BDBM50406762 CHEMBL37462
SMILES CN(C)CCc1c[nH]c2ccc(Cc3nc(N)ns3)cc12
InChI Key InChIKey=BEDGPDAVDXHRMR-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50406762
Affinity DataIC50: 2nMAssay Description:Compound was tested for the displacement of [3H]-5-HT to 5-hydroxytryptamine 1D receptor recognition sites in pig caudate membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of radioligand [3H]5-HT binding to 5-hydroxytryptamine 1D receptor in pig caudate membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of [3H]-Q-ICS 205-930 from rat cortex homogenate 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Displacement of [3H]mesulergine from pig cortex 5-hydroxytryptamine 1C receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:isplacement of [3H]DOB from rat cortex homogenate 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]8-OH-DPAT from pig cortex 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair