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BDBM86493 CAS_27943::NALTREXONE-HCl::NSC_27943::Naltrexone

SMILES: Oc1ccc2CC3N(CC4CC4)CCC45C(Oc1c24)C(=O)CCC35O

InChI Key:

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 86493
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mu-type opioid receptor (Human)	BDBM86493 (CAS_27943 \| NALTREXONE-HCl \| NSC_27943 \| Naltrexon...) Show SMILES Show InChI	GoogleScholar	UniChem		0.300	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Human)	BDBM86493 (CAS_27943 \| NALTREXONE-HCl \| NSC_27943 \| Naltrexon...) Show SMILES Show InChI	GoogleScholar	UniChem		0.810	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mu-type opioid receptor (Human)	BDBM86493 (CAS_27943 \| NALTREXONE-HCl \| NSC_27943 \| Naltrexon...) Show SMILES Show InChI	GoogleScholar	UniChem		2.39	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Delta-type opioid receptor (Human)	BDBM86493 (CAS_27943 \| NALTREXONE-HCl \| NSC_27943 \| Naltrexon...) Show SMILES Show InChI	GoogleScholar	UniChem		16.3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Nociceptin receptor (Mouse)	BDBM86493 (CAS_27943 \| NALTREXONE-HCl \| NSC_27943 \| Naltrexon...) Show SMILES Show InChI	GoogleScholar	UniChem		1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Nociceptin receptor (Mouse)	BDBM86493 (CAS_27943 \| NALTREXONE-HCl \| NSC_27943 \| Naltrexon...) Show SMILES Show InChI	GoogleScholar	UniChem		1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair