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BDBM50376057 CHEMBL259141::US10227357, Compound P-0541

SMILES: NC1CCN(CC1)c1ncnc2[nH]ccc12

InChI Key: InChIKey=SOYJTCRGELSHIV-UHFFFAOYSA-N

Data: 2 KI 2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50376057
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glycogen synthase kinase-3 beta (Human)	BDBM50376057 (CHEMBL259141 \| US10227357, Compound P-0541) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
RAC-beta serine/threonine-protein kinase (Human)	BDBM50376057 (CHEMBL259141 \| US10227357, Compound P-0541) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	180	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mast/stem cell growth factor receptor Kit [D816V] (Human)	BDBM50376057 (CHEMBL259141 \| US10227357, Compound P-0541) Show SMILES Show InChI	GoogleScholar	UniChem		5.50E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mast/stem cell growth factor receptor Kit (Human)	BDBM50376057 (CHEMBL259141 \| US10227357, Compound P-0541) Show SMILES Show InChI	GoogleScholar	UniChem		1.05E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair