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BDBM50341540 3-(4-tert-Butylbenzoylamino)-5-(pyridin-4-yl)-(1H)-pyridin-2-one::CHEMBL1765770

SMILES: CC(C)(C)c1ccc(cc1)C(=O)Nc1cc(c[nH]c1=O)-c1ccncc1

InChI Key: InChIKey=GJYHDNFJPKFHRH-UHFFFAOYSA-N

Data: 4 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50341540
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Receptor-type tyrosine-protein kinase FLT3 (Human)	BDBM50341540 (3-(4-tert-Butylbenzoylamino)-5-(pyridin-4-yl)-(1H)...) Show SMILES Show InChI	GoogleScholar	UniChem		11	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mast/stem cell growth factor receptor Kit (Human)	BDBM50341540 (3-(4-tert-Butylbenzoylamino)-5-(pyridin-4-yl)-(1H)...) Show SMILES Show InChI	GoogleScholar	UniChem		27	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase ITK/TSK (Human)	BDBM50341540 (3-(4-tert-Butylbenzoylamino)-5-(pyridin-4-yl)-(1H)...) Show SMILES Show InChI	GoogleScholar	UniChem		120	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (Human)	BDBM50341540 (3-(4-tert-Butylbenzoylamino)-5-(pyridin-4-yl)-(1H)...) Show SMILES Show InChI	GoogleScholar	UniChem		1.32E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair