BDBM50423464 CHEMBL252231

SMILES CN1C[C@H](C[C@@H]2[C@@H]1Cc1c(Br)[nH]c3cccc2c13)C(=O)N1CCN(CC1)c1cccc(=O)n1C

InChI Key InChIKey=AWFDCTXCTHGORH-MDKPJZGXSA-N

Data  7 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50423464   

TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  8.13E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  9.33E+3nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  1.95E+3nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  5.37E+3nMAssay Description:Binding affinity to human recombinant sst3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  2.04E+4nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  6.92E+4nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(RAT)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  417nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed