BindingDB PrimarySearch

BDBM82463 Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-amino*heptanoyl-L-Phe-)]::L-362,855::L-362855

SMILES: C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CCCCCCNC(=O)[C@H](Cc2ccccc2)NC1=O

InChI Key: InChIKey=CDHQUESZSCDTRS-UHFFFAOYSA-N

Data: 58 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 58 hits for monomerid = 82463
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Somatostatin receptor type 4 (Rat)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.00500	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Rat)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.0100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.670	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.670	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.670	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.760	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	0.790	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	1.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	2.04	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	2.04	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	2.96	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	4.36	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	4.36	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	4.37	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	5.12	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	5.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	5.62	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	6.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Rat)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	12	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	24.0	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	24.0	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	28.8	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	29	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	30.2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 3 (Rat)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	33	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	49.0	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	49.0	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Rat)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	51	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	63	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	63.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	67.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	67.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	67.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	67.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 5 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	67.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	83.2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 2 (Mouse)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	98	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 1 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	174	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	174	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Human)	BDBM82463 (L-362855 \| Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...) Show SMILES Show InChI	GoogleScholar	UniChem	467	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair

Displayed 1 to 50 (of 58 total ) | Next | Last >>