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BDBM50304501 6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine::CHEMBL473662

SMILES: CN1CCN(CC1)c1cc(N)nc(N)n1

InChI Key: InChIKey=RBHNSRTVBDSNLG-UHFFFAOYSA-N

Data: 3 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50304501
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histamine H4 receptor (Human)	BDBM50304501 (6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine \|...) Show SMILES Show InChI	GoogleScholar	UniChem		290	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM50304501 (6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine \|...) Show SMILES Show InChI	GoogleScholar	UniChem		530	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM50304501 (6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine \|...) Show SMILES Show InChI	GoogleScholar	UniChem		1.08E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair