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H2 receptor (Human)	BDBM50292603 (2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...) Show SMILES Show InChI	GoogleScholar	UniChem		540	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cholinesterase (Human)	BDBM50292603 (2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...) Show SMILES Show InChI	GoogleScholar	UniChem		650	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 3A (Human)	BDBM50292603 (2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...) Show SMILES Show InChI	GoogleScholar	UniChem		1.90E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair