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BDBM50340902 (4-amino-2-(pyridin-3-ylamino)thiazol-5-yl)(2-fluorophenyl)methanone::CHEMBL1761791

SMILES: Nc1nc(Nc2cccnc2)sc1C(=O)c1ccccc1F

InChI Key: InChIKey=XHJMMMPXTUEBMQ-UHFFFAOYSA-N

Data: 3 IC50 1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50340902
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cyclin-dependent kinase 5 activator 1 (Human)	BDBM50340902 ((4-amino-2-(pyridin-3-ylamino)thiazol-5-yl)(2-fluo...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-dependent kinase 2 (Human)	BDBM50340902 ((4-amino-2-(pyridin-3-ylamino)thiazol-5-yl)(2-fluo...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glycogen synthase kinase-3 beta (Human)	BDBM50340902 ((4-amino-2-(pyridin-3-ylamino)thiazol-5-yl)(2-fluo...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	45	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Microtubule-associated protein tau (Rat)	BDBM50340902 ((4-amino-2-(pyridin-3-ylamino)thiazol-5-yl)(2-fluo...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	5.50E+3	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair