BDBM5410 4-(2-(4-(3-phenylpyrazolo[1,5- a]pyrimidin-6-yl)phenoxy)ethyl)morpholine::4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phenoxy)ethyl]morpholine::US9040694, 4::pyrazolo[1,5-a]pyrimidine 4b

SMILES: C(CN1CCOCC1)Oc1ccc(cc1)-c1cnc2c(cnn2c1)-c1ccccc1

InChI Key: InChIKey=SKZQZGSPYYHTQG-UHFFFAOYSA-N

Data: 9 IC50  2 EC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 5410   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Vascular endothelial growth factor receptor 2 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	9	n/a	n/a	n/a	n/a	7.4	22
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Receptor protein serine/threonine kinase (Zebrafish)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a
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Receptor protein serine/threonine kinase (Zebrafish)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a
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Activin receptor type-1 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.56E+3	n/a	n/a	n/a	n/a	n/a	n/a
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5'-AMP-activated protein kinase subunit beta-1/5'-AMP-activated protein kinase subunit gamma-1/Dual specificity protein kinase CLK2 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8.04E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Vascular endothelial growth factor receptor 2 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	161	n/a	n/a	n/a	n/a	n/a	n/a
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Activin receptor type-1 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.57E+3	n/a	n/a	n/a	n/a	n/a	n/a
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5'-AMP-activated protein kinase subunit beta-1 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.92E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Vascular endothelial growth factor receptor 2 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	235	n/a	n/a	n/a	n/a	n/a	n/a
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Vascular endothelial growth factor receptor 2 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	9	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Human)	BDBM5410 (4-[2-(4-{3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}phe...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	32	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair