BDBM50373487 CHEMBL254589
SMILES CC[C@H](NC(C)=O)c1cc(Cl)ccc1C1CCN(CC1)C(=O)[C@@H]1CN(C[C@H]1c1ccc(Cl)cc1F)C(C)(C)C
InChI Key InChIKey=PWADIMGJQZHREF-GKRYNVPLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50373487
Affinity DataIC50: 1.49E+3nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Agonist activity at human MC3R expressed in CHO cells assessed as cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Agonist activity at human MC4R expressed in CHO cells assessed as cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Binding affinity to rat MC4RMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Binding affinity to human MC5RMore data for this Ligand-Target Pair
Affinity DataEC50: 372nMAssay Description:Agonist activity at human MC5R expressed in CHO cells assesses as cAMP releaseMore data for this Ligand-Target Pair