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BDBM82469 BIM 23003::BIM-23003::EC5-21::L-Cys(1)-L-Lys-L-Asn-4-Chloro-L-Phe-L-Phe-D-Trp-L-Lys-L-Thr-L-Phe-L-Thr-L-Ser-L-Cys(1)-OH
SMILES: C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(Cl)cc2)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)[C@@H](C)O)C(O)=O
InChI Key: InChIKey=YQLNLYWSBOYGSN-UHFFFAOYSA-N
Data: 8 KI
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Somatostatin receptor type 2 (Mouse) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 0.00500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 2 (Mouse) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 0.0100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 5 (Human) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 4 (Mouse) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 1.81 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 4 (Rat) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 3 (Mouse) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 2.08 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 3 (Mouse) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Somatostatin receptor type 5 (Human) | BDBM82469![]() (EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...) | GoogleScholar | UniChem | 560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||