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BDBM81806 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-dihydro-1-(2-propenyl)-1h-indole mono(4-methylbenzenesulfonate)::WIN 53024::WIN 53782

SMILES: C=CCn1c(cc2ccccc12)C1=NCCN1

InChI Key: InChIKey=CUOQKQBYZYMBSP-UHFFFAOYSA-N

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 81806
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Alpha-2A adrenergic receptor (Human)	BDBM81806 (WIN 53782 \| 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...) Show SMILES Show InChI	GoogleScholar	UniChem		0.0500	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-2C adrenergic receptor (OK)	BDBM81806 (WIN 53782 \| 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...) Show SMILES Show InChI	GoogleScholar	UniChem		0.0500	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-2B adrenergic receptor (Rat)	BDBM81806 (WIN 53782 \| 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...) Show SMILES Show InChI	GoogleScholar	UniChem		0.270	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-2A adrenergic receptor (Human)	BDBM81806 (WIN 53782 \| 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...) Show SMILES Show InChI	GoogleScholar	UniChem		4.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-2C adrenergic receptor (OK)	BDBM81806 (WIN 53782 \| 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...) Show SMILES Show InChI	GoogleScholar	UniChem		18	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Alpha-2B adrenergic receptor (Rat)	BDBM81806 (WIN 53782 \| 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...) Show SMILES Show InChI	GoogleScholar	UniChem		67	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair